Discovery of Substituted (2-Aminooxazol-4-yl)Isoxazole-3-carboxylic Acids as Inhibitors of Bacterial Serine Acetyltransferase in the Quest for Novel Potential Antibacterial AdjuvantsPHARMACEUTICALSIF4.82021-02-237OAAI
Investigational Studies on a Hit Compound Cyclopropane-Carboxylic Acid Derivative Targeting O-Acetylserine Sulfhydrylase as a Colistin AdjuvantACS INFECTIOUS DISEASESIF3.82021-01-2915PRE
Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase InhibitorACS MEDICINAL CHEMISTRY LETTERSIF42020-02-1318OAAI
Refining the structure-activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoformsJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRYIF5.42018-10-2612OAAI
Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand-based drug designJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRYIF5.42018-09-1717OAAI
Endoperoxide-8-aminoquinoline hybrids as dual-stage antimalarial agents with enhanced metabolic stabilityEUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92018-04-0129PREAI
Integration of Enhanced Sampling Methods with Saturation Transfer Difference Experiments to Identify Protein Druggable PocketsJOURNAL OF CHEMICAL INFORMATION AND MODELINGIF5.32018-02-2615PREAI
Cyclopropane-1,2-dicarboxylic acids as new tools for the biophysical investigation of O-acetylserine sulfhydrylases by fluorimetric methods and saturation transfer difference (STD) NMRJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRYIF5.42016-08-3119OAAI
From hybrid compounds to targeted drug delivery in antimalarial therapyBIOORGANIC & MEDICINAL CHEMISTRYIF32015-08-0149PREAI
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