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Structure-Activity Investigations and Optimisations of Non-metabolite Agonists for the Succinate Receptor 1SCIENTIFIC REPORTSIF3.92018-07-0320OAAI
Receptor structure-based discovery of non-metabolite agonists for the succinate receptor GPR91MOLECULAR METABOLISMIF6.62017-12-0149OAAI
Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitorsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92017-04-0149OAAI
Linker-switch approach towards new ATP binding site inhibitors of DNA gyrase BEUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92017-01-0113PREAI
Molecular Mechanism of Action for Allosteric Modulators and Agonists in CC-chemokine Receptor 5 (CCR5)JOURNAL OF BIOLOGICAL CHEMISTRYIF3.92016-12-0111OAAI
New N-phenyl-4,5-dibromopyrrolamides and N-Phenylindolamides as ATPase inhibitors of DNA gyraseEUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92016-07-0134PREAI
N-Phenyl-4,5-dibromopyrrolamides and N-Phenylindolamides as ATP Competitive DNA Gyrase B Inhibitors: Design, Synthesis, and EvaluationJOURNAL OF MEDICINAL CHEMISTRYIF6.82015-07-1557PREAI
Discovery of 4,5,6,7-Tetrahydrobenzo[1,2-d]thiazoles as Novel DNA Gyrase Inhibitors Targeting the ATP-Binding SiteJOURNAL OF MEDICINAL CHEMISTRYIF6.82015-07-08105PREAI
Discovery of Mono- and Disubstituted 1H-Pyrazolo[3,4]pyrimidines and 9H-Purines as Catalytic Inhibitors of Human DNA Topoisomerase IIαCHEMMEDCHEMIF3.42014-12-1730PREAI
Discovery of the first inhibitors of bacterial enzyme D-aspartate ligase from Enterococcus faecium (ASlfm)EUROPEAN JOURNAL OF MEDICINAL CHEMISTRYIF5.92013-09-0128PREAI
Structure-Based Discovery of Substituted 4,5′-Bithiazoles as Novel DNA Gyrase InhibitorsJOURNAL OF MEDICINAL CHEMISTRYIF6.82012-07-05153PREAI
In silico discovery and biophysical evaluation of novel 5-(2-hydroxybenzylidene) rhodanine inhibitors of DNA gyrase BBIOORGANIC & MEDICINAL CHEMISTRYIF32012-04-0148PRE