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Design and synthesis of multifunctional microtubule targeting agents endowed with dual pro-apoptotic and anti-autophagic efficacyEUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92022-05-018OAAI
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A non-toxic, reversibly released imaging probe for oral cancer that is derived from natural compoundsSCIENTIFIC REPORTSIF3.92021-07-077OAAI
Selective Fatty Acid Amide Hydrolase Inhibitors as Potential Novel Antiepileptic AgentsACS CHEMICAL NEUROSCIENCEIF3.92021-04-2315OA
Synthesis and biological evaluation of benzhydryl-based antiplasmodial agents possessing Plasmodium falciparum chloroquine resistance transporter (PfCRT) inhibitory activityEUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92021-04-016PREAI
Novel quinolone-based potent and selective HDAC6 inhibitors: Synthesis, molecular modeling studies and biological investigationEUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92021-02-0132PREAI
Spiroindoline-Capped Selective HDAC6 Inhibitors: Design, Synthesis, Structural Analysis, and Biological EvaluationACS MEDICINAL CHEMISTRY LETTERSIF42020-09-2934OAAI
Modulation of the Innate Immune Response by Targeting Toll-like Receptors: A Perspective on Their Agonists and AntagonistsJOURNAL OF MEDICINAL CHEMISTRYIF6.82020-08-2686PREAI
Retinitis Pigmentosa and Retinal Degenerations: Deciphering Pathways and Targets for Drug Discovery and DevelopmentACS CHEMICAL NEUROSCIENCEIF3.92020-06-2616PREAI
Development of novel multipotent compounds modulating endocannabinoid and dopaminergic systemsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92019-12-0114OAAI
Autophagy modulators for the treatment of oral and esophageal squamous cell carcinomas自噬调节剂用于治疗口腔和食管鳞状细胞癌MEDICINAL RESEARCH REVIEWSIF11.62019-11-1960PREAI
Screening and Phenotypical Characterization of Schistosoma mansoni Histone Deacetylase 8 (SmHDAC8) Inhibitors as Multistage Antischistosomal AgentsACS INFECTIOUS DISEASESIF3.82019-10-2930PREAI
Raising the bar in anticancer therapy: recent advances in, and perspectives on, telomerase inhibitorsDRUG DISCOVERY TODAYIF7.52019-07-0133OAAI
A light in the dark: state of the art and perspectives in optogenetics and optopharmacology for restoring visionFUTURE MEDICINAL CHEMISTRYIF3.42019-03-257PREAI
Enantioselective Synthesis of a Cyclopropane Derivative of Spliceostatin A and Evaluation of BioactivityORGANIC LETTERSIF52018-11-0517OAAI
Enantioselective Synthesis of Thailanstatin A Methyl Ester and Evaluation of in Vitro Splicing InhibitionJOURNAL OF ORGANIC CHEMISTRYIF3.62018-04-2627OAAI
Structure-based discovery of the first non-covalent inhibitors of Leishmania major tryparedoxin peroxidase by high throughput dockingSCIENTIFIC REPORTSIF3.92015-05-0757OAAI