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Ajiroghene Thomas

University of Camerino

H指数:14

被引数:497

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Imidazo[1,2-a]pyrazin-8-amine core for the design of new adenosine receptor antagonists: Structural exploration to target the A3 and A2A subtypes

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2017-01-0119

OAAI

Overview on Radiolabel-Free in vitro Assays for GPCRs

MINI-REVIEWS IN MEDICINAL CHEMISTRY

IF3.3

2016-11-185

OA

The G Protein-Coupled Receptor GPR17: Overview and Update

G蛋白偶联受体GPR17: 概述和更新

IF3.4

2016-11-1436

OAAI

2',3'-O-Substituted ATP derivatives as potent antagonists of purinergic P2X3 receptors and potential analgesic agents

PURINERGIC SIGNALLING

IF2.4

2016-10-1812

OAAI

The Length and Flexibility of the 2-Substituent of 9-Ethyladenine Derivatives Modulate Affinity and Selectivity for the Human A2A Adenosine Receptor

IF3.4

2016-04-0113

OA

A Novel Class of Dopamine D4 Receptor Ligands Bearing an Imidazoline Nucleus

IF3.4

2016-03-157

OA

Exploring the 7-oxo-thiazolo[5,4-d]pyrimidine core for the design of new human adenosine A3 receptor antagonists. Synthesis, molecular modeling studies and pharmacological evaluation

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2015-05-0124

PREAI

Medicinal Chemistry of P2X Receptors: Agonists and Orthosteric Antagonists

CURRENT MEDICINAL CHEMISTRY

IF3.5

2015-02-0248

PRE

Purinergic P2X receptors: Structural models and analysis of ligand-target interaction

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2015-01-0143

PREAI

1,2,4-Triazolo[1,5-a]quinoxaline derivatives and their simplified analogues as adenosine A3 receptor antagonists. Synthesis, structure-affinity relationships and molecular modeling studies

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2015-01-0122

OAAI

Different efficacy of adenosine and NECA derivatives at the human A3 adenosine receptor: Insight into the receptor activation switch

BIOCHEMICAL PHARMACOLOGY

IF5.6

2014-01-0122

PREAI

8-(2-Furyl)adenine derivatives as A2A adenosine receptor ligands

8-(2-呋喃基) 腺嘌呤衍生物作为A2A腺苷受体配体

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2013-12-0116

PREAI

Evaluation of adenine as scaffold for the development of novel P2X3 receptor antagonists

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2013-07-017

PREAI

Innovative functional cAMP assay for studying G protein-coupled receptors: application to the pharmacological characterization of GPR17

PURINERGIC SIGNALLING

IF2.4

2011-07-2048

OA

Evidence for the Existence of a Specific G Protein-Coupled Receptor Activated by Guanosine

IF3.4

2011-04-1546

PREAI

Neuropeptide S Receptor: Recent Updates on Nonpeptide Antagonist Discovery

IF3.4

2011-03-3012

PREAI

Molecular modeling study on potent and selective adenosine A3 receptor agonists

强效选择性腺苷A3受体激动剂的分子模拟研究

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2010-11-1525

PRE