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收藏Synthesis and antibacterial evaluation of new naphthalimide-coumarin hybrids against multidrug-resistant S. aureus and M. tuberculosis
Rana, Preeti; Supriya, Manchella Sai; Kalam, Abdul; Eedulakanti, Chaitanya; Kaul, Grace; Akhir, Abdul; Sindhuja, Rachiraju Hema; Roy, Arnab; Agnivesh, Puja Kumari; Saxena, Deepanshi; Ahmad, Mohammad Naiyaz; Madhavi, Y. V.; Dasgupta, Arunava; Kalia, Nitin Pal; Nagesh, Narayana; Chopra, Sidharth; Nanduri, Srinivas
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收藏Design, synthesis and in vitro cytotoxic evaluation of 8-carboline tethered quinoline-4-carboxamide conjugates as DNA-interactive Topo II inhibitors
Soni, Jay Prakash; Devi, Priyanka; Chemitikanti, Sowjanya; Sharma, Anamika; Swamy, Chintha Venkata Dinesh; Phanindranath, Regur; Sathish, Manda; Nagesh, Narayana; Godugu, Chandraiah; Shankaraiah, Nagula
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收藏Benzimidazole based bis-carboxamide derivatives as promising cytotoxic agents: Design, synthesis, in silico and tubulin polymerization inhibition
Laxmikeshav, Kritika; Sharma, Pooja; Palepu, Manisurya; Sharma, Pravesh; Mahale, Ashutosh; George, Joel; Phanindranath, Regur; Dandekar, Manoj P.; Kulkarni, Onkar Prakash; Nagesh, Narayana; Shankaraiah, Nagula
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收藏Design, synthesis of DNA-interactive 4-thiazolidinone-based indolo-/pyrroloazepinone conjugates as potential cytotoxic and topoisomerase I inhibitors设计,合成DNA相互作用的基于4-噻唑烷酮的吲哚-/吡咯并氮杂酮缀合物作为潜在的细胞毒性和拓扑异构酶I抑制剂
Kadagathur, Manasa; Patra, Sandip; Devabattula, Geetanjali; George, Joel; Phanindranath, Regur; Shaikh, Arbaz Sujat; Sigalapalli, Dilep Kumar; Godugu, Chandraiah; Nagesh, Narayana; Tangellamudi, Neelima D.; Shankaraiah, Nagula
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收藏Synthesis and biological evaluation of novel imidazo[1,2-a] pyridine-oxadiazole hybrids as anti-proliferative agents: Study of microtubule polymerization inhibition and DNA binding
Sigalapalli, Dilep Kumar; Kiranmai, Gaddam; Devi, G. Parimala; Tokala, Ramya; Sana, Sravani; Tripura, Chaturvedula; Jadhav, Govinda Shivaji; Kadagathur, Manasa; Shankaraiah, Nagula; Nagesh, Narayana; Babu, Bathini Nagendra; Tangellamudi, Neelima D.
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收藏Benzimidazole-1,2,3-triazole hybrid molecules: synthesis and study of their interaction with G-quadruplex DNA
Singu, Padma S.; Chitakamarthi, Ushasri; Mahadik, Namita S.; Keerti, Bhamidipati; Valipenta, Narasimhulu; Mokale, Santosh N.; Nagesh, Narayana; Kumbhare, Ravindra M.
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收藏Design and synthesis of substituted (1-(benzyl)-1H-1,2,3-triazol-4-yl)(piperazin-1-yl)methanone conjugates: study on their apoptosis inducing ability and tubulin polymerization inhibition
Manasa, Kesari Lakshmi; Thatikonda, Sowjanya; Sigalapalli, Dilep Kumar; Vuppaladadium, Sowmya; Devi, Ganthala Parimala; Godugu, Chandraiah; Alvala, Mallika; Nagesh, Narayana; Babu, Bathini Nagendra
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收藏Synthesis and biological evaluation of pyrazole linked benzothiazole-β-naphthol derivatives as topoisomerase I inhibitors with DNA binding ability具有DNA结合能力的吡唑连接苯并噻唑-β-萘酚衍生物作为拓扑异构酶I抑制剂的合成和生物学评价
Nagaraju, Burri; Kovvuri, Jeshma; Kumar, C. Ganesh; Routhu, Sunitha Rani; Shareef, Md. Adil; Kadagathur, Manasa; Adiyala, Praveen Reddy; Alavala, Sateesh; Nagesh, Narayana; Kamal, Ahmed
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收藏Synthesis of DNA interactive C3-trans-cinnamide linked β-carboline conjugates as potential cytotoxic and DNA topoisomerase I inhibitors合成DNA相互作用的C3-trans-cinnamide连接的 β-咔啉缀合物作为潜在的细胞毒性和DNA拓扑异构酶I抑制剂
Sathish, Manda; Dushantrao, Sabanis Chetan; Nekkanti, Shalini; Tokala, Ramya; Thatikonda, Soujanya; Tangella, Yellaiah; Srinivas, Gunda; Cherukommu, Shirisha; Krishna, Namballa Hari; Shankaraiah, Nagula; Nagesh, Narayana; Kamal, Ahmed
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收藏Iodine-mediated one-pot intramolecular decarboxylation domino reaction for accessing functionalised 2-(1,3,4-oxadiazol-2-yl)anilines with carbonic anhydrase inhibitory action
Angapelly, Srinivas; Ramya, P. V. Sri; Sodhi, Rohini; Angeli, Andrea; Rangan, Krishnan; Nagesh, Narayana; Supuran, Claudiu T.; Arifuddin, Mohammed
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收藏Synthesis of podophyllotoxin linked β-carboline congeners as potential anticancer agents and DNA topoisomerase II inhibitors鬼臼毒素连接的 β-咔啉同源物作为潜在的抗癌剂和DNA拓扑异构酶II抑制剂的合成
Sathish, Manda; Kavitha, Botla; Nayak, V. Lakshma; Tangella, Yellaiah; Ajitha, Ayyappan; Nekkanti, Shalini; Alarifi, Abdullah; Shankaraiah, Nagula; Nagesh, Narayana; Kamal, Ahmed
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收藏Design, synthesis and biological evaluation of new β-carboline-bisindole compounds as DNA binding, photocleavage agents and topoisomerase I inhibitors新型 β-咔啉-双吲哚类化合物作为DNA结合,光裂解剂和拓扑异构酶I抑制剂的设计,合成和生物学评价
Kovvuri, Jeshma; Nagaraju, Burri; Nayak, V. Lakshma; Akunuri, Ravikumar; Rao, M. P. Narasimha; Ajitha, Ayyappan; Nagesh, Narayan; Kamal, Ahmed
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收藏Design, Synthesis, and in vitro and in vivo Evaluations of (Z)-3,4,5-Trimethoxystyrylbenzenesulfonamides/sulfonates as Highly Potent Tubulin Polymerization Inhibitors
Mahesh, Rasala; Nayak, Vadithe Lakshma; Babu, Korrapati Suresh; Riyaz, Syed; Shaik, Thokhir Basha; Kumar, Gajjela Bharth; Mallipeddi, Prema Latha; Reddy, Challa Ratna; Shekar, Kunta Chandra; Jose, Jedy; Nagesh, Narayana; Kamal, Ahmed
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