Frédéric Rodriguez - Publications, H-index & Citations

Frédéric Rodriguez

université toulouse iii – paul sabatier (ut3)

20H指数

87论文数

1.1K被引数

收录论文 26

发表时间

Is Mycobacterial InhA a Suitable Target for Rational Drug Design?分枝杆菌 InhA 是否是合理药物设计的合适靶点？

CHEMMEDCHEM

IF3.4

2025-04-29

PREAI

Julien Rizet; Laurent Maveyraud; David Rengel; Valérie Guillet; Gabriel Publicola; Frédéric Rodriguez; Christian Lherbet; Lionel Mourey

Imidazoquinoline Derivatives as Potential Inhibitors of InhA Enzyme and Mycobacterium tuberculosis

MOLECULES

IF4.6

2024-06-27

OAAI

Hoffmann, Pascal; Azema-Despeyroux, Joelle; Goncalves, Fernanda; Stamilla, Alessandro; Saffon-Merceron, Nathalie; Rodriguez, Frederic; Degiacomi, Giulia; Pasca, Maria Rosalia; Lherbet, Christian

Discovery of new diaryl ether inhibitors against Mycobacterium tuberculosis targeting the minor portal of InhA

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2023-11-01

OAAI

Chebaiki, Melina; Delfourne, Evelyne; Tamhaev, Rasoul; Danoun, Saida; Rodriguez, Frederic; Hoffmann, Pascal; Grosjean, Emeline; Goncalves, Fernanda; Azema-Despeyroux, Joelle; Pal, Adrian; Kordulakova, Jana; Preuilh, Nadege; Britton, Sebastien; Constant, Patricia; Marrakchi, Hedia; Maveyraud, Laurent; Mourey, Lionel; Lherbet, Christian

Phenyl dialkynylcarbinols, a Bioinspired Series of Synthetic Antitumor Acetylenic Lipids

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2023-10-10

OAAI

Bossuat, Margaux; Rulliere, Pauline; Preuilh, Nadege; Peixoto, Antonio; Joly, Etienne; Gomez, Jean-Guillaume; Bourkhis, Maroua; Rodriguez, Frederic; Goncalves, Fernanda; Fabing, Isabelle; Gaspard, Hafida; Bernardes-Genisson, Vania; Maraval, Valerie; Ballereau, Stephanie; Chauvin, Remi; Britton, Sebastien; Genisson, Yves

Isolation and identification of ten new sildenafil derivatives in an alleged herbal supplement for sexual enhancement

JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS

IF3.1

2020-11-01

OAAI

Assemat, Gaetan; Balayssac, Stephane; Gilard, Veronique; Martins-Froment, Nathalie; Fabing, Isabelle; Rodriguez, Frederic; Genisson, Yves; Martino, Robert; Malet-Martino, Myriam

Modification of endothelial nitric oxide synthase by 4-oxo-2(E)-nonenal (ONE) in preeclamptic placentas

FREE RADICAL BIOLOGY AND MEDICINE

IF8.2

2019-09-01

OAAI

Guerby, Paul; Swiader, Audrey; Tasta, Oriane; Pont, Frederic; Rodriguez, Frederic; Parant, Olivier; Vayssiere, Christophe; Shibata, Takahiro; Uchida, Koji; Salvayre, Robert; Negre-Salvayre, Anne

Selective Targeting of the Interconversion between Glucosylceramide and Ceramide by Scaffold Tailoring of Iminosugar Inhibitors

MOLECULES

IF4.6

2019-01-19

OAAI

Baudoin-Dehoux, Cecile; Castellan, Tessa; Rodriguez, Frederic; Rives, Arnaud; Stauffert, Fabien; Garcia, Virginie; Levade, Thierry; Compain, Philippe; Genisson, Yves

Iminosugar-based ceramide mimicry for the design of new CERT START domain ligands

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2017-03-01

PREAI

Santos, Cecile; Stauffert, Fabien; Ballereau, Stephanie; Dehoux, Cecile; Rodriguez, Frederic; Bodlenner, Anne; Compain, Philippe; Genisson, Yves

Pyrrolidinone and pyrrolidine derivatives: Evaluation as inhibitors of InhA and Mycobacterium tuberculosis 吡咯烷酮和吡咯烷衍生物: 作为InhA和结核分枝杆菌抑制剂的评估

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2016-11-01

PREAI

Matviiuk, Tetiana; Madacki, Jan; Mori, Giorgia; Orena, Beatrice Silvia; Menendez, Christophe; Kysil, Andrii; Andre-Barres, Christiane; Rodriguez, Frederic; Kordulakova, Jana; Mallet-Ladeira, Sonia; Voitenko, Zoia; Pasca, Maria Rosalia; Lherbet, Christian; Baltas, Michel

Asymmetric Synthesis and Binding Study of New Long-Chain HPA-12 Analogues as Potent Ligands of the Ceramide Transfer Protein CERT

CHEMISTRY-A EUROPEAN JOURNAL

IF3.7

2016-03-31

OAAI

Duris, Andrej; Daich, Adam; Santos, Cecile; Fleury, Laurence; Ausseil, Frederic; Rodriguez, Frederic; Ballereau, Stephanie; Genisson, Yves; Berkes, Dusan

Hemisynthesis, Antitumoral Effect, and Molecular Docking Studies of Ferutinin and Its Analogues

CHEMICAL BIOLOGY & DRUG DESIGN

IF3.3

2015-11-05

PREAI

Safi, Remi; Rodriguez, Frederic; Hilal, Georges; Diab-Assaf, Mona; Diab, Youssef; El-Sabban, Marwan; Najjar, Fadia; Delfourne, Evelyne

Design, synthesis and evaluation of new GEQ derivatives as inhibitors of InhA enzyme and Mycobacterium tuberculosis growth

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2015-08-01

OAAI

Chollet, Aurelien; Mori, Giorgia; Menendez, Christophe; Rodriguez, Frederic; Fabing, Isabelle; Pasca, Maria Rosalia; Madacki, Jan; Kordulakova, Jana; Constant, Patricia; Quemard, Annaik; Bernardes-Genisson, Vania; Lherbet, Christian; Baltas, Michel

The CERT antagonist HPA-12: First practical synthesis and individual binding evaluation of the four stereoisomers

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2015-05-01

PREAI

Santos, Cecile; Fleury, Laurence; Rodriguez, Frederic; Markus, Jozef; Berkes, Dusan; Daich, Adam; Ausseil, Frederic; Baudoin-Dehoux, Cecile; Ballereau, Stephanie; Genisson, Yves

Synthesis and In Vitro Antiproliferative Activity of Amido and Amino Analogues of the Marine Alkaloid Isogranulatimide

CHEMMEDCHEM

IF3.4

2015-03-03

PREAI

Lavrard, Hubert; Salvetti, Beatrice; Mathieu, Veronique; Rodriguez, Frederic; Kiss, Robert; Delfourne, Evelyne

Design of granulatimide and isogranulatimide analogues as potential Chk1 inhibitors: Study of amino-platforms for their synthesis

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2014-09-01

PREAI

Lavrard, Hubert; Rodriguez, Frederic; Delfourne, Evelyne

Synthesis of 3-heteryl substituted pyrrolidine-2,5-diones via catalytic Michael reaction and evaluation of their inhibitory activity against InhA and Mycobacterium tuberculosis

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2014-01-01

PREAI

Matviiuk, Tetiana; Mori, Giorgia; Lherbet, Christian; Rodriguez, Frederic; Pasca, Maria Rosalia; Gorichko, Marian; Guidetti, Brigitte; Voitenko, Zoia; Baltas, Michel

Design, chemical synthesis of 3-(9H-fluoren-9-yl)pyrrolidine-2,5-dione derivatives and biological activity against enoyl-ACP reductase (InhA) and Mycobacterium tuberculosis

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2013-12-01

PREAI

Matviiuk, Tetiana; Rodriguez, Frederic; Saffon, Nathalie; Mallet-Ladeira, Sonia; Gorichko, Marian; Ribeiro, Ana Luisa de Jesus Lopes; Pasca, Maria Rosalia; Lherbet, Christian; Voitenko, Zoia; Baltas, Michel

Synthesis and evaluation of α-ketotriazoles and α,β-diketotriazOles as inhibitors of Mycobacterium tuberculosis

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2013-11-01

PREAI

Menendez, Christophe; Rodriguez, Frederic; Ribeiro, Ana Luisa de Jesus Lopes; Zara, Francesca; Frongia, Celine; Lobjois, Valerie; Saffon, Nathalie; Pasca, Maria Rosalia; Lherbet, Christian; Baltas, Michel

Chemical synthesis and biological evaluation of triazole derivatives as inhibitors of InhA and antituberculosis agents

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2012-06-01

PREAI

Menendez, Christophe; Chollet, Aurelien; Rodriguez, Frederic; Inard, Cyril; Pasca, Maria Rosalia; Lherbet, Christian; Baltas, Michel

In vitro toxicological effects of estrogenic mycotoxins on human placental cells: Structure activity relationships

TOXICOLOGY AND APPLIED PHARMACOLOGY

IF3.4

2012-03-01

PREAI

Prouillac, Caroline; Koraichi, Farah; Videmann, Bernadette; Mazallon, Michelle; Rodriguez, Frederic; Baltas, Michel; Lecoeur, Sylvaine

研究方向