未登录G9a/DNMT1 co-targeting inhibits non-small cell lung cancer growth and reprograms tumor cells to respond to cancer-drugs through SCARA5 and AOX1
Exposito, Francisco; Redrado, Miriam; Serrano, Diego; Calabuig-Farinas, Silvia; Bao-Caamano, Aida; Gallach, Sandra; Jantus-Lewintre, Eloisa; Diaz-Lagares, Angel; Rodriguez-Casanova, Aitor; Sandoval, Juan; San Jose-Eneriz, Edurne; Garcia, Javier; Redin, Esther; Senent, Yaiza; Leon, Sergio; Pio, Ruben; Lopez, Rafael; Oyarzabal, Julen; Pineda-Lucena, Antonio; Agirre, Xabier; Montuenga, Luis M.; Prosper, Felipe; Calvo, Alfonso
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收藏Epigenetic-based differentiation therapy for Acute Myeloid Leukemia
San Jose-Eneriz, Edurne; Gimenez-Camino, Naroa; Rabal, Obdulia; Garate, Leire; Miranda, Estibaliz; Gomez-Echarte, Nahia; Garcia, Fernando; Charalampopoulou, Stella; Saez, Elena; Vilas-Zornoza, Amaia; San Martin-Uriz, Patxi; Valcarcel, Luis V.; Barrena, Naroa; Alignani, Diego; Tamariz-Amador, Luis Esteban; Perez-Ruiz, Ana; Hilscher, Sebastian; Schutkowski, Mike; Alfonso-Pierola, Ana; Martinez-Calle, Nicolas; Larrayoz, Maria Jose; Paiva, Bruno; Calasanz, Maria Jose; Munoz, Javier; Isasa, Marta; Martin-Subero, Jose Ignacio; Pineda-Lucena, Antonio; Oyarzabal, Julen; Agirre, Xabier; Prosper, Felipe
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收藏CM-352 Efficacy in a Mouse Model of Anticoagulant-Associated Intracranial Hemorrhage
Navarro-Oviedo, Manuel; Marta-Enguita, Juan; Roncal, Carmen; Rodriguez, Jose A.; Zandio, Beatriz; Lecumberri, Ramon; Hermida, Jose; Oyarzabal, Julen; Pineda-Lucena, Antonio; Paramo, Jose A.; Munoz, Roberto; Orbe, Josune
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收藏Omipalisib inspired macrocycles as dual PI3K/mTOR inhibitors (vol 211, 113109, 2021)
Alvarez, Rosa M.; Garcia, Ana Belen; Riesco-Fagundo, Concepion; Martin, Jose I.; Varela, Carmen; Hergueta, Antonio Rodriguez; Cantalapiedra, Esther Gonzalez; Oyarzabal, Julen; Di Geronimo, Bruno; Lorenzo, Milagros; Albarran, M. Isabel; Cebria, Antonio; Cebrian, David; Martinez-Gonzalez, Sonia; Blanco-Aparicio, Carmen; Pastor, Joaquin
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收藏mRNA-based therapy in a rabbit model of variegate porphyria offers new insights into the pathogenesis of acute attacks
Jerico, Daniel; Cordoba, Karol M.; Jiang, Lei; Schmitt, Caroline; Moran, Maria; Sampedro, Ana; Alegre, Manuel; Collantes, Maria; Santamaria, Eva; Alegre, Estibaliz; Culerier, Corinne; de Mendoza, Ander Estella-Hermoso; Oyarzabal, Julen; Penuelas, Ivan; Martin, Miguel A.; avila, Matias A.; Gouya, Laurent; Martini, Paolo G. V.; Fontanellas, Antonio
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收藏Dual Targeting of G9a and DNA Methyltransferase-1 for the Treatment of Experimental Cholangiocarcinoma
Colyn, Leticia; Barcena-Varela, Marina; Alvarez-Sola, Gloria; Ujue Latasa, M.; Uriarte, Iker; Santamaria, Eva; Herranz, Jose M.; Santos-Laso, Alvaro; Arechederra, Maria; Ruiz de Gauna, Mikel; Aspichueta, Patricia; Canale, Matteo; Casadei-Gardini, Andrea; Francesconi, Maria; Carotti, Simone; Morini, Sergio; Nelson, Leonard J.; Iraburu, Maria J.; Chen, Chaobo; Sangro, Bruno; Marin, Jose J. G.; Martinez-Chantar, Maria L.; Banales, Jesus M.; Arnes-Benito, Robert; Huch, Meritxell; Patino, John M.; Dar, Altaf A.; Nosrati, Mehdi; Oyarzabal, Julen; Prosper, Felipe; Urman, Jesus; Javier Cubero, Francisco; Trautwein, Christian; Berasain, Carmen; Fernandez-Barrena, Maite G.; Avila, Matias A.
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收藏Design and Synthesis of Novel Epigenetic Inhibitors Targeting Histone Deacetylases, DNA Methyltransferase 1, and Lysine Methyltransferase G9a with In Vivo Efficacy in Multiple Myeloma
Rabal, Obdulia; San Jose-Eneriz, Edurne; Agirre, Xabier; Antonio Sanchez-Arias, Juan; de Miguel, Irene; Ordonez, Raquel; Garate, Leire; Miranda, Estibaliz; Saez, Elena; Vilas-Zornoza, Amaia; Pineda-Lucena, Antonio; Estella, Ander; Zhang, Feifei; Wu, Wei; Xu, Musheng; Prosper, Felipe; Oyarzabal, Julen
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收藏Searching for Peptide Inhibitors of T Regulatory Cell Activity by Targeting Specific Domains of FOXP3 Transcription Factor
Lozano, Teresa; Casares, Noelia; Martil-Otal, Celia; Anega, Blanca; Gorraiz, Marta; Parker, Jonathan; Ruiz, Marta; Belsue, Virginia; Pineda-Lucena, Antonio; Oyarzabal, Julen; Lasarte, Juan Jose
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收藏Omipalisib inspired macrocycles as dual PI3K/mTOR inhibitors
Alvarez, Rosa M.; Belen Garcia, Ana; Riesco-Fagundo, Concepcion; Martin, Jose, I; Varela, Carmen; Rodriguez Hergueta, Antonio; Gonzalez Cantalapiedra, Esther; Oyarzabal, Julen; Di Geronimo, Bruno; Lorenzo, Milagros; Isabel Albarran, M.; Cebria, Antonio; Cebrian, David; Martinez-Gonzalez, Sonia; Blanco-Aparicio, Carmen; Pastor, Joaquin
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收藏Targeting aberrant DNA methylation in mesenchymal stromal cells as a treatment for myeloma bone disease
Garcia-Gomez, Antonio; Li, Tianlu; de la Calle-Fabregat, Carlos; Rodriguez-Ubreva, Javier; Ciudad, Laura; Catala-Moll, Francesc; Godoy-Tena, Gerard; Martin-Sanchez, Montserrat; San-Segundo, Laura; Muntion, Sandra; Morales, Xabier; Ortiz-de-Solorzano, Carlos; Oyarzabal, Julen; San Jose-Eneriz, Edurne; Esteller, Manel; Agirre, Xabier; Prosper, Felipe; Garayoa, Mercedes; Ballestar, Esteban
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收藏Endogenous Retroelement Activation by Epigenetic Therapy Reverses the Warburg Effect and Elicits Mitochondrial-Mediated Cancer Cell Death
Fresquet, Vicente; Garcia-Barchino, Maria J.; Larrayoz, Marta; Celay, Jon; Vicente, Carmen; Fernandez-Galilea, Marta; Larrayoz, Maria J.; Calasanz, Maria J.; Panizo, Carlos; Junza, Alexandra; Han, Jiahuai; Prior, Celia; Fortes, Puri; Pio, Ruben; Oyarzabal, Julen; Martinez-Baztan, Alvaro; Paiva, Bruno; Moreno-Aliaga, Maria J.; Odero, Maria D.; Agirre, Xabier; Yanes, Oscar; Prosper, Felipe; Martinez-Climent, Jose A.
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收藏2-Oxaadamant-1-yl Ureas as Soluble Epoxide Hydrolase Inhibitors: In Vivo Evaluation in a Murine Model of Acute Pancreatitis
Codony, Sandra; Pujol, Eugenia; Pizarro, Javier; Feixas, Ferran; Valverde, Elena; Isabel Loza, M.; Brea, Jose M.; Saez, Elena; Oyarzabal, Julen; Pineda-Lucena, Antonio; Perez, Belen; Perez, Concepcion; Isabel Rodriguez-Franco, Maria; Leiva, Rosana; Osuna, Silvia; Morisseau, Christophe; Hammock, Bruce D.; Vaquez-Carrera, Manuel; Vazquez, Santiago
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收藏A novel FTY720 analogue targets SET-PP2A interaction and inhibits growth of acute myeloid leukemia cells without inducing cardiac toxicity
Vicente, Carmen; Arriazu, Elena; Martinez-Balsalobre, Elena; Peris, Irene; Marcotegui, Nerea; Garcia-Ramirez, Patricia; Pippa, Raffaella; Rabal, Obdulia; Oyarzabal, Julen; Guruceaga, Elizabeth; Prosper, Felipe; Mateos, Maria C.; Cayuela, Maria L.; Odero, Maria D.
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收藏Trimethylamine-N-Oxide (TMAO) Predicts Cardiovascular Mortality in Peripheral Artery Disease
Roncal, Carmen; Martinez-Aguilar, Esther; Orbe, Josune; Ravassa, Susana; Fernandez-Montero, Alejandro; Saenz-Pipaon, Goren; Ugarte, Ana; Estella-Hermoso de Mendoza, Ander; Rodriguez, Jose A.; Fernandez-Alonso, Sebastian; Fernandez-Alonso, Leopoldo; Oyarzabal, Julen; Paramo, Jose A.
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收藏Multitarget Approach for the Treatment of Alzheimer's Disease: Inhibition of Phosphodiesterase 9 (PDE9) and Histone Deacetylases (HDACs) Covering Diverse Selectivity Profiles
Rabal, Obdulia; Sanchez-Arias, Juan A.; Cuadrado-Tejedor, Mar; de Miguel, Irene; Perez-Gonzalez, Marta; Garcia-Barroso, Carolina; Ugarte, Ana; Estella-Hermoso de Mendoza, Ander; Saez, Elena; Espelosin, Maria; Ursua, Susana; Tan, Haizhong; Wu, Wei; Xu, Musheng; Pineda-Lucena, Antonio; Garcia-Osta, Ana; Oyarzabal, Julen
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收藏Inhibition of a G9a/DNMT network triggers immune-mediated bladder cancer regression
Segovia, Cristina; San Jose-Eneriz, Edurne; Munera-Maravilla, Ester; Martinez-Fernandez, Monica; Garate, Leire; Miranda, Estibaliz; Vilas-Zornoza, Amaia; Lodewijk, Iris; Rubio, Carolina; Segrelles, Carmen; Vitores Valcarcel, Luis; Rabal, Obdulia; Casares, Noelia; Bernardini, Alejandra; Suarez-Cabrera, Cristian; Lopez-Calderon, Fernando F.; Fortes, Puri; Casado, Jose A.; Duenas, Marta; Villacampa, Felipe; Jose Lasarte, Juan; Guerrero-Ramos, Felix; de Velasco, Guillermo; Oyarzabal, Julen; Castellano, Daniel; Agirre, Xabier; Prosper, Felipe; Paramio, Jesus M.
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收藏Taking Advantage of the Selectivity of Histone Deacetylases and Phosphodiesterase Inhibitors to Design Better Therapeutic Strategies to Treat Alzheimer's Disease
Cuadrado-Tejedor, Mar; Perez-Gonzalez, Marta; Garcia-Munoz, Cristina; Muruzabal, Damian; Garcia-Barroso, Carolina; Rabal, Obdulia; Segura, Victor; Sanchez-Arias, Juan A.; Oyarzabal, Julen; Garcia-Osta, Ana
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收藏Discovery of novel triazolo[4,3-b]pyridazin-3-yl-quinoline derivatives as PIM inhibitors
Martinez-Gonzalez, Sonia; Rodriguez-Aristegui, Sonsoles; Gomez de la Oliva, Cristina Ana; Isabel Hernandez, Ana; Gonzalez Cantalapiedra, Esther; Varela, Carmen; Belen Garcia, Ana; Rabal, Obdulia; Oyarzabal, Julen; Bischoff, James R.; Klett, Javier; Isabel Albarran, Maria; Cebria, Antonio; Ajenjo, Nuria; Garcia-Serelde, Beatriz; Gomez-Casero, Elena; Cuadrado-Urbano, Manuel; Cebrian, David; Blanco-Aparicio, Carmen; Pastor, Joaquin
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收藏Identification of new epigenetic targets in hepatic fibrosis
Barcena-Varela, Marina; Paish, Hannah; Alvarez, Laura; Oyarzabal, Julen; Prosper, Felipe; Mazza, Giuseppe; Rombouts, Krista; Oakley, Fiona; Mann, Jelena; Berasain, Carmen; Avila, Matias A.; Fernandez-Barrena, Maite G.
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