未登录
分享
收藏
分享
收藏
分享
收藏
分享
收藏High ligand efficiency quinazoline compounds as novel A2A adenosine receptor antagonists高配体效率喹唑啉类化合物作为新型A2A腺苷受体拮抗剂
Bolteau, Raphael; Duroux, Romain; Laversin, Amelie; Vreulz, Brandon; Shiriaeva, Anna; Stauch, Benjamin; Han, Gye Won; Cherezov, Vadim; Renault, Nicolas; Barczyk, Amelie; Ravez, Severine; Coevoet, Mathilde; Melnyk, Patricia; Liberelle, Maxime; Yous, Said
分享
收藏GPCR Agonist-to-Antagonist Conversion: Enabling the Design of Nucleoside Functional Switches for the A2A Adenosine Receptor
Shiriaeva, Anna; Park, Daejin; Kim, Gyudong; Lee, Yoonji; Hou, Xiyan; Jarhad, Dnyandev B.; Kim, Gibae; Yu, Jinha; Hyun, Young Eum; Kim, Woomi; Gao, Zhan-Guo; Jacobson, Kenneth A.; Han, Gye Won; Stevens, Raymond C.; Jeong, Lak Shin; Choi, Sun; Cherezov, Vadim
分享
收藏
分享
收藏Molecular basis for lipid recognition by the prostaglandin D2 receptor CRTH2
Liu, Heng; Deepak, R. N. V. Krishna; Shiriaeva, Anna; Gati, Cornelius; Batyuk, Alexander; Hu, Hao; Weierstall, Uwe; Liu, Wei; Wang, Lei; Cherezov, Vadim; Fan, Hao; Zhang, Cheng
分享
收藏Structure-based mechanism of cysteinyl leukotriene receptor inhibition by antiasthmatic drugs
Luginina, Aleksandra; Gusach, Anastasiia; Marin, Egor; Mishin, Alexey; Brouillette, Rebecca; Popov, Petr; Shiriaeva, Anna; Besserer-Offroy, Elie; Longpre, Jean-Michel; Lyapina, Elizaveta; Ishchenko, Andrii; Patel, Nilkanth; Polovinkin, Vitaly; Safronova, Nadezhda; Bogorodskiy, Andrey; Edelweiss, Evelina; Hu, Hao; Weierstall, Uwe; Liu, Wei; Batyuk, Alexander; Gordeliy, Valentin; Han, Gye Won; Sarret, Philippe; Katritch, Vsevolod; Borshchevskiy, Valentin; Cherezov, Vadim
分享
收藏