Kenneth Goossens

Universite Paris Cite

H指数:6

被引数:464

浏览量:0

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A Computational Community Blind Challenge on Pan-Coronavirus Drug Discovery Data

Journal of Chemical Information and Modeling

IF5.3

2026-03-231

PRE

MacDermott-Opeskin, Hugo; Scheen, Jenke; Wognum, Cas; Horton, Joshua T.; West, Devany; Payne, Alexander Matthew; Castellanos, Maria A.; Colby, Sean; Griffen, Edward; Cousins, David; Stacey, Jessica; Reid, Lauren; Aschenbrenner, Jasmin Cara; Fearon, Daren; Balcomb, Blake; Marples, Peter; Tomlinson, Charles W. E.; Lithgo, Ryan; Godoy, Andre S.; Winokan, Max; Barr, Haim; Lahav, Noa; Lavi, Michael; Duberstein, Shirley; Cohen, Galit; Fate, Gwendolyn; Lefker, Bruce; Robinson, Ralph; Szommer, Tamas; Lynch, Nick; Minh, David D. L.; Van Ngoc Thuy La; Kang, Lulu; Huddleston, Kate; Renslow, Ryan; Tollefson, Mallory; Walters, W. Patrick; Xu, Cynthia; Hsu, Jonny; St-Laurent, Julien; Etsmoberg, Honore; Zhu, Lu; Quirke, Andrew; Haleem, Mohamed Iliyas Abdul; Alibay, Irfan; Baid, Gunjan; Birnbaum, Benjamin; Bishop, Kevin P.; Bohorquez, Hugo; Bose, Ashmita; Brown, C. J.; Burns, Jackson; Cai, Lianjin; Cedeno, Ruel; de Cesco, Stephane; Chupakhin, Vladimir; Clark, Finlay; Cole, Daniel J.; Corbi-Verge, Carles; Danial, Muhammad; Davi, Alec; Dehaen, Wim; Doering, Niklas Piet; Dougha, Alexis; Dreanic, Marie-Pierre; Eakin, Bryce; Ehrlich, Anatol; Elijosius, Rokas; Fulop, Jozef; Gitter, Anthony; Goossens, Kenneth; Gu, Yaowen; Head-Gordon, Teresa; Hoffer, Laurent; Hofmans, Johan; Jiang, Ellena; Kaminow, Benjamin; Khosravi, Sina; Khoualdi, Asma Feriel; Lenselink, Eelke Bart; Liu, Zhirong; Liu, Yue; Liu, Sijie; Ma, Yizhou; Maher, Patrick; Mayer, Imke; Mendez-Lucio, Oscar; Mey, Antonia S. J. S.; Michel, Julien; Montanari, Floriane; Niu, Taoyu; Ogino, Ryusei; Palaniappan, Ashok; Pan, Xiaolin; Patnaik, Auro; Pham, Long-Hung; Pinto, Luis; Purnomo, Justin; Rich, Alex; Schaaf, Lars; Schran, Christoph; Singh, Rajeev Kumar; Srilakshmi, Mounika; Srivastava, Satya Pratik; Sun, Kunyang; Sun, Zhaoxi; Talagayev, Valerij; Balakrishnan, Balamurugan Thirukonda Subramanian; Titus, Ida; Tkatchenko, Alexandre; Treyde, Wojtek; Tricarico, Giovanni; Tripp, Austin; Vithayapalert, Nopsinth; Wang, Yingze; Wasi, Azmine Toushik; Wedig, Steffen; Wolber, Gerhard; Xu, Bofei; Zhou, Weijun; von Delft, Frank; Lee, Alpha; Kirkegaard, Karla; Sjo, Peter; Fraser, James S.; Chodera, John D.

Structure activity relationship exploration of imidazo[1,2-a]pyridine series to reverse isoform selectivity and identify potent SIK1 selective inhibitors

咪唑并[1,2-a]吡啶类化合物的构效关系研究，旨在逆转同种异型选择性并鉴定高活性SIK1选择性抑制剂

Bioorganic & Medicinal Chemistry Letters

IF2.2

2025-09-080

PRE

Structure–Activity Relationship Guided Scaffold Hopping Resulted in the Identification of GLPG4970; a Highly Potent Dual SIK2/SIK3 Inhibitor

基于构效关系指导的骨架跳跃发现了GLPG4970；一种高活性双重SIK2/SIK3抑制剂

Journal of Medicinal Chemistry

IF6.8

2025-07-250

PRE

Hans Kelgtermans; Maxim De Wachter; Stijn Heyndrickx; Sandy El Bkassiny; Tatiana Lacarriere; Chris Laruelle; Jörg Heiermann; Wendy van Bruggen; Katarzyna Drabik; Denis Bucher; Thomas Coudrat; Emilie Jigorel; Kenneth Goossens; Michael Drennan; Martine Vrints; Maarten Verbeeck; Bas Housmans; Damien Ronsse; David Moreno-Delgado; Vahid Nassiri; Mia Jans; Maarten Gees; Emanuelle Wakselman; Line Oste; Monica Borgonovi; Elena Borregán-Ochando; Vladyslav Sushko; Alain Monjardet; Camille Dusserre; Frederique Van Acker; Anouk Blaauw; Stephanie Lavazais; Catherine Jagerschmidt; Didier Merciris; Michael Török-Schafroth; Christian A. Seemayer; Katja Conrath; Fabrice A. Kolb; Pierre Raboisson; Reginald Brys; David Amantini; Romain Gosmini; Alexis Denis; Juan-Miguel Jimenez; Steve De Vos; Nicolas Desroy

Modulation of taxane binding to tubulin curved and straight conformations by systematic 3′N modification provides for improved microtubule binding, persistent cytotoxicity and in vivo potency

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2023-11-012

PRE

From PERK to RIPK1: Design, synthesis and evaluation of novel potent and selective necroptosis inhibitors

从PERK到RIPK1: 新型有效和选择性坏死性凋亡抑制剂的设计，合成和评估

FRONTIERS IN CHEMISTRY

IF4.2

2023-04-073

OAAI

Assessment of the Fragment Docking Program SEED