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Optimization of 4-Amino-2-Pyridone Inhibitors of Proprotein Convertase Subtilisin/Kexin Type 9: Integrating Structure-Activity and Structure-Metabolism Relationships 4-氨基-2-吡啶酮前蛋白转化酶枯草杆菌/kreplin型9抑制剂的优化:整合构效关系和构代谢关系 Giannessi, Lisa; Lupo, Maria Giovanna; Ugolotti, Martina; Papotti, Bianca; Mattina, Beatrice; Martina, Maria Grazia; Demurtas, Anna; Padula, Cristina; Nicoli, Sara; Crescenzo, Marco; Ferri, Nicola; Zimetti, Francesca; Radi, Marco 分享 收藏
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Discovery of p-Trifluoromethylbenzohydrazide Derivatives as Potent Antiviral Agents against Monkeypox Virus Rossi, Sara; Pozzetti, Luca; Carullo, Gabriele; Dichiara, Maria; Butini, Stefania; Radi, Marco; Ramunno, Anna; Terrosi, Chiara; Barra, Giovanni; Berisio, Rita; Gemma, Sandra; Cusi, Maria Grazia; Campiani, Giuseppe 分享 收藏
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Identification of 4-amino-2-Pyridones as new potent PCSK9 inhibitors: From phenotypic hit discovery to in vivo tolerability Giannessi, Lisa; Lupo, Maria Giovanna; Rossi, Ilaria; Martina, Maria Grazia; Vilella, Antonietta; Bodria, Martina; Giuliani, Daniela; Zimetti, Francesca; Zanotti, Ilaria; Poti, Francesco; Bernini, Franco; Ferri, Nicola; Radi, Marco 分享 收藏
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4-Trifluoromethyl bithiazoles as broad-spectrum antimicrobial agents for virus-related bacterial infections or co-infections Barbieri, Francesca; Carlen, Vincent; Martina, Maria Grazia; Sannio, Filomena; Cancade, Sacha; Perini, Cecilia; Restori, Margherita; Crespan, Emmanuele; Maga, Giovanni; Docquier, Jean-Denis; Cagno, Valeria; Radi, Marco 分享 收藏
eHydrogenation: Hydrogen-free Electrochemical Hydrogenation Russo, Camilla; Leech, Matthew C.; Walsh, Jamie M.; Higham, Joe I.; Giannessi, Lisa; Lambert, Emmanuelle; Kiaku, Cyrille; Poole, Darren L.; Mason, Joseph; Goodall, Charles A. I.; Devo, Perry; Giustiniano, Mariateresa; Radi, Marco; Lam, Kevin 分享 收藏
Nucleoside Derivatives of 2,6-Diaminopurine Antivirals: Base-Modified Nucleosides with Broad-Spectrum Antimicrobial Properties 2,6-二氨基嘌呤抗病毒药物的核苷衍生物: 具有广谱抗菌特性的碱基修饰核苷 Martina, Maria Grazia; Giammarino, Federica; Vicenti, Ilaria; Groaz, Elisabetta; Rozenski, Jef; Incerti, Matteo; Sannio, Filomena; Docquier, Jean Denis; Zazzi, Maurizio; Radi, Marco 分享 收藏
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Discovery of small-molecules targeting the CCL20/CCR6 axis as first-in-class inhibitors for inflammatory bowel diseases Martina, Maria Grazia; Giorgio, Carmine; Allodi, Marika; Palese, Simone; Barocelli, Elisabetta; Ballabeni, Vigilio; Szpakowska, Martyna; Chevigne, Andy; van Hamburg, Jan Piet; Davelaar, Nadine; Lubberts, Erik; Bertoni, Simona; Radi, Marco 分享 收藏
Towards Innovative Antibacterial Correctors for Cystic Fibrosis Targeting the Lung Microbiome with a Multifunctional Effect Martina, Maria Grazia; Sannio, Filomena; Crespan, Emmanuele; Pavone, Marialaura; Simoncini, Alice; Barbieri, Francesca; Perini, Cecilia; Pesce, Emanuela; Maga, Giovanni; Pedemonte, Nicoletta; Docquier, Jean-Denis; Radi, Marco 分享 收藏
System-oriented optimization of multi-target 2,6-diaminopurine derivatives: Easily accessible broad-spectrum antivirals active against flaviviruses, influenza virus and SARS-CoV-2 多目标2,6-二氨基嘌呤衍生物的系统导向优化: 易于获得的对黄病毒,流感病毒和SARS-CoV-2具有活性的广谱抗病毒药物 Vicenti, Ilaria; Martina, Maria Grazia; Boccuto, Adele; De Angelis, Marta; Giavarini, Giorgia; Dragoni, Filippo; Marchi, Serena; Trombetta, Claudia Maria; Crespan, Emmanuele; Maga, Giovanni; Eydoux, Cecilia; Decroly, Etienne; Montomoli, Emanuele; Nencioni, Lucia; Zazzi, Maurizio; Radi, Marco 分享 收藏
Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIIIβ) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human Rhinoviruses 磷脂酰肌醇4-激酶 (PI4KIIIβ) 的双噻唑抑制剂作为广谱抗病毒药物阻断SARS-CoV-2,寨卡病毒和人类鼻病毒的复制 Grazia Martina, Maria; Vicenti, Ilaria; Bauer, Lisa; Crespan, Emmanuele; Rango, Enrico; Boccuto, Adele; Olivieri, Noemi; Incerti, Matteo; Zwaagstra, Marleen; Allodi, Marika; Bertoni, Simona; Dreassi, Elena; Zazzi, Maurizio; van Kuppeveld, Frank J. M.; Maga, Giovanni; Radi, Marco 分享 收藏
Multitarget CFTR Modulators Endowed with Multiple Beneficial Side Effects for Cystic Fibrosis Patients: Toward a Simplified Therapeutic Approach Tassini, Sabrina; Langron, Emily; Delang, Leen; Mirabelli, Carmen; Lanko, Kristina; Crespan, Emmanuele; Kissova, Miroslava; Tagliavini, Giulia; Fonto, Greta; Bertoni, Simona; Palese, Simone; Giorgio, Carmine; Ravanetti, Francesca; Ragionieri, Luisa; Zamperini, Claudio; Mancini, Arianna; Dreassi, Elena; Maga, Giovanni; Vergani, Paola; Neyts, Johan; Radi, Marco 分享 收藏
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