arrow
返回
J

Jan Korábečný

university hospital hradec kralove

43H指数
268论文数
6.0K被引数
收录论文 121
发表时间
Exploring the Structural Requirements of Fluorinated Benzylidene-Thiazolidinediones for Selective Antitrypanosomal Activity探索氟化苯亚甲基-噻唑烷二酮选择性抗锥虫活性的结构要求
err2026-09-29
err0
PREAI
errMichal Kolařík; Nuno Santarém; Anabela Cordeiro-da-Silva; Joana Tavares; Martin Novák; Vendula Rydlova; Jan Korábečný; Lucie Brulíková
err分享
err收藏
Chiral Separation of Tacrine-Based Metabolites: A Step Towards a Safe, Highly Active Drug他克林基代谢物的手性分离:迈向安全、高活性药物的一步
err2026-09-14
err0
errOAAI
errMartin Novak; Ondrej Horacek; Lucie Faltinova; Barbora Svobodova; Jan Korabecny; Martina Hrabinova; Ales Ruzicka; Martin Juhás; Sabine Willems; Volker Martin Lauschke; Lucie Novakova; Ondrej Soukup; Radim Kučera
err分享
err收藏
Why choose between prediction power and mechanistic insight in QSRR modeling? A case study of artificial membrane chromatography and machine learning为何在QSRR建模中需要在预测能力和机制洞察之间进行选择?——人工膜色谱与机器学习的案例研究
err2026-09-01
err0
PREAI
errNisterenko, Wiktor; Nicman, Julia; Deng, Jiayin; Singh, Yash Raj; Rozycka, Alicja; Greber, Katarzyna Ewa; Szulczyk, Daniel; Nowacki, Michal; Dawidowski, Maciej; Drabczyk, Anna; Jaskowska, Jolanta; Zareba, Przemyslaw; Kulaga, Damian; Staszewski, Marek; Wujec, Monika; Krzeczynski, Piotr; Michalak, Olga; Klejborowska, Greta; Scarpellini, Camilla; Augustyns, Koen; Dernovsek, Jaka; Tomasic, Tihomir; Korabecny, Jan; Fedorowicz, Joanna; Saczewski, Jaroslaw; Sawicki, Wieslaw; Ouyang, Defang; Ciura, Krzesimir
err分享
err收藏
Advancing Therapies for Mycobacterial Diseases: From Small Molecules to Host-Directed Strategies分枝杆菌疾病疗法的进展:从小分子到宿主导向策略
err2026-08-05
err0
errOAAI
errTânia Silva; Alessandra Aiello; Tonino Alonzi; M. Alice Carvalho; Vladimir Finger; Delia Goletti; Sven Hoffner; Yousra Kherabi; Jan Korabecny; Julia Kulczyńska; Agnieszka Kyzioł
err分享
err收藏
Carltonine B derivatives: Synthesis and structure-activity relationship insights for selective butyrylcholinesterase inhibition卡兰亭B衍生物:选择性丁酰胆碱酯酶抑制作用的合成与构效关系研究
err2026-04-20
err0
errOAAI
errAbdullah Al Mamun; Jan Konecny; Martina Hrabinova; Ales Sorf; Lubica Muckova; Jakub Fibigar; Tomas Kucera; Lenka Pulkrabkova; Daniel Jun; Lukas Prchal; Dawid Panek; Vladimir Finger; Ondrej Soukup; Thomas Cailly; Valérie Collot; Lucie Novakova; Lucie Cahlikova; Jan Korabecny
err分享
err收藏
Next-generation broad-spectrum reactivators for effective countermeasure against organophosphorus poisoning下一代广谱重活化剂,用于有效对抗有机磷中毒的对策
err2026-03-16
err0
errOAAI
errJana Zdarova Karasova; Martina Hrabinova; Alzbeta Dlabkova; Vendula Hepnarova; Natalie Zivna; Monika Schmidt; Valeria Sheshko; Carilyn Torruellas; Jakub Opravil; Lukas Prchal; Natalie Vanova; Jakub Fibigar; Zbynek Vecera; Tomas Kucera; Jaroslav Chladek; Gabriele Horn; Franz Worek; Jan Marek; Jaroslav Pejchal; Daniel Jun; Ondrej Soukup; Jan Korabecny; Lukas Gorecki
err分享
err收藏
Novel pyrimidine derivatives as promising antimycobacterial agents新型嘧啶衍生物作为有希望的抗分枝杆菌药物
err2026-01-21
err0
PREAI
errKufa, Martin; Finger, Vladimir; Kovar, Ondrej; Prchal, Lukas; Muckova, Lubica; Novak, Martin; Hympanova, Michaela; Janousek, Jiri; Benkova, Marketa; Kunes, Jiri; Bartacek, Jan; Soukup, Ondrej; Pavlis, Oto; Zdarova-Karasova, Jana; Odvarkova, Jitka; Savkova, Karin; Kordulakova, Jana; Roh, Jaroslav; Korabecny, Jan
err分享
err收藏
Reactivation screening of A-234-inhibited human recombinant acetylcholinesterase in vitroA-234抑制的人重组乙酰胆碱酯酶的体外重激活筛选
err2025-11-04
err0
PREAI
errJakub Opravil; Jaroslav Pejchal; Martina Hrabinova; Lubica Muckova; Lukas Prchal; Jan Korabecny; Tomas Rozsypal; Lukas Gorecki; Jakub Fibigar; Ondrej Soukup; Kamil Musilek; Daniel Jun
err分享
err收藏
Balancing rigidity and flexibility: Optimised 4-(hexyloxy)benzoate antagonists with enhanced affinity and tuneable duration at muscarinic receptors平衡刚性与柔性:具有增强亲和力和可调作用时长的优化4-(己氧基)苯甲酸酯拮抗剂在毒蕈碱受体上
err2025-10-22
err0
errOAAI
errEva Dolejší; Eva Mezeiova; Jana Bláhová; Nikolai Chetverikov; Alena Janoušková-Randáková; Dominik Nelic; Lukas Prchal; Barbora Svobodova; John Boulos; Jan Korabecny; Jan Jakubík
err分享
err收藏
Scaffold Hopping in Tuberculosis Drug Discovery: Principles; Applications; and Case Studies结核病药物发现中的骨架跃迁:原理、应用及案例研究
err2025-10-07
err0
errOAAI
errOndrej Kovar; Martin Kufa; Vladimir Finger; Ondrej Soukup; Martin Kratky; Carilyn Torruellas; Jaroslav Roh; Jan Korabecny
err分享
err收藏
Novel antitubercular agents based on 2,4-disubstituted 5-(aryl-2-ylmethyl)-5H-pyrrolo[3,2-d]pyrimidines基于2,4-二取代-5-(芳基-2-基甲基)-5H-吡咯并[3,2-d]嘧啶的新型抗结核药物
err2025-09-12
err0
PREAI
errVladimir Finger; Martin Vrbicky; Lubica Muckova; Lukas Prchal; Martin Novak; Jan Marek; Ondrej Soukup; Michaela Hympanova; Ales Sorf; Marketa Benkova; Jan Bartacek; Pavel Drabina; Martin Kufa; Ondrej Kovar; Lenka Fikejzlová; Martin Hruby; Oksana Ozhelevska; Johannes Jagob; Jana Zdarova-Karasova; Jitka Odvarkova; Iveta Kaderavková; Tomas Rozsypal; Katarzyna Ewa Greber; Krzesimir Ciura; Jiri Janousek; Martin Kratky; Ivone C. Igreja Sa; Pavel Bostik; Radek Sleha; Jaroslav Roh; Jan Korabecny
err分享
err收藏
err分享
err收藏
Dizocilpine derivatives as neuroprotective NMDA receptor antagonists without psychomimetic side effects
err2024-12-01
err0
errOAAI
errKonecny, Jan; Misiachna, Anna; Chvojkova, Marketa; Kleteckova, Lenka; Kolcheva, Marharyta; Novak, Martin; Prchal, Lukas; Ladislav, Marek; Hemelikova, Katarina; Netolicky, Jakub; Hrabinova, Martina; Kobrlova, Tereza; Karasova, Jana Zdarova; Pejchal, Jaroslav; Fibigar, Jakub; Vecera, Zbynek; Kucera, Tomas; Jendelova, Pavla; Zahumenska, Petra; Langore, Emily; Doderovic, Jovana; Pang, Yuan-Ping; Vales, Karel; Korabecny, Jan; Soukup, Ondrej; Horak, Martin
err分享
err收藏
Multifunctional, Fluorene-Based Modulator of Cholinergic and GABAergic Neurotransmission as a Novel Drug Candidate for Palliative Treatment of Alzheimer's Disease
err2024-11-22
err0
errOAAI
errPanek, Dawid; Pasieka, Anna; Jonczyk, Jakub; Gawlinska, Milena; Zareba, Paula; Siwek, Agata; Wolak, Malgorzata; Mordyl, Barbara; Gluch-Lutwin, Monika; Latacz, Gniewomir; Brazzolotto, Xavier; Chantegreil, Fabien; Nachon, Florian; Zdarova Karasova, Jana; Pejchal, Jaroslav; Mzik, Martin; Sestak, Vit; Prchal, Lukas; Odvarkova, Jitka; Soukup, Ondrej; Korabecny, Jan; Sorf, Ales; Hamsikova, Marie; Zemanova, Lucie; Muckova, Lubica; Vanova, Nela; Dryja, Pola; Salat, Kinga; Hoefner, Georg; Wanner, Klaus; Wieckowska, Anna; Malawska, Barbara
err分享
err收藏
Potent and reversible open-channel blocker of NMDA receptor derived from dizocilpine with enhanced membrane-to-channel inhibition
err2024-09-01
err1
errOAAI
errMisiachna, Anna; Konecny, Jan; Kolcheva, Marharyta; Ladislav, Marek; Prchal, Lukas; Netolicky, Jakub; Kortus, Stepan; Zahumenska, Petra; Langore, Emily; Novak, Martin; Hemelikova, Katarina; Hermanova, Zuzana; Hrochova, Michaela; Pelikanova, Anezka; Odvarkova, Jitka; Pejchal, Jaroslav; Kassa, Jiri; Karasova, Jana Zdarova; Korabecny, Jan; Soukup, Ondrej; Horak, Martin
err分享
err收藏
Pro-cognitive effects of dual tacrine derivatives acting as cholinesterase inhibitors and NMDA receptor antagonists
err2024-07-01
err2
errOAAI
errChvojkova, Marketa; Kolar, David; Kovacova, Katarina; Cejkova, Lada; Misiachna, Anna; Hakenova, Kristina; Gorecki, Lukas; Horak, Martin; Korabecny, Jan; Soukup, Ondrej; Vales, Karel
err分享
err收藏