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Flexibility-tuning of dual-display DNA-encoded chemical libraries facilitates cyclic peptide ligand discovery 双显示DNA编码化合物库的灵活性调控有助于环肽配体的发现 Petrov, Dimitar; Plais, Louise; Schira, Kristina; Cai, Junyu; Keller, Michelle; Lessing, Alice; Bassi, Gabriele; Cazzamalli, Samuele; Neri, Dario; Gloger, Andreas; Scheuermann, Jorg 分享 收藏
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Computational methods to analyze and predict the binding mode of inhibitors targeting both human and mushroom tyrosinase Ricci, Federico; Schira, Kristina; Khettabi, Lyna; Lombardo, Lisa; Mirabile, Salvatore; Gitto, Rosaria; Soler-Lopez, Montserrat; Scheuermann, Joerg; Wolber, Gerhard; De Luca, Laura 分享 收藏
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A DNA-encoded chemical library based on chiral 4-amino-proline enables stereospecific isozyme-selective protein recognition Oehler, Sebastian; Lucaroni, Laura; Migliorini, Francesca; Elsayed, Abdullah; Prati, Luca; Puglioli, Sara; Matasci, Mattia; Schira, Kristina; Scheuermann, Jorg; Yudin, Denis; Jia, Min; Ban, Nenad; Bushnell, Dave; Kornberg, Roger; Cazzamalli, Samuele; Neri, Dario; Favalli, Nicholas; Bassi, Gabriele 分享 收藏
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Selective tumor targeting enabled by picomolar fibroblast activation protein inhibitors isolated from a DNA-encoded affinity maturation library Puglioli, Sara; Schmidt, Eleonore; Pellegrino, Christian; Prati, Luca; Oehler, Sebastian; De Luca, Roberto; Galbiati, Andrea; Comacchio, Claudia; Nadal, Lisa; Scheuermann, Jorg; Manz, Markus G.; Neri, Dari; Cazzamalli, Samuele; Bassi, Gabriele; Favalli, Nicholas 分享 收藏
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Isolation of a Natural Killer Group 2D Small-Molecule Ligand from DNA-Encoded Chemical Libraries Dakhel, Sheila; Galbiati, Andrea; Migliorini, Francesca; Comacchio, Claudia; Oehler, Sebastian; Prati, Luca; Scheuermann, Joerg; Cazzamalli, Samuele; Neri, Dario; Bassi, Gabriele; Favalli, Nicholas 分享 收藏
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Affinity Selections of DNA-Encoded Chemical Libraries on Carbonic Anhydrase IX-Expressing Tumor Cells Reveal a Dependence on Ligand Valence Oehler, Sebastian; Catalano, Marco; Scapozza, Ilario; Bigatti, Martina; Bassi, Gabriele; Favalli, Nicholas; Mortensen, Michael R.; Samain, Florent; Scheuermann, Jorg; Neri, Dario 分享 收藏
Stereo- and regiodefined DNA-encoded chemical libraries enable efficient tumour-targeting applications Favalli, Nicholas; Bassi, Gabriele; Pellegrino, Christian; Millul, Jacopo; De Luca, Roberto; Cazzamalli, Samuele; Yang, Su; Trenner, Anika; Mozaffari, Nour L.; Myburgh, Renier; Moroglu, Mustafa; Conway, Stuart J.; Sartori, Alessandro A.; Manz, Markus G.; Lerner, Richard A.; Vogt, Peter K.; Scheuermann, Jorg; Neri, Dario 分享 收藏