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Adriano Martinelli

University of Pisa

40H指数
289论文数
4.4K被引数
收录论文 97
发表时间
Development of a cheminformatics platform for selectivity analyses of carbonic anhydrase inhibitors
err2019-12-19
err11
errOAAI
errPoli, Giulio; Galati, Salvatore; Martinelli, Adriano; Supuran, Claudiu T.; Tuccinardi, Tiziano
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Discovery of long-chain salicylketoxime derivatives as monoacylglycerol lipase (MAGL) inhibitors发现长链水杨酮肟衍生物作为单酰基甘油脂肪酶 (MAGL) 抑制剂
err2018-09-01
err30
errOAAI
errBononi, Giulia; Granchi, Carlotta; Lapillo, Margherita; Giannotti, Massimiliano; Nieri, Daniela; Fortunato, Serena; El Boustani, Maguie; Caligiuri, Isabella; Poli, Giulio; Carlson, Kathryn E.; Kim, Sung Hoon; Macchia, Marco; Martinelli, Adriano; Rizzolio, Flavio; Chicca, Andrea; Katzenellenbogen, John A.; Minutolo, Filippo; Tuccinardi, Tiziano
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Discovery of 1,5-Diphenylpyrazole-3-Carboxamide Derivatives as Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors
err2018-01-22
err43
errOAAI
errTabrizi, Mojgan Aghazadeh; Baraldi, Pier Giovanni; Baraldi, Stefania; Ruggiero, Emanuela; De Stefano, Lucia; Rizzolio, Flavio; Mannelli, Lorenzo Di Cesare; Ghelardini, Carla; Chicca, Andrea; Lapillo, Margherita; Gertsch, Jurg; Manera, Clementina; Macchia, Marco; Martinelli, Adriano; Granchi, Carlotta; Minutolo, Filippo; Tuccinardi, Tiziano
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Development of terphenyl-2-methyloxazol-5(4H)-one derivatives as selective reversible MAGL inhibitors
err2017-09-22
err28
errOAAI
errGranchi, Carlotta; Caligiuri, Isabella; Bertelli, Eleonora; Poli, Giulio; Rizzolio, Flavio; Macchia, Marco; Martinelli, Adriano; Minutolo, Filippo; Tuccinardi, Tiziano
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Structural Optimization of 4-Chlorobenzoylpiperidine Derivatives for the Development of Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors
err2016-11-14
err49
errOAAI
errGranchi, Carlotta; Rizzolio, Flavio; Palazzolo, Stefano; Carmignani, Sara; Macchia, Marco; Saccomanni, Giuseppe; Manera, Clementina; Martinelli, Adriano; Minutolo, Filippo; Tuccinardi, Tiziano
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Targeting Different Transthyretin Binding Sites with Unusual Natural Compounds
err2016-05-09
err18
PREAI
errOrtore, Gabriella; Orlandini, Elisabetta; Braca, Alessandra; Ciccone, Lidia; Rossello, Armando; Martinelli, Adriano; Nencetti, Susanna
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N-O-Isopropyl Sulfonamido-Based Hydroxamates as Matrix Metalloproteinase Inhibitors: Hit Selection and in Vivo Antiangiogenic Activity
err2015-08-28
err56
errOAAI
errNuti, Elisa; Cantelmo, Anna Rita; Gallo, Cristina; Bruno, Antonino; Bassani, Barbara; Camodeca, Caterina; Tuccinardi, Tiziano; Vera, Laura; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A.; Martinelli, Adriano; Dive, Vincent; Albini, Adriana; Rossello, Armando
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Identification of a new STAT3 dimerization inhibitor through a pharmacophore-based virtual screening approach
err2015-08-24
err32
errOAAI
errPoli, Giulio; Gelain, Arianna; Porta, Federica; Asai, Akira; Martinelli, Adriano; Tuccinardi, Tiziano
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Phenylpropanoids and flavonoids from Phlomis kurdica as inhibitors of human lactate dehydrogenase
err2015-08-01
err44
errOAAI
errBader, Ammar; Tuccinardi, Tiziano; Granchi, Carlotta; Martinelli, Adriano; Macchia, Marco; Minutolo, Filippo; De Tommasi, Nunziatina; Braca, Alessandra
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Pyrazole phenylcyclohexylcarbamates as inhibitors of human fatty acid amide hydrolases (FAAH)吡唑苯基环己基氨基甲酸酯作为人类脂肪酸酰胺水解酶 (FAAH) 的抑制剂
err2015-06-01
err19
PREAI
errTabrizi, Mojgan Aghazadeh; Baraldi, Pier Giovanni; Ruggiero, Emanuela; Saponaro, Giulia; Baraldi, Stefania; Romagnoli, Romeo; Martinelli, Adriano; Tuccinardi, Tiziano
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Development and Validation of a Docking-Based Virtual Screening Platform for the Identification of New Lactate Dehydrogenase Inhibitors
err2015-05-15
err22
errOAAI
errGranchi, Carlotta; Capecchi, Alice; Del Frate, Gianluca; Martinelli, Adriano; Macchia, Marco; Minutolo, Filippo; Tuccinardi, Tiziano
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4-Aryliden-2-methyloxazol-5(4H)-one as a new scaffold for selective reversible MAGL inhibitors
err2015-02-11
err20
errOAAI
errGranchi, Carlotta; Rizzolio, Flavio; Bordoni, Vittorio; Caligiuri, Isabella; Manera, Clementina; Macchia, Marco; Minutolo, Filippo; Martinelli, Adriano; Giordano, Antonio; Tuccinardi, Tiziano
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Highly Selective Salicylketoxime-Based Estrogen Receptor β Agonists Display Antiproliferative Activities in a Glioma Model
err2015-01-14
err22
errOAAI
errPaterni, Ilaria; Bertini, Simone; Granchi, Carlotta; Tuccinardi, Tiziano; Macchia, Marco; Martinelli, Adriano; Caligiuri, Isabella; Toffoli, Giuseppe; Rizzolio, Flavio; Carlson, Kathryn E.; Katzenellenbogen, Benita S.; Katzenellenbogen, John A.; Minutolo, Filippo
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Receptor-based virtual screening evaluation for the identification of estrogen receptor β ligands
err2014-09-29
err18
errOAAI
errTuccinardi, Tiziano; Poli, Giulio; Dell'Agnello, Marco; Granchi, Carlotta; Minutolo, Filippo; Martinelli, Adriano
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Extensive Consensus Docking Evaluation for Ligand Pose Prediction and Virtual Screening Studies
err2014-09-18
err95
PREAI
errTuccinardi, Tiziano; Poli, Giulio; Romboli, Veronica; Giordano, Antonio; Martinelli, Adriano
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Identification and characterization of a new reversible MAGL inhibitor
err2014-07-01
err54
PREAI
errTuccinardi, Tiziano; Granchi, Carlotta; Rizzolio, Flavio; Caligiuri, Isabella; Battistello, Vittoria; Toffoli, Giuseppe; Minutolo, Filippo; Macchia, Marco; Martinelli, Adriano
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