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Karl‐Norbert Klotz

University of Wurzburg

47H指数
252论文数
1.1W被引数
收录论文 100
发表时间
A2A Adenosine Receptor Antagonists and Their Efficacy in Rat Models of Parkinson's Disease
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IF5.2
err2025-02-26
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errOAAI
errSpinaci, Andrea; Buccioni, Michela; Dal Ben, Diego; Francucci, Beatrice; Klotz, Karl-Norbert; Marucci, Gabriella; Simola, Nicola; Morelli, Micaela; Pinna, Annalisa; Volpini, Rosaria; Lambertucci, Catia
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[1,2,4]Triazolo[1,5-c]pyrimidines as Tools to Investigate A3 Adenosine Receptors in Cancer Cell Lines[1,2,4] 三唑并 [1,5-c] 嘧啶作为研究癌细胞系中A3腺苷受体的工具
err2023-09-22
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PREAI
errFederico, Stephanie; Persico, Margherita; Trevisan, Letizia; Biasinutto, Chiara; Bolcato, Giovanni; Salmaso, Veronica; Da Ros, Tatiana; Gianferrara, Teresa; Prencipe, Filippo; Kachler, Sonja; Klotz, Karl-Norbert; Pacor, Sabrina; Moro, Stefano; Spalluto, Giampiero
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A2A Adenosine Receptor Antagonists: Are Triazolotriazine and Purine Scaffolds Interchangeable?
err2022-04-07
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errOAAI
errSpinaci, Andrea; Lambertucci, Catia; Buccioni, Michela; Dal Ben, Diego; Graiff, Claudia; Barbalace, Maria Cristina; Hrelia, Silvana; Angeloni, Cristina; Tayebati, Seyed Khosrow; Ubaldi, Massimo; Masi, Alessio; Klotz, Karl-Norbert; Volpini, Rosaria; Marucci, Gabriella
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Pharmacological characterisation of novel adenosine A3 receptor antagonists
err2020-11-27
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errBarkan, Kerry; Lagarias, Panagiotis; Stampelou, Margarita; Stamatis, Dimitrios; Hoare, Sam; Safitri, Dewi; Klotz, Karl-Norbert; Vrontaki, Eleni; Kolocouris, Antonios; Ladds, Graham
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Adenosine Receptor Ligands: Coumarin-Chalcone Hybrids as Modulating Agents on the Activity of hARs
err2020-09-19
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errOAAI
errVazquez-Rodriguez, Saleta; Vilar, Santiago; Kachler, Sonja; Klotz, Karl-Norbert; Uriarte, Eugenio; Borges, Fernanda; Matos, Maria Joao
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Targeting G Protein-Coupled Receptors with Magnetic Carbon Nanotubes: The Case of the A3Adenosine Receptor用磁性碳纳米管靶向g蛋白偶联受体: a3腺苷受体的情况
err2020-09-08
err4
PREAI
errPineux, Florent; Federico, Stephanie; Klotz, Karl-Norbert; Kachler, Sonja; Michiels, Carine; Sturlese, Mattia; Prato, Maurizio; Spalluto, Giampiero; Moro, Stefano; Bonifazi, Davide
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Structure-Based Optimization of Coumarin hA3 Adenosine Receptor Antagonists
err2019-11-18
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PREAI
errMatos, Maria Joao; Vilar, Santiago; Vazquez-Rodriguez, Saleta; Kachler, Sonja; Klotz, Karl-Norbert; Buccioni, Michela; Delogu, Giovanna; Santana, Lourdes; Uriarte, Eugenio; Borges, Fernanda
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Design, Synthesis and Evaluation of New Indolylpyrimidylpiperazines for Gastrointestinal Cancer Therapy
err2019-10-11
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errOAAI
errTan, Aaron; Babak, Maria, V; Venkatesan, Gopalakrishnan; Lim, Clarissa; Klotz, Karl-Norbert; Herr, Deron Raymond; Cheong, Siew Lee; Federico, Stephanie; Spalluto, Giampiero; Ong, Wei-Yi; Chen, Yu Zong; Loo, Jason Siau Ee; Pastorin, Giorgia
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A novel small molecule A2A adenosine receptor agonist, indirubin-3′-monoxime, alleviates lipid-induced inflammation and insulin resistance in 3T3-L1 adipocytes
err2019-08-30
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PREAI
errChoudhary, Saynaz A.; Bora, Nikita; Banerjee, Dipanjan; Arora, Leena; Das, Anindhya Sundar; Yadav, Rakesh; Klotz, Karl-Norbert; Pal, Durba; Jha, Anupam Nath; Dasgupta, Suman
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7-Amino-2-aryl/hetero-aryl-5-oxo-5,8-dihydro[1,2,4]triazolo[1,5-a]pyridine-6-carbonitriles: Synthesis and adenosine receptor binding studies
err2019-05-15
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PREAI
errShaik, Khasim; Deb, Pran Kishore; Mailavaram, Raghu Prasad; Chandrasekaran, Balakumar; Kachler, Sonja; Klotz, Karl-Norbert; Jaber, Abdul Muttaleb Yousef
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New potent and selective A1 adenosine receptor antagonists as potential tools for the treatment of gastrointestinal diseases
err2018-05-01
err13
PREAI
errLambertucci, Catia; Marucci, Gabriella; Dal Ben, Diego; Buccioni, Michela; Spinaci, Andrea; Kachler, Sonja; Klotz, Karl-Norbert; Volpini, Rosaria
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Discovery of Novel Adenosine Receptor Antagonists through a Combined Structure- and Ligand-Based Approach Followed by Molecular Dynamics Investigation of Ligand Binding Mode
err2018-02-27
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errLagarias, Panagiotis; Vrontaki, Eleni; Lambrinidis, George; Stamatis, Dimitrios; Convertino, Marino; Ortore, Gabriella; Mavromoustakos, Thomas; Klotz, Karl-Norbert; Kolocouris, Antonios
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Structure-Based Design, Synthesis, and In Vivo Antinociceptive Effects of Selective A1 Adenosine Receptor Agonists
err2018-01-03
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PREAI
errPetrelli, Riccardo; Scortichini, Mirko; Belardo, Carmela; Boccella, Serena; Luongo, Livio; Capone, Fabio; Kachler, Sonja; Vita, Patrizia; Del Bello, Fabio; Maione, Sabatino; Lavecchia, Antonio; Klotz, Karl-Norbert; Cappellacci, Loredana
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Synthesis, adenosine receptor binding and molecular modelling studies of novel thieno[2,3-d]pyrimidine derivatives
err2017-12-22
err32
PREAI
errDeb, Pran Kishore; Mailavaram, Raghuprasad; Chandrasekaran, Balakumar; Kaki, Venkata Rao; Kaur, Rajwinder; Kachler, Sonja; Klotz, Karl-Norbert; Akkinepally, Raghuram Rao
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