未登录Design, Synthesis and Evaluation of Novel Pyrrolidinone-Based ACE2 Inhibitors: Preliminary Study基于吡咯烷酮类的新型ACE2抑制剂的分子设计、合成与评价:初步研究
Nigro, Ilaria; Armentano, Maria Francesca; Caruso, Anna; El-Kashef, Hussein; Giuzio, Federica; Vassallo, Antonio; Finelli, Francesca; Monne, Magnus; Saturnino, Carmela
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收藏Widespread non-adherence to guidelines in the operative management of diabetes-related foot disease complications在糖尿病相关足部疾病并发症的手术管理中普遍不遵守指南
Renwick, B.; Gannon, M.; Kerr, S.; Melvin, R.; Ingram, A.; Bosanquet, D.; Fabre, I; Yew, S.; Moreau, J.; Dewi, M.; Lowry, D.; Clothier, A.; Hutchings, T.; Boyle, J.; Wijewardena, C.; Chowdhury, M.; La Torre, G.; Grewal, H.; Ansaripour, A.; Lawson, D.; Nandhra, S.; Ugwumba, L.; El-Sayed, T.; Altahir, A.; Elkashef, H.; Jones, S.; Arkle, J.; Khalil, R.; Ramsay, J.; Nesbitt, C.; Paravastu, S.; Jayaprakash, V. V.; Flumignan, R. L. G.; Flumignan, C. D. Q.; Nakano, L. C. U.; Schippers, P.; Pereira, F. A., Jr.; Pegas, N. C.; Hitchman, L.; Walshaw, J.; Ravindhran, B.; Lathan, R.; Smith, G.; Shalhoub, J.; Ahmad, M.; Shea, J.; Howard, T.; Elsanhoury, K.; Eskandar, G.; Mekhaeil, K.; Scott, K.; Enc, M.; Mannan, F.; Chowdhury, S.; Abdelmageed, A. E.; Russell, D.; Jones, A.; Dattani, N.; El-nakhal, T.; Katsogridakis, E.; Duncan, A.; Musto, L.; Proctor, D.; Parsapour, S.; Lewis, S.; Hassan, A.; Abdelal, A.; Elzefzaf, N.; Yasser, N.; Antoniou, G. A.; Singh, A.; Alhoussan, L.; Venkateswaran, V.; Feil, F.; Dindyal, S.; Lyons, O.; Benson, R.; Lim, E.; Sze, M.; Khashram, M.; Hart, O.; Vincent, Z.; Xue, N.; Pottier, M.; Gormley, S.; Tong, C.; Pang, D.; Patil, A.; Ngam, L.; Macleod, C.; Aziz, I; Stather, P.; Abuduruk, A.; Manson, J.; Howard, D.; Hussain, S.; Glatzel, H.; James, N.; Rafil, M.; Marlow, N.; Meldrum, A.; Hussey, K.; Jones, C.; Shepherd, E.; Fitridge, R.; Hon, K.; Kour, K.; Ng, S.; Hardy, T.; Muse, S.; Ching, D.; Donoghue, S.; Thompson, D.; Forsythe, R.; Chan, S.; Powezka, K.; Wu, D.; Kuronen-Stewart, C.; Winarski, A.; Lapolla, P.; Cirillo, B.; Al-Saadi, N.; Dowdeswell, M.; McDonald, S.; Al-Hashimi, K.; Merriman, K.; Hassouneh, A.; Sadia, U.; Jaipersad, A.; Moulakakis, K. G.; Papageorgopoulou, C.; Kakkos, S.; Tsimpoukis, A.; Papadoulas, S.; Kouri, N.; Nikolakopoulos, K.; D'Oria, M.; Lepidi, S.; Grando, B.; Nickinson, A.; Gamtkitsulashvili, G.; Enemosah, I; Storer, N.; Gabab, K.; Dingwell, M.; Premadasan, Y.; Karkos, C.; Mitka, M.; Soteriou, A.; Asaloumidis, N.; Papazoglou, K.; Condie, N.; Abdullahi, H.; Shafeek, F.; Lyons, T.; Ambler, G.; Benson, R. A.; Birmpili, P.; Blair, R. H. J.; Bosanquet, D. C.; Gwilym, B. L.; Hurndall, K.; Machin, M.; Onida, S.; Saratzis, A.; Singh, A. A.; Shelmerdine, L.
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收藏Synthesis of Nitrostyrylthiazolidine-2,4-dione Derivatives Displaying Antileishmanial Potential
Khoumeri, Omar; Hutter, Sebastien; Primas, Nicolas; Castera-Ducros, Caroline; Carvalho, Sandra; Wyllie, Susan; Efrit, Mohamed Lotfi; Fayolle, Dimitri; Since, Marc; Vanelle, Patrice; Verhaeghe, Pierre; Azas, Nadine; El-Kashef, Hussein
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收藏Novel Thiazolidine-2,4-dione-trimethoxybenzene-thiazole Hybrids as Human Topoisomerases Inhibitors
Sinicropi, Maria Stefania; Ceramella, Jessica; Vanelle, Patrice; Iacopetta, Domenico; Rosano, Camillo; Khoumeri, Omar; Abdelmohsen, Shawkat; Abdelhady, Wafaa; El-Kashef, Hussein
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收藏N-Heterocyclic Carbene (NHC) Silver Complexes as Versatile Chemotherapeutic Agents Targeting Human Topoisomerases and Actin
Mariconda, Annaluisa; Iacopetta, Domenico; Sirignano, Marco; Ceramella, Jessica; Costabile, Chiara; Pellegrino, Michele; Rosano, Camillo; Catalano, Alessia; Saturnino, Carmela; El-Kashef, Hussein; Aquaro, Stefano; Sinicropi, Maria Stefania; Longo, Pasquale
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收藏Benzothienoquinazolinones as new multi-target scaffolds: Dual inhibition of human Topoisomerase I and tubulin polymerization
Ceramella, Jessica; Caruso, Anna; Occhiuzzi, Maria Antonietta; Lacopetta, Domenico; Barbarossa, Alexia; Rizzuti, Bruno; Dallemagne, Patrick; Rault, Sylvain; El-Kashef, Hussein; Saturnino, Carmela; Grande, Fedora; Sinicropi, Maria Stefania
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收藏Antitrypanosomatid Pharmacomodulation at Position 3 of the 8-Nitroquinolin-2(1H)-one Scaffold Using Palladium-Catalysed Cross-Coupling Reactions
Pedron, Julien; Boudot, Clotilde; Bourgeade-Delmas, Sandra; Sournia-Saquet, Alix; Paloque, Lucie; Rastegari, Maryam; Abdoulaye, Mansour; El-Kashef, Hussein; Bonduelle, Colin; Pratviel, Genevieve; Wyllie, Susan; Fairlamb, Alan H.; Courtioux, Bertrand; Verhaeghe, Pierre; Valentin, Alexis
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收藏Discovery of new hit-molecules targeting Plasmodium falciparum through a global SAR study of the 4-substituted-2-trichloromethylquinazoline antiplasmodial scaffold
Desroches, Justine; Kieffer, Charline; Primas, Nicolas; Hutter, Sebastien; Gellis, Armand; El-Kashef, Hussein; Rathelot, Pascal; Verhaeghe, Pierre; Azas, Nadine; Vanelle, Patrice
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收藏3-(Dipropylamino)-5-hydroxybenzofuro[2,3-f]quinazolin-1 (2H)-one (DPA-HBFQ-1) plays an inhibitory role on breast cancer cell growth and progression
Rizza, Pietro; Pellegrino, Michele; Caruso, Anna; Iacopetta, Domenico; Sinicropi, Maria Stefania; Rault, Sylvain; Lancelot, Jean Charles; El-Kashef, Hussein; Lesnard, Aurelien; Rochais, Christophe; Dallemagne, Patrick; Saturnino, Carmela; Giordano, Francesca; Catalano, Stefania; Ando, Sebastiano
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收藏Indenopyrazole oxime ethers: Synthesis and β1-adrenergic blocking activity
Angelone, Tommaso; Caruso, Anna; Rochais, Christophe; Caputo, Angela Maria; Cerra, Maria Carmela; Dallemagne, Patrick; Filice, Elisabetta; Genest, David; Pasqua, Teresa; Puoci, Francesco; Saturnino, Carmela; Sinicropi, Maria Stefania; El-Kashef, Hussein
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收藏Enhanced cellular uptake by pharmaceutically oriented devices of new simplified analogs of Linezolid with antimicrobial activity
Parisi, Ortensia Ilaria; Fiorillo, Marco; Caruso, Anna; Cappello, Anna Rita; Saturnino, Carmela; Puoci, Francesco; Panno, Antonella; Dolce, Vincenza; El-Kashef, Hussein; Sinicropi, Maria Stefania
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收藏Antiproliferative activity of some 1,4-dimethylcarbazoles on cells that express estrogen receptors: part I
Caruso, Anna; Chimento, Adele; El-Kashef, Hussein; Lancelot, Jean-Charles; Panno, Antonella; Pezzi, Vincenzo; Saturnino, Carmela; Sinicropi, Maria Stefania; Sirianni, Rosa; Rault, Sylvain
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收藏Synthesis, inhibition of NO production and antiproliferative activities of some indole derivatives
Sinicropi, Maria Stefania; Caruso, Anna; Conforti, Filomena; Marrelli, Mariangela; El Kashef, Hussein; Lancelot, Jean-charles; Rault, Sylvain; Statti, Giancarlo A.; Menichini, Francesco
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收藏Unexpected hydrazinolysis behaviour of 1-chloro-4-methyl-5H-pyridazino[4,5-b]indole and a convenient synthesis of new[1,2,4]-triazolo [4′,3′:1,6]pyridazino[4,5-b]indoles
El-Kashef, H; Farghaly, AAH; Haider, N; Wobus, A
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