未登录 Characterization of 2,4-Dianilinopyrimidines Against Five P. falciparum Kinases PfARK1, PfARK3, PfNEK3, PfPK9, and PfPKB Ong, Han Wee; de Silva, Chandi; Avalani, Krisha; Kwarcinski, Frank; Mansfield, Christopher R.; Chirgwin, Michael; Truong, Anna; Derbyshire, Emily R.; Zutshi, Reena; Drewry, David H. 分享 收藏
Discovery of potent Plasmodium falciparum protein kinase 6 (PfPK6) inhibitors with a type II inhibitor pharmacophore Ong, Han Wee; Truong, Anna; Kwarcinski, Frank; de Silva, Chandi; Avalani, Krisha; Havener, Tammy M.; Chirgwin, Michael; Galal, Kareem A.; Willis, Caleb; Kramer, Andreas; Liu, Shubin; Knapp, Stefan; Derbyshire, Emily R.; Zutshi, Reena; Drewry, David H. 分享 收藏
Identification of Novel 2,4,5-Trisubstituted Pyrimidines as Potent Dual Inhibitors of Plasmodial PfGSK3/PfPK6 with Activity against Blood Stage Parasites In Vitro Galal, Kareem A.; Truong, Anna; Kwarcinski, Frank; de Silva, Chandi; Avalani, Krisha; Havener, Tammy M.; Chirgwin, Michael E.; Merten, Eric; Ong, Han Wee; Willis, Caleb; Abdelwaly, Ahmad; Helal, Mohamed A.; Derbyshire, Emily R.; Zutshi, Reena; Drewry, David H. 分享 收藏
Identification of 4-Anilinoquin(az)oline as a Cell-Active Protein Kinase Novel 3 (PKN3) Inhibitor Chemotype Asquith, Christopher R. M.; Temme, Louisa; East, Michael P.; Laitinen, Tuomo; Pickett, Julie; Kwarcinski, Frank E.; Sinha, Parvathi; Wells, Carrow, I; Johnson, Gary L.; Zutshi, Reena; Drewry, David H. 分享 收藏
A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation Picado, Alfredo; Chaikuad, Apirat; Wells, Carrow, I; Shrestha, Safal; Zuercher, William J.; Pickett, Julie E.; Kwarcinski, Frank E.; Sinha, Parvathi; de Silva, Chandi S.; Zutshi, Reena; Liu, Shubin; Kannan, Natarajan; Knapp, Stefan; Drewry, David H.; Willson, Timothy M. 分享 收藏
SGC-AAK1-1: A Chemical Probe Targeting AAK1 and BMP2K Wells, Carrow; Counago, Rafael M.; Limas, Juanita C.; Almeida, Tuanny L.; Cook, Jeanette Gowen; Drewry, David H.; Elkins, Jonathan M.; Gileadi, Opher; Kapadia, Nirav R.; Lorente-Macias, Alvaro; Pickett, Julie E.; Riemen, Alexander; Ruela-de-Sousa, Roberta R.; Willson, Timothy M.; Zhang, Cunyu; Zuercher, William J.; Zutshi, Reena; Axtman, Alison D. 分享 收藏
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