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Michael J. Roy

Adelaide University

14H指数
46论文数
1.6K被引数
收录论文 19
发表时间
DesignMaster: A Multi-Conditional Diffusion Framework for Rational PROTAC DesignDesignMaster:一种用于理性PROTAC设计的多条件扩散框架
err2026-09-24
err0
errOAAI
errBinze Shi; Yi Hao; Jie Liu; Tong Pan; Luke Isbel; Michael Roy; Ashley P Ng; Xuequn Shang; Fuyi Li; null; null
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Expanding the toolbox to develop IAP-based degraders of TEAD transcription factors
err2026-01-19
err0
errOAAI
errNishma Gupta; Nicole Trainor; Mona Radwan; Stephanie Nguyen; Luke Duncan; Andrew X. Tang; Julia Beveridge; Natasha Silke; Jumana Yousef; Ceren Bilgilier; Johannes Wachter; Peter Greb; Zuzana Jandova; Ján Eliaš; Sara Kopf; Thomas Gerstberger; Peggy Stolt-Bergner; Nina Braun; Harald Weinstabl; Darryl B. McConnell; Federico Mauri; Isabelle S. Lucet; John Silke; Nicola E. A. Chessum; Michael J. Roy
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Sequence differences between BAX and BAK core domains manifest as differences in their interactions with lipids
err2024-01-19
err4
PREAI
errMiller, Michelle S.; Cowan, Angus D.; Brouwer, Jason M.; Smyth, Sean T.; Peng, Liuyu; Wardak, Ahmad Z.; Uren, Rachel T.; Luo, Cindy; Roy, Michael J.; Shah, Sayali; Tan, Ziwen; Reid, Gavin E.; Colman, Peter M.; Czabotar, Peter E.
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Structural mapping of PEAK pseudokinase interactions identifies 14-3-3 as a molecular switch for PEAK3 signaling
err2023-06-19
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errOAAI
errRoy, Michael J.; Surudoi, Minglyanna G.; Kropp, Ashleigh; Hou, Jianmei; Dai, Weiwen; Hardy, Joshua M.; Liang, Lung-Yu; Cotton, Thomas R.; Lechtenberg, Bernhard C.; Dite, Toby A.; Ma, Xiuquan; Daly, Roger J.; Patel, Onisha; Lucet, Isabelle S.
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A selective and orally bioavailable VHL-recruiting PROTAC achieves SMARCA2 degradation in vivo
err2022-10-10
err99
errOAAI
errKofink, Christiane; Trainor, Nicole; Mair, Barbara; Woehrle, Simon; Wurm, Melanie; Mischerikow, Nikolai; Roy, Michael J.; Bader, Gerd; Greb, Peter; Garavel, Geraldine; Diers, Emelyne; McLennan, Ross; Whitworth, Claire; Vetma, Vesna; Rumpel, Klaus; Scharnweber, Maximilian; Fuchs, Julian E.; Gerstberger, Thomas; Cui, Yunhai; Gremel, Gabriela; Chetta, Paolo; Hopf, Stefan; Budano, Nicole; Rinnenthal, Joerg; Gmaschitz, Gerhard; Mayer, Moriz; Koegl, Manfred; Ciulli, Alessio; Weinstabl, Harald; Farnaby, William
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Distinct PEAK3 interactors and outputs expand the signaling potential of the PEAK pseudokinase family不同的PEAK3相互作用物和输出扩大了峰值假激酶家族的信号传导潜力
err2022-02-22
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PREAI
errHou, Jianmei; Nguyen, Elizabeth, V; Surudoi, Minglyanna; Roy, Michael J.; Patel, Onisha; Lucet, Isabelle S.; Ma, Xiuquan; Daly, Roger J.
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Structural basis for small molecule targeting of Doublecortin Like Kinase 1 with DCLK1-IN-1
err2021-09-20
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errOAAI
errPatel, Onisha; Roy, Michael J.; Kropp, Ashleigh; Hardy, Joshua M.; Dai, Weiwen; Lucet, Isabelle S.
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The intracellular domains of the EphB6 and EphA10 receptor tyrosine pseudokinases function as dynamic signalling hubs
err2021-09-14
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errOAAI
errLiang, Lung-Yu; Roy, Michael; Horne, Christopher R.; Sandow, Jarrod J.; Surudoi, Minglyanna; Dagley, Laura F.; Young, Samuel N.; Dite, Toby; Babon, Jeffrey J.; Janes, Peter W.; Patel, Onisha; Murphy, James M.; Lucet, Isabelle S.
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Synthesis of C-Mannosylated Glycopeptides Enabled by Ni-Catalyzed Photoreductive Cross-Coupling Reactions
err2021-08-04
err55
PREAI
errMao, Runyu; Xi, Shiyi; Shah, Sayali; Roy, Michael J.; John, Alan; Lingford, James P.; Gade, Gerd; Scott, Nichollas E.; Goddard-Borger, Ethan D.
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Structure-Guided Development of Potent Benzoylurea Inhibitors of BCL-XL and BCL-2
err2021-04-27
err8
PREAI
errRoy, Michael J.; Vom, Amelia; Okamoto, Toru; Smith, Brian J.; Birkinshaw, Richard W.; Yang, Hong; Abdo, Houda; White, Christine A.; Segal, David; Huang, David C. S.; Baell, Jonathan B.; Colman, Peter M.; Czabotar, Peter E.; Lessene, Guillaume
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BAK core dimers bind lipids and can be bridged by them
err2020-09-14
err50
PREAI
errCowan, Angus D.; Smith, Nicholas A.; Sandow, Jarrod J.; Kapp, Eugene A.; Rustam, Yepy H.; Murphy, James M.; Brouwer, Jason M.; Bernardini, Jonathan P.; Roy, Michael J.; Wardak, Ahmad Z.; Tan, Iris K.; Webb, Andrew I.; Gulbis, Jacqueline M.; Smith, Brian J.; Reid, Gavin E.; Dewson, Grant; Colman, Peter M.; Czabotar, Peter E.
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The PEAK family of pseudokinases, their role in cell signalling and cancer
err2019-11-06
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errOAAI
errPatel, Onisha; Roy, Michael J.; Murphy, James M.; Lucet, Isabelle S.
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BAF complex vulnerabilities in cancer demonstrated via structure-based PROTAC design (vol 15, pg 672, 2019)
err2019-07-02
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errOAAI
errFarnaby, William; Koegl, Manfred; Roy, Michael J.; Whitworth, Claire; Diers, Emelyne; Trainor, Nicole; Zollman, David; Steurer, Steffen; Karolyi-Oezguer, Jale; Riedmueller, Carina; Gmaschitz, Teresa; Wachter, Johannes; Dank, Christian; Galant, Michael; Sharps, Bernadette; Rumpel, Klaus; Traxler, Elisabeth; Gerstberger, Thomas; Schnitzer, Renate; Petermann, Oliver; Greb, Peter; Weinstabl, Harald; Bader, Gerd; Zoephel, Andreas; Weiss-Puxbaum, Alexander; Ehrenhofer-Wolfer, Katharina; Wohrle, Simon; Boehmelt, Guido; Rinnenthal, Joerg; Arnhof, Heribert; Wiechens, Nicola; Wu, Meng-Ying; Owen-Hughes, Tom; Ettmayer, Peter; Pearson, Mark; McConnell, Darryl B.; Ciulli, Alessio
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BAF complex vulnerabilities in cancer demonstrated via structure-based PROTAC design
err2019-06-10
err381
errOAAI
errFarnaby, William; Koegl, Manfred; Roy, Michael J.; Whitworth, Claire; Diers, Emelyne; Trainor, Nicole; Zollman, David; Steurer, Steffen; Karolyi-Oezguer, Jale; Riedmueller, Carina; Gmaschitz, Teresa; Wachter, Johannes; Dank, Christian; Galante, Michael; Sharps, Bernadette; Rumpel, Klaus; Traxler, Elisabeth; Gerstberger, Thomas; Schnitzer, Renate; Petermann, Oliver; Grebe, Peter; Weinstabl, Harald; Bader, Gerd; Zoephel, Andreas; Weiss-Puxbaum, Alexander; Ehrenhoefer-Woelfer, Katharina; Woehrle, Simon; Boehmelt, Guido; Rinnenthal, Joerg; Arnhof, Heribert; Wiechens, Nicola; Wu, Meng-Ying; Owen-Hughes, Tom; Ettmayer, Peter; Pearson, Mark; McConnell, Darryl B.; Ciulli, Alessio
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SPR-Measured Dissociation Kinetics of PROTAC Ternary Complexes Influence Target Degradation Rate
err2019-02-05
err237
errOAAI
errRoy, Michael J.; Winkler, Sandra; Hughes, Scott J.; Whitworth, Claire; Galant, Michael; Farnaby, William; Rumpel, Klaus; Ciulli, Alessio
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De-Novo Designed Library of Benzoylureas as Inhibitors of BCL-XL: Synthesis, Structural and Biochemical Characterization
err2014-02-05
err35
PREAI
errBrady, Ryan M.; Vom, Amelia; Roy, Michael J.; Toovey, Nathan; Smith, Brian J.; Moss, Rebecca M.; Hatzis, Effie; Huang, David C. S.; Parisot, John P.; Yang, Hong; Street, Ian P.; Colman, Peter M.; Czabotar, Peter E.; Baell, Jonathan B.; Lessene, Guillaume
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