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Comprehensive overview of biased pharmacology at the opioid receptors: biased ligands and bias factorsRSC MEDICINAL CHEMISTRYIF3.62021-01-0129OA
Neuromedin U and Structural Analogs: An Overview of their Structure, Function and SelectivityCURRENT MEDICINAL CHEMISTRYIF3.52020-11-247OA
Structure-Based Design of Melanocortin 4 Receptor Ligands Based on the SHU-9119-hMC4R Cocrystal StructureJOURNAL OF MEDICINAL CHEMISTRYIF6.82020-11-1413PREAI
Optimized Opioid-Neurotensin Multitarget Peptides: From Design to Structure-Activity Relationship StudiesJOURNAL OF MEDICINAL CHEMISTRYIF6.82020-09-0923OAAI
Neurotensin Analogues Containing Cyclic Surrogates of Tyrosine at Position 11 Improve NTS2 Selectivity Leading to Analgesia without Hypotension and HypothermiaACS CHEMICAL NEUROSCIENCEIF3.92019-10-0724OAAI
Synthesis and in Vitro Evaluation of Stabilized and Selective Neuromedin U-1 Receptor AgonistsACS MEDICINAL CHEMISTRY LETTERSIF42018-04-2310OAAI
Development of potent and proteolytically stable human neuromedin U receptor agonistsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92018-01-0116OAAI
χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone ScaffoldsACS MEDICINAL CHEMISTRY LETTERSIF42017-10-098OA
Analgesic Properties of Opioid/NK1 Multitarget Ligands with Distinct in Vitro Profiles in Naive and Chronic Constriction Injury MiceACS CHEMICAL NEUROSCIENCEIF3.92017-07-2632OAAI
Hydrazone Linker as a Useful Tool for Preparing Chimeric Peptide/Nonpeptide Bifunctional CompoundsACS MEDICINAL CHEMISTRY LETTERSIF42016-11-0829OAAI
Side Chain Cyclized Aromatic Amino Acids: Great Tools as Local Constraints in Peptide and Peptidomimetic DesignJOURNAL OF MEDICINAL CHEMISTRYIF6.82016-10-1235PREAI
Bifunctional Peptide-Based Opioid Agonist Nociceptin Antagonist Ligands for Dual Treatment of Acute and Neuropathic PainJOURNAL OF MEDICINAL CHEMISTRYIF6.82016-04-1441OAAI
Dual Alleviation of Acute and Neuropathic Pain by Fused Opioid Agonist-Neurokinin 1 Antagonist PeptidomimeticsACS MEDICINAL CHEMISTRY LETTERSIF42015-11-0322OAAI
T3P-Promoted, Mild, One-Pot Syntheses of Constrained Polycyclic Lactam Dipeptide Analogues via Stereoselective Pictet-Spengler and Meyers Lactamization ReactionsORGANIC LETTERSIF52015-08-3115PREAI
Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist - Neurokinin-1 antagonist peptidomimeticsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92015-03-0133OAAI
Structural basis for bifunctional peptide recognition at human δ-opioid receptorNATURE STRUCTURAL & MOLECULAR BIOLOGYIF10.12015-02-16168OAAI
Azepinone-Containing Tetrapeptide Analogues of Melanotropin Lead to Selective hMC4R Agonists and hMC5R AntagonistACS MEDICINAL CHEMISTRY LETTERSIF42014-12-0511OAAI
Synthesis of Fused 3-Aminoazepinones via Trapping of a New Class of Cyclic Seven-Membered Allenamides with FuranORGANIC LETTERSIF52014-07-0919PREAI
In Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt1-DALDA AnaloguesACS MEDICINAL CHEMISTRY LETTERSIF42014-02-0614OA
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