未登录A2A Adenosine Receptor Antagonists and Their Efficacy in Rat Models of Parkinson's Disease
Spinaci, Andrea; Buccioni, Michela; Dal Ben, Diego; Francucci, Beatrice; Klotz, Karl-Norbert; Marucci, Gabriella; Simola, Nicola; Morelli, Micaela; Pinna, Annalisa; Volpini, Rosaria; Lambertucci, Catia
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收藏[1,2,4]Triazolo[1,5-c]pyrimidines as Tools to Investigate A3 Adenosine Receptors in Cancer Cell Lines[1,2,4] 三唑并 [1,5-c] 嘧啶作为研究癌细胞系中A3腺苷受体的工具
Federico, Stephanie; Persico, Margherita; Trevisan, Letizia; Biasinutto, Chiara; Bolcato, Giovanni; Salmaso, Veronica; Da Ros, Tatiana; Gianferrara, Teresa; Prencipe, Filippo; Kachler, Sonja; Klotz, Karl-Norbert; Pacor, Sabrina; Moro, Stefano; Spalluto, Giampiero
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收藏A2A Adenosine Receptor Antagonists: Are Triazolotriazine and Purine Scaffolds Interchangeable?
Spinaci, Andrea; Lambertucci, Catia; Buccioni, Michela; Dal Ben, Diego; Graiff, Claudia; Barbalace, Maria Cristina; Hrelia, Silvana; Angeloni, Cristina; Tayebati, Seyed Khosrow; Ubaldi, Massimo; Masi, Alessio; Klotz, Karl-Norbert; Volpini, Rosaria; Marucci, Gabriella
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收藏Pharmacological characterisation of novel adenosine A3 receptor antagonists
Barkan, Kerry; Lagarias, Panagiotis; Stampelou, Margarita; Stamatis, Dimitrios; Hoare, Sam; Safitri, Dewi; Klotz, Karl-Norbert; Vrontaki, Eleni; Kolocouris, Antonios; Ladds, Graham
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收藏Targeting G Protein-Coupled Receptors with Magnetic Carbon Nanotubes: The Case of the A3Adenosine Receptor用磁性碳纳米管靶向g蛋白偶联受体: a3腺苷受体的情况
Pineux, Florent; Federico, Stephanie; Klotz, Karl-Norbert; Kachler, Sonja; Michiels, Carine; Sturlese, Mattia; Prato, Maurizio; Spalluto, Giampiero; Moro, Stefano; Bonifazi, Davide
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收藏Structure-Based Optimization of Coumarin hA3 Adenosine Receptor Antagonists
Matos, Maria Joao; Vilar, Santiago; Vazquez-Rodriguez, Saleta; Kachler, Sonja; Klotz, Karl-Norbert; Buccioni, Michela; Delogu, Giovanna; Santana, Lourdes; Uriarte, Eugenio; Borges, Fernanda
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收藏Design, Synthesis and Evaluation of New Indolylpyrimidylpiperazines for Gastrointestinal Cancer Therapy
Tan, Aaron; Babak, Maria, V; Venkatesan, Gopalakrishnan; Lim, Clarissa; Klotz, Karl-Norbert; Herr, Deron Raymond; Cheong, Siew Lee; Federico, Stephanie; Spalluto, Giampiero; Ong, Wei-Yi; Chen, Yu Zong; Loo, Jason Siau Ee; Pastorin, Giorgia
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收藏A novel small molecule A2A adenosine receptor agonist, indirubin-3′-monoxime, alleviates lipid-induced inflammation and insulin resistance in 3T3-L1 adipocytes
Choudhary, Saynaz A.; Bora, Nikita; Banerjee, Dipanjan; Arora, Leena; Das, Anindhya Sundar; Yadav, Rakesh; Klotz, Karl-Norbert; Pal, Durba; Jha, Anupam Nath; Dasgupta, Suman
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收藏7-Amino-2-aryl/hetero-aryl-5-oxo-5,8-dihydro[1,2,4]triazolo[1,5-a]pyridine-6-carbonitriles: Synthesis and adenosine receptor binding studies
Shaik, Khasim; Deb, Pran Kishore; Mailavaram, Raghu Prasad; Chandrasekaran, Balakumar; Kachler, Sonja; Klotz, Karl-Norbert; Jaber, Abdul Muttaleb Yousef
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收藏[1,2,4]Triazolo[1,5-c]pyrimidines as adenosine receptor antagonists: Modifications at the 8 position to reach selectivity towards A3 adenosine receptor subtype[1,2,4] 三唑并 [1,5-c] 嘧啶作为腺苷受体拮抗剂: 在8位进行修饰以实现对A3腺苷受体亚型的选择性
Federico, Stephanie; Margiotta, Enrico; Salmaso, Veronica; Pastorin, Giorgia; Kachler, Sonja; Klotz, Karl-Norbert; Moro, Stefano; Spalluto, Giampiero
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收藏Structure-Based Design, Synthesis, and In Vivo Antinociceptive Effects of Selective A1 Adenosine Receptor Agonists
Petrelli, Riccardo; Scortichini, Mirko; Belardo, Carmela; Boccella, Serena; Luongo, Livio; Capone, Fabio; Kachler, Sonja; Vita, Patrizia; Del Bello, Fabio; Maione, Sabatino; Lavecchia, Antonio; Klotz, Karl-Norbert; Cappellacci, Loredana
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收藏Synthesis, adenosine receptor binding and molecular modelling studies of novel thieno[2,3-d]pyrimidine derivatives
Deb, Pran Kishore; Mailavaram, Raghuprasad; Chandrasekaran, Balakumar; Kaki, Venkata Rao; Kaur, Rajwinder; Kachler, Sonja; Klotz, Karl-Norbert; Akkinepally, Raghuram Rao
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