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Daulat Bikram Khadka

chonnam national university

H指数:19

被引数:1,048

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Structure-based discovery of pyrazolamides as novel ERR? inverse agonists

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2023-03-013

PRE

SAR study of bisamides as cyclophilin a inhibitors for the development of host-targeting therapy for hepatitis C virus infection

双酰胺作为亲环素a抑制剂的SAR研究，用于开发针对丙型肝炎病毒感染的宿主靶向治疗

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2020-10-015

PREAI

Molecular design, synthesis, and biological evaluation of bisamide derivatives as cyclophilin A inhibitors for HCV treatment

亲环素A抑制剂双酰胺衍生物的分子设计、合成及生物学评价

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2020-02-0116

PREAI

A maresin 1/RORα/12-lipoxygenase autoregulatory circuit prevents inflammation and progression of nonalcoholic steatohepatitis

JOURNAL OF CLINICAL INVESTIGATION

IF13.6

2019-03-11114

OA

Synthesis of Aryl Trimethylstannane via BF3•OEt2-Mediated Cross-Coupling of Hexaalkyl Distannane Reagent with Aryl Triazene at Room Temperature

JOURNAL OF ORGANIC CHEMISTRY

IF3.6

2018-12-1228

PREAI

Design, synthesis, and systematic evaluation of 4-arylpiperazine- and 4-benzylpiperidine napthyl ethers as inhibitors of monoamine neurotransmitters reuptake

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2018-11-013

PREAI

Design, synthesis and docking study of 4-arylpiperazine carboxamides as monoamine neurotransmitters reuptake inhibitors

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2018-08-018

PREAI

Design, synthesis, and biological evaluation of 1,3-diarylisoquinolines as novel topoisomerase I catalytic inhibitors

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2018-01-0113

PREAI

Triple reuptake inhibitors: Design, synthesis and structure-activity relationship of benzylpiperidine-tetrazoles

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2017-10-0116

PREAI

Berberine bioisostere Q8 compound stimulates osteoblast differentiation and function in vitro

PHARMACOLOGICAL RESEARCH

IF10.5

2017-05-0116

PREAI

Discovery of Isoquinolinoquinazolinones as a Novel Class of Potent PPARγ Antagonists with Anti-adipogenic Effects

SCIENTIFIC REPORTS

IF3.9

2016-10-039

OAAI

Insights into the Structural Features Essential for JAK2 Inhibition and Selectivity

CURRENT MEDICINAL CHEMISTRY

IF3.5

2016-05-067

PRE

Design and synthesis of novel androgen receptor antagonists via molecular modeling

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2016-02-018

PREAI

Structure-Based Discovery of Novel Cyclophilin A Inhibitors for the Treatment of Hepatitis C Virus Infections

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2015-12-0822

PREAI

Pharmacological effects of berberine and its derivatives: a patent update

EXPERT OPINION ON THERAPEUTIC PATENTS

IF4.6

2015-12-04148

PREAI

Substituted 2-arylquinazolinones: Design, synthesis, and evaluation of cytotoxicity and inhibition of topoisomerases

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2015-10-0121

PREAI

Modification of 3-arylisoquinolines into 3,4-diarylisoquinolines and assessment of their cytotoxicity and topoisomerase inhibition

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2015-03-0126

PREAI

Computer-aided discovery of aminopyridines as novel JAK2 inhibitors

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2015-03-0110

PREAI

Design, synthesis and systematic evaluation of cytotoxic 3-heteroarylisoquinolinamines as topoisomerases inhibitors

作为拓扑异构酶抑制剂的细胞毒性3-杂芳基异喹啉胺的设计，合成和系统评价

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2014-07-0126

PREAI

Topoisomerase inhibitors as anticancer agents: a patent update

EXPERT OPINION ON THERAPEUTIC PATENTS

IF4.6

2013-04-2382

PREAI