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New diarylsulfonamide inhibitors of Leishmania infantum amastigotesINTERNATIONAL JOURNAL FOR PARASITOLOGY-DRUGS AND DRUG RESISTANCEIF3.42021-08-017OAAI
Methoxy and bromo scans on N-(5-methoxyphenyl) methoxybenzenesulphonamides reveal potent cytotoxic compounds, especially against the human breast adenocarcinoma MCF7 cell lineJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRYIF5.42021-06-098OAAI
Methylsulfanylpyridine based diheteroaryl isocombretastatin analogs as potent anti-proliferative agentsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92021-01-018OAAI
The Masked Polar Group Incorporation (MPGI) Strategy in Drug Design: Effects of Nitrogen Substitutions on Combretastatin and Isocombretastatin Tubulin InhibitorsMOLECULESIF4.62019-11-2618OAAI
Antitubulin sulfonamides: The successful combination of an established drug class and a multifaceted targetMEDICINAL RESEARCH REVIEWSIF11.62018-10-2533PREAI
Substitution at the indole 3 position yields highly potent indolecombretastatins against human tumor cellsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92018-10-0121OAAI
Pyridine Based Antitumour Compounds Acting at the Colchicine SiteCURRENT MEDICINAL CHEMISTRYIF3.52016-04-2043OA
Exploring the size adaptability of the B ring binding zone of the colchicine site of tubulin with para-nitrogen substituted isocombretastatinsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92015-07-0132PREAI
p,p-Dihydroxydihydrostilbenophanes Related to Antimitotic Combretastatins. Conformational Analysis and Its Relationship to Tubulin InhibitionJOURNAL OF ORGANIC CHEMISTRYIF3.62014-07-234PREAI
Endowing Indole-Based Tubulin Inhibitors with an Anchor for Derivatization: Highly Potent 3-Substituted Indolephenstatins and IndoleisocombretastatinsJOURNAL OF MEDICINAL CHEMISTRYIF6.82013-03-2072PREAI
New para-para Stilbenophanes: Synthesis by McMurry Coupling, Conformational Analysis and Inhibition of Tubulin PolymerisationCHEMISTRY-A EUROPEAN JOURNALIF3.72011-02-239PREAI
Exploring the effect of 2,3,4-trimethoxy-phenyl moiety as a component of indolephenstatinsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92010-02-0144PREAI
Isocombretastatins A: 1,1-Diarylethenes as potent inhibitors of tubulin polymerization and cytotoxic compoundsBIOORGANIC & MEDICINAL CHEMISTRYIF32009-09-0159PRE
Naphthalene combretastatin analogues:: Synthesis, cytotoxicity and antitubulin activityJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRYIF5.42008-10-0366OAAI
Naphthylphenstatins as tubulin ligands:: Synthesis and biological evaluationBIOORGANIC & MEDICINAL CHEMISTRYIF32008-10-0144PRE
Diarylmethyloxime and hydrazone derivatives with 5-indolyl moieties as potent inhibitors of tubulin polymerizationBIOORGANIC & MEDICINAL CHEMISTRYIF32008-06-0149PRE
Synthesis and conformational analysis of macrocyclic dihydroxystilbenes linked between the para-para positionsCHEMISTRY-A EUROPEAN JOURNALIF3.72007-08-159PREAI
Novel bile acid derivatives (BANBs) with cytostatic activity obtained by conjugation of their side chain with nitrogenated basesBIOCHEMICAL PHARMACOLOGYIF5.62007-05-0124PREAI
Novel cationic and neutral glycocholic acid and polyamine conjugates able to inhibit transporters involved in hepatic and intestinal bile acid uptakeBIOORGANIC & MEDICINAL CHEMISTRYIF32007-03-0126PRE
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