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Discovery of YJZ5118: A Potent and Highly Selective Irreversible CDK12/13 Inhibitor with Synergistic Effects in Combination with Akt Inhibition YJZ5118的发现:一种具有协同效应的强效且高度选择性的不可逆CDK12/13抑制剂,可与Akt抑制联合用药。 Yang, Jianzhang; Chang, Yu; Zhou, Kaijie; Huang, Weixue; Tien, Jean Ching-Yi; Zhang, Pujuan; Liu, Wenyan; Zhou, Licheng; Zhou, Yang; Ren, Xiaomei; Mannan, Rahul; Mahapatra, Somnath; Zhang, Yuping; Hamadeh, Rudana; Ervine, Grafton; Wang, Zhen; Wang, George Xiaoju; Chinnaiyan, Arul M.; Ding, Ke 分享 收藏
Discovery of the first potent ROR1 degrader for the treatment of non-small cell lung cancer Li, Jinlin; Li, Lin; Hou, Caiyun; Tian, Zhaodi; Zhou, Yang; Zhang, Jinwei; Ren, Xiaomei; Wang, Zhen; Huang, Weixue; Ding, Ke; Zhou, Fengtao 分享 收藏
Discovery of the first selective and potent PROTAC degrader for the pseudokinase TRIB2 假激酶TRIB2的第一个选择性和有效的PROTAC降解剂的发现 Wen, Chaowei; Gajjala, Prathibha R.; Liu, Yihan; Chen, Bingzhong; Bal, Mehtab S.; Sutaria, Payal; Qiao, Yuanyuan; Zheng, Yang; Zhou, Yang; Zhang, Jinwei; Huang, Weixue; Ren, Xiaomei; Wang, Zhen; Ding, Ke; Chinnaiyan, Arul M.; Zhou, Fengtao 分享 收藏
Structure-Based Design of Head-to-Tail Macrocyclic PROTACs Li, Chungen; Chen, Yihan; Huang, Weixue; Qiu, Yudi; Huang, Shengjie; Zhou, Yang; Zhou, Fengtao; Xu, Jian; Ren, Xiaomei; Zhang, Jinwei; Wang, Zhen; Ding, Ming; Ding, Ke 分享 收藏
Discovery of ZLC491 as a Potent, Selective, and Orally Bioavailable CDK12/13 PROTAC Degrader Zhou, Licheng; Zhou, Kaijie; Chang, Yu; Yang, Jianzhang; Fan, Bohai; Su, Yuhan; Li, Zilu; Mannan, Rahul; Mahapatra, Somnath; Ding, Ming; Zhou, Fengtao; Huang, Weixue; Ren, Xiaomei; Xu, Jian; Wang, George Xiaoju; Zhang, Jinwei; Wang, Zhen; Chinnaiyan, Arul M.; Ding, Ke 分享 收藏
RGT-264 a highly potent, selective and orally bioavailable HPK1 (MAP4K1) inhibitor augments immune activation and anti-tumor immunity Xiao, F.; Liu, H.; Wu, L.; Feng, S.; Liu, Y.; Xiao, H.; Li, H.; Huang, W.; Ren, X.; Ren, B.; Yao, L.; Lin, J.; Zhong, W.; Xie, Z. 分享 收藏
Analytical and clinical evaluation of a novel real-time PCR-based detection kit for Mpox virus Bunse, Till; Ziel, Anne; Hagen, Philipp; Rigopoulos, George; Yasar, Umit; Inan, Hakan; Koese, Gurbet; Eigner, Ulrich; Kaiser, Rolf; Bardeck, Nils; Koeffer, Jasmin; Kolb, Melissa; Ren, Xiaomei; Tan, Deyong; Dai, Lizhong; Protzer, Ulrike; Wettengel, Jochen M. 分享 收藏
Mechanisms of acquired resistance to HER2-Positive breast cancer therapies induced by HER3: A comprehensive review Geng, Wujun; Thomas, Holly; Chen, Zhiyuan; Yan, Zhixiu; Zhang, Pujuan; Zhang, Meiying; Huang, Weixue; Ren, Xiaomei; Wang, Zhen; Ding, Ke; Zhang, Jinwei 分享 收藏
Amine response smartphone-based portable and intelligent polyvinyl alcohol films for real-time detection of shrimp freshness 基于胺响应智能手机的便携式智能聚乙烯醇薄膜实时检测虾新鲜度 Luo, Man; Liu, Ji; Zhang, Yating; Wang, Tao; Ren, Xiaomei; Gui, Lijuan; Zhao, Junyuan; Zhang, Xuwei; Tang, Yunqing; Zeng, Ziting; Hou, Fengzhen; Zhong, Qifeng; Yuan, Zhenwei; Xu, Hui 分享 收藏
Discovery of LLC355 as an Autophagy-Tethering Compound for the Degradation of Discoidin Domain Receptor 1 Liu, Lianchao; Zhao, Lijie; Yang, Lujun; Chai, Minxue; Liu, Zhengyong; Ma, Nan; Wang, Yongxing; Wu, Qinxue; Guo, Jing; Zhou, Fengtao; Huang, Weixue; Ren, Xiaomei; Wang, Jian; Ding, Ming; Wang, Zhen; Ding, Ke 分享 收藏