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Santina Bruzzone

Università degli Studi di Genova

52H指数
217论文数
7.9K被引数
收录论文 110
发表时间
Design, Synthesis, and Biological Evaluation of Pyrazolyl Thioureas (PTUs) as SIRT1 and SIRT2 Inhibitors吡唑硫脲(PTUs)的设计、合成及其作为SIRT1和SIRT2抑制剂的生物评价
err2026-09-25
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errMatteo Lusardi; Cecilia Astigiano; Deianira Bellitto; Matteo Raineri; Giorgia Guccione; Annalisa Salis; Elena Cichero; Chiara Brullo; Marco Ponassi; Santina Bruzzone; Andrea Spallarossa
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Probing pyrazolo-pyrimidines as SIRT2 inhibitors via molecular modelling and biological assays通过分子建模和生物实验研究吡唑嘧啶类化合物作为SIRT2抑制剂的探针
err2026-08-19
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PREAI
errFrancesca Musumeci; Cecilia Astigiano; Naomi Scarano; Marta Falesiedi; Giorgia Guccione; Jade Calamano; Annalisa Salis; Caterina Miro; Chiara Brullo; Monica Dentice; Elena Cichero Corresponding Author; Santina Bruzzone; Silvia Schenone
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The pivotal role of endoplasmic reticulum in cancer glucose metabolism内质网在癌症糖代谢中的关键作用
err2025-12-19
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errCecilia Marini; Maddalena Ghelardoni; Sonia Carta; Tiziana Bachetti; Silvia Bruno; Isotta Cainero; Silvia Ravera; Roberto Benelli; Marco Scotto; Francesca Vitale; Santina Bruzzone; Serena Losacco; Sabrina Chiesa; Matteo Bauckneht; Gabriele Tancreda; Matteo Raineri; Anna Maria Orengo; Andrea Benzi; Gianmario Sambuceti
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Membrane IL-18 identifies a human macrophage subset with distinct proteomic and functional traits膜IL-18识别具有独特蛋白质组学和功能特征的人类巨噬细胞亚群
err2025-11-05
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errChiara Vitale; Andrea Petretto; Katia Cortese; Sonia Carta; Alessandra Dondero; Chiara Lavarello; Davide Cangelosi; Martina Morini; Francesca Bellora; Pietro Arnaldi; Fabrizio Loiacono; Santina Bruzzone; Francesco Piacente; Silvia Bruno; Martina Serra; Annamaria Pessino; Serafina Mammoliti; Alberto Garaventa; Massimo Conte; Massimo Locati; Giuseppe Danilo Norata; Marco Colonna; Eric Vivier; Cristina Bottino; Roberta Castriconi
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From Bench to Clinic: The 2024 FASEB Scientific Research Conference on NAD Metabolism and Signaling从实验室到临床:2024年FASEB科学研討会关于NAD代谢与信号传导
err2025-10-31
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errShin-ichiro Imai; Eija Pirinen; Michael N. Sack; Jonas T. Treebak; Charalampos Tzoulis; Santina Bruzzone; Andreas H. Guse; Michael O. Hottiger; Xiaolu A. Cambronne
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Harnessing metabolic control for synaptic stability: REST/NRSF links glycolytic inhibition to excitatory neurotransmission利用代谢调控以维持突触稳定性:REST/NRSF将糖酵解抑制与兴奋性神经传递联系起来
err2025-10-10
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errDaniele Ferrante; Barbara Parisi; Antonella Marte; Dionisi Marianna; Cosimo Prestigio; Andrea Benzi; Santina Bruzzone; Fabio Benfenati; Franco Onofri; Pierluigi Valente; Pietro Baldelli
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Recent Advances in the Discovery of SIRT1/2 Inhibitors via Computational Methods: A Perspective
err2024-05-08
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errScarano, Naomi; Brullo, Chiara; Musumeci, Francesca; Millo, Enrico; Bruzzone, Santina; Schenone, Silvia; Cichero, Elena
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The TRPM2 ion channel regulates metabolic and thermogenic adaptations in adipose tissue of cold-exposed miceTRPM2离子通道调节冷暴露小鼠脂肪组织的代谢和生热适应
err2024-02-06
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errBenzi, Andrea; Heine, Markus; Spinelli, Sonia; Salis, Annalisa; Worthmann, Anna; Diercks, Bjorn; Astigiano, Cecilia; Mato, Raul Perez; Memushaj, Adela; Sturla, Laura; Vellone, Valerio; Damonte, Gianluca; Jaeckstein, Michelle Y.; Koch-Nolte, Friedrich; Mittrucker, Hans-Willi; Guse, Andreas H.; De Flora, Antonio; Heeren, Joerg; Bruzzone, Santina
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SIRT6 pharmacological inhibition delays skin cancer progression in the squamous cell carcinoma
err2023-10-01
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errAbbotto, Elena; Miro, Caterina; Piacente, Francesco; Salis, Annalisa; Murolo, Melania; Nappi, Annarita; Millo, Enrico; Russo, Eleonora; Cichero, Elena; Sturla, Laura; Del Rio, Alberto; De Flora, Antonio; Nencioni, Alessio; Dentice, Monica; Bruzzone, Santina
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Novel Thiazole-Based SIRT2 Inhibitors Discovered via Molecular Modelling Studies and Enzymatic Assays
err2023-09-18
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errAbbotto, Elena; Casini, Beatrice; Piacente, Francesco; Scarano, Naomi; Cerri, Elena; Tonelli, Michele; Astigiano, Cecilia; Millo, Enrico; Sturla, Laura; Bruzzone, Santina; Cichero, Elena
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PLX4032 resistance of patient-derived melanoma cells: crucial role of oxidative metabolism患者来源的黑色素瘤细胞的PLX4032抗性: 氧化代谢的关键作用
err2023-07-18
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errGarbarino, Ombretta; Valenti, Giulia Elda; Monteleone, Lorenzo; Pietra, Gabriella; Mingari, Maria Cristina; Benzi, Andrea; Bruzzone, Santina; Ravera, Silvia; Leardi, Riccardo; Farinini, Emanuele; Vernazza, Stefania; Grottoli, Melania; Marengo, Barbara; Domenicotti, Cinzia
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Targeting the deacetylase SIRT6 unveils spliceosome deregulation as exploitable vulnerability for aggressive myeloma
err2023-07-13
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errGelli, Elisa; Soncini, Debora; Becherini, Pamela; Martinuzzi, Claudia; Todoerti, Katia; Cagnetta, Antonia; Aquino, Sara; Guolo, Fabio; Miglino, Maurizio; Bruzzone, Santina; Nencioni, Alessio; Neri, Antonino; Lemoli, Roberto M.; Cea, Michele
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The influence of redox modulation on hypoxic endothelial cell metabolic and proteomic profiles through a small thiol-based compound tuning glutathione and thioredoxin systems
err2023-07-06
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errBruschi, Michela; Biancucci, Federica; Masini, Sofia; Piacente, Francesco; Ligi, Daniela; Bartoccini, Francesca; Antonelli, Antonella; Mannello, Ferdinando; Bruzzone, Santina; Menotta, Michele; Fraternale, Alessandra; Magnani, Mauro
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Mitochondrial rewiring drives metabolic adaptation to NAD(H) shortage in triple negative breast cancer cells线粒体重新布线驱动三阴性乳腺癌细胞对NAD(H) 短缺的代谢适应
err2023-07-01
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errCarreira, Agata Sofia Assuncao; Ravera, Silvia; Zucal, Chiara; Thongon, Natthakan; Irene, Caffa; Astigiano, Cecilia; Bertola, Nadia; Buongiorno, Arianna; Roccuzzo, Michela; Bisio, Alessandra; Pardini, Barbara; Nencioni, Alessio; Bruzzone, Santina; Provenzani, Alessandro
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Iminosugar-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors as Potential Anti-Pancreatic Cancer Agents
err2023-05-11
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errConforti, Irene; Benzi, Andrea; Caffa, Irene; Bruzzone, Santina; Nencioni, Alessio; Marra, Alberto
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Aberrant Adenosine Triphosphate Release and Impairment of P2Y2-Mediated Signaling in Sarcoglycanopathies
err2023-03-01
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errBenzi, Andrea; Baratto, Serena; Astigiano, Cecilia; Sturla, Laura; Panicucci, Chiara; Mamchaoui, Kamel; Raffaghello, Lizzia; Bruzzone, Santina; Gazzerro, Elisabetta; Bruno, Claudio
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Synthesis and structure-activity relationship of new nicotinamide phosphoribosyltransferase inhibitors with antitumor activity on solid and haematological cancer
err2023-03-01
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errFratta, Simone; Biniecka, Paulina; Moreno-Vargas, Antonio J.; Carmona, Ana T.; Nahimana, Aimable; Duchosal, Michel A.; Piacente, Francesco; Bruzzone, Santina; Caffa, Irene; Nencioni, Alessio; Robina, Inmaculada
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Anticancer Activities of Novel Nicotinamide Phosphoribosyltransferase Inhibitors in Hematological Malignancies新型烟酰胺磷酸核糖转移酶抑制剂在血液系统恶性肿瘤中的抗癌活性
err2023-02-16
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errBiniecka, Paulina; Matsumoto, Saki; Belotti, Axel; Joussot, Jessie; Bai, Jian Fei; Majjigapu, Somi Reddy; Thoueille, Paul; Spaggiari, Dany; Desfontaine, Vincent; Piacente, Francesco; Bruzzone, Santina; Cea, Michele; Decosterd, Laurent A. A.; Vogel, Pierre; Nencioni, Alessio; Duchosal, Michel A. A.; Nahimana, Aimable
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CD38-Induced Metabolic Dysfunction Primes Multiple Myeloma Cells for NAD+-Lowering AgentsCD38-Induced代谢功能障碍为多发性骨髓瘤细胞提供降低NAD的药物
err2023-02-15
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errBecherini, Pamela; Soncini, Debora; Ravera, Silvia; Gelli, Elisa; Martinuzzi, Claudia; Giorgetti, Giulia; Cagnetta, Antonia; Guolo, Fabio; Ivaldi, Federico; Miglino, Maurizio; Aquino, Sara; Todoerti, Katia; Neri, Antonino; Benzi, Andrea; Passalacqua, Mario; Nencioni, Alessio; Perrotta, Ida; Cantafio, Maria Eugenia Gallo; Amodio, Nicola; De Flora, Antonio; Bruzzone, Santina; Lemoli, Roberto M.; Cea, Michele
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A Versatile Continuous Fluorometric Enzymatic Assay for Targeting Nicotinate Phosphoribosyltransferase
err2023-01-18
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errMinazzato, Gabriele; Marangoni, Elisa; Fortunato, Carlo; Petrelli, Riccardo; Cappellacci, Loredana; Del Bello, Fabio; Sorci, Leonardo; Gasparrini, Massimiliano; Piacente, Francesco; Bruzzone, Santina; Raffaelli, Nadia
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