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M

M. Paul Gleeson

King Mongkut's Institute of Technology

24H指数
113论文数
4.1K被引数
收录论文 47
发表时间
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3-[[4-(Benzylamino)quinazolin-2-yl] Amino] Benzenesulfonamide, a Quinazoline-Based PDE5 Inhibitor, Induces Vasorelaxation in Rat Mesenteric Arteries via Multiple Mechanisms3-[[4-(苄基氨基)喹唑啉-2-基]氨基]苯磺酰胺，一种基于喹唑啉的PDE5抑制剂，通过多种机制诱导大鼠肠系膜动脉血管舒张
errBASIC & CLINICAL PHARMACOLOGY & TOXICOLOGY
IF3.3
err2026-10-25
err0
PREAI
errUsana Chatturong; Krongkarn Chootip; M. Paul Gleeson; Guntur Guntur; Yasuteru Shigeta; Kowit Hengphasatporn; Perle Totoson; Céline Demougeot
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Selective pulmonary vasorelaxant effects of an N2,N4-diaminoquinazoline PDE5 inhibitor involving endothelial signaling and ion channel modulationN2,N4-二氨基喹唑啉类PDE5抑制剂的选择性肺血管舒张作用涉及内皮信号传导和离子通道调节
errEuropean Journal of Pharmacology
IF4.7
err2026-07-17
err0
PREAI
errUsana Chatturong; Tipparat Meebangsue; Guntur Guntur; M. Paul Gleeson; Krongkarn Chootip
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Computationally guided optimization of the antimalarial activity and physicochemical properties of 2; 4-diaminopyrimidines计算指导下的2;4-二氨基嘧啶的抗疟活性与理化性质优化
errRSC Med. Chem.
IF3.6
err2025-08-22
err0
PREAI
errGuntur Guntur; Duangkamol Gleeson; Mark Anderson; Nicole Mutter; Lauren Webster; Kevin D. Read; M. Paul Gleeson
err分享
err收藏
Synthesis of Functionalized Benzo[h]Quinolines via Base-Catalyzed 1,4-Addition/Intramolecular Annulation Cascade通过碱催化的1,4-加成/分子内环化串联反应合成功能化苯并[h]喹啉
errChemistry – An Asian Journal
IF0
err2025-06-23
err0
PREAI
errDr. Wannaporn Disadee; Assoc. Prof. Dr. M. Paul Gleeson; Prof. Dr. Em. Somsak Ruchirawat
err分享
err收藏
Probing the Effect of Protein and Inhibitor Conformational Flexibility on the Reaction of Rocelitinib-Like Covalent Inhibitors of Epidermal Growth Factor Receptor. A Quantum Mechanics/Molecular Mechanics Study探究蛋白质和抑制剂构象柔韧性对表皮生长因子受体罗塞替尼样共价抑制剂反应的影响：一项量子力学/分子力学研究
errJOURNAL OF CHEMICAL INFORMATION AND MODELING
IF5.3
err2025-03-18
err0
errOAAI
errKaewkham, Orathai; Gleeson, Duangkamol; Fukasem, Poowadon; Santatiwongchai, Jirapat; Jones, Donald J. L.; Britton, Robert G.; Gleeson, M. Paul
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Design, preparation and biological evaluation of new Rociletinib-inspired analogs as irreversible EGFR inhibitors to treat non-small-cell-lung cancer
errBIOORGANIC & MEDICINAL CHEMISTRY
IF3
err2024-11-01
err1
PREAI
errKonsue, Adchata; Lamtha, Thomanai; Gleeson, Duangkamol; Jones, Donald J. L.; Britton, Robert G.; Pickering, James D.; Choowongkomon, Kiattawee; Gleeson, M. Paul
err分享
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Estimation of the Skin Sensitization Potential of Chemicals of the Acyl Domain Using DFT-Based Calculations
errCHEMICAL RESEARCH IN TOXICOLOGY
IF3.8
err2024-10-19
err0
PREAI
errLimluan, Pichayapa; Gleeson, M. Paul; Gleeson, Duangkamol
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Comparison of feline and human immunodeficiency virus reverse transcriptase enzymes through chemical screening and computational analysis
errCHEMICAL BIOLOGY & DRUG DESIGN
IF3.3
err2024-05-09
err0
PREAI
errThammajong, Phanicha; Aiebchun, Thitinan; Boonyarattanakalin, Kanokthip; Gleeson, Duangkamol; Pobsuk, Nattakarn; Hannongbua, Supa; Choowongkomon, Kiattawee; Gleeson, M. Paul
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The new quinazoline derivative (N2-methyl-N4-[(thiophen-2-yl)methyl] quinazoline-2,4-diamine) vasodilates isolated mesenteric arteries through endothelium-independent mechanisms and has acute hypotensive effects in Wistar rats
errEUROPEAN JOURNAL OF PHARMACOLOGY
IF4.7
err2023-08-01
err4
PREAI
errChatturong, Usana; Chootip, Krongkarn; Martin, Helene; Tournier-Nappey, Maude; Ingkaninan, Kornkanok; Temkitthawon, Prapapan; Sermsenaphorn, Saharat; Somarin, Thanachon; Konsue, Adchatawut; Gleeson, M. Paul; Totoson, Perle; Demougeot, Celine
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Quinazoline-based human phosphodiesterase 5 inhibitors exhibited a selective vasorelaxant effect on rat isolated pulmonary arteries involving NO-sGC-cGMP pathway and calcium inhibitory effects
errVASCULAR PHARMACOLOGY
IF3.5
err2022-12-01
err3
PREAI
errChatturong, Usana; Martin, Helene; Totoson, Perle; Ingkaninan, Kornkanok; Temkitthawon, Prapapan; Sermsenaphorn, Saharat; Somarin, Thanachon; Konsue, Adchatawut; Gleeson, M. Paul; Demougeot, Celine; Chootip, Krongkarn
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Computational design, synthesis and biological evaluation of PDE5 inhibitors based on N2,N4-diaminoquinazoline and N2, N6-diaminopurine scaffolds
errBIOORGANIC & MEDICINAL CHEMISTRY
IF3
err2022-12-01
err4
PREAI
errSomnarin, Thanachon; Pobsuk, Nattakarn; Chantakul, Ruttanaporn; Panklai, Teerapap; Temkitthawon, Prapapan; Hannongbua, Supa; Chootip, Krongkarn; Ingkaninan, Kornkanok; Boonyarattanakalin, Kanokthip; Gleeson, Duangkamol; Gleeson, M. Paul
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DFT Investigation of the catalytic conversion of acetic acid to acetone on the zeolite H-ZSM5
errMOLECULAR CATALYSIS
IF4.9
err2022-12-01
err5
PREAI
errKonsue, Adchatawut; Gleeson, M. Paul; Gleeson, Duangkamol
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Computational investigation of the radical-mediated mechanism of formation of difluoro methyl oxindoles: Elucidation of the reaction selectivity and yields
errJOURNAL OF COMPUTATIONAL CHEMISTRY
IF4.8
err2022-11-18
err0
PREAI
errSomnarin, Thanachon; Krawmanee, Pacharaporn; Gleeson, Matthew Paul; Gleeson, Duangkamol
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4-Aryl-N-phenylpyrimidin-2-amines targeting EGFR-tyrosine kinase attenuated EGFR-expressing cell lines
errEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY REPORTS
IF4.1
err2022-08-01
err2
errOAAI
errTabtimmai, Lueacha; Supakun, Prapasri; Toviwek, Borvornvat; Jiwacharoenchai, Nattanan; Kiriwan, Duangnapa; Aiebchun, Thitinan; Gleeson, M. Paul; Choowongkomon, Kiattawee
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Circular Polarization Conversion in Single Plasmonic Spherical Particles
errNANO LETTERS
IF9.1
err2022-02-03
err3
errOAAI
errKhan, Pritam; Brennan, Grace; Li, Zhe; Al Hassan, Luluh; Rice, Daragh; Gleeson, Matthew; Mani, Aladin A.; Tofail, Syed A. M.; Xu, Hongxing; Liu, Ning; Silien, Christophe
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Preparation, biological evaluation and QSAR analysis of urea substituted 2,4-diamino-pyrimidine anti-malarials
errRSC MEDICINAL CHEMISTRY
IF3.6
err2022-01-01
err5
errOAAI
errToviwek, Borvornwat; Riley, Jennifer; Mutter, Nicole; Anderson, Mark; Webster, Lauren; Hallyburton, Irene; Gleeson, Duangkamol; Read, Kevin D.; Gleeson, M. Paul
err分享
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A Piezoelectric Ionic Cocrystal of Glycine and Sulfamic Acid
errCRYSTAL GROWTH & DESIGN
IF3.4
err2021-09-27
err25
errOAAI
errGuerin, Sarah; Khorasani, Sanaz; Gleeson, Matthew; O'Donnell, Joseph; Sanii, Rana; Zwane, Reabetswe; Reilly, Anthony M.; Silien, Christophe; Tofail, Syed A. M.; Liu, Ning; Zaworotko, Michael; Thompson, Damien
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Preparation, biological & cheminformatics-based assessment of N2, N4-diphenylpyrimidine-2,4-diamine as potential Kinase-targeted antimalarials
errBIOORGANIC & MEDICINAL CHEMISTRY
IF3
err2021-09-01
err9
PREAI
errToviwek, Borvornwat; Phuangsawai, Oraphan; Konsue, Adchatawut; Hannongbua, Supa; Riley, Jennifer; Mutter, Nicole; Anderson, Mark; Webster, Lauren; Hallyburton, Irene; Read, Kevin D.; Gleeson, M. Paul
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Quantitative Polarization-Resolved Second-Harmonic-Generation Microscopy of Glycine Microneedles
errADVANCED MATERIALS
IF26.8
err2020-10-14
err13
PREAI
errGleeson, Matthew; O'Dwyer, Kevin; Guerin, Sarah; Rice, Daragh; Thompson, Damien; Tofail, Syed A. M.; Silien, Christophe; Liu, Ning
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Towards reproducible computational drug discovery走向可重复的计算药物发现
errJOURNAL OF CHEMINFORMATICS
IF5.7
err2020-01-28
err116
errOAAI
errSchaduangrat, Nalini; Lampa, Samuel; Simeon, Saw; Gleeson, Matthew Paul; Spjuth, Ola; Nantasenamat, Chanin
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研究方向

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