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Paul L. Ornstein

Eli Lilly

47H指数
140论文数
6.7K被引数
收录论文 39
发表时间
Excellence in Medicinal Chemistry: Celebrating ACS Medicinal Chemistry Division (MEDI) Awards. A Call for Nominations
err2023-05-18
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errOAAI
errBlanco, Maria-Jesus; Bryant-Friedrich, Amanda; Georg, Gunda; Ali, Amjad; Ornstein, Paul L.; Ferrins, Lori; Trippier, Paul C.
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Excellence in Medicinal Chemistry: Celebrating ACS Medicinal Chemistry Division (MEDI) Awards. A Call for Nominations
err2023-05-18
err0
PREAI
errBlanco, Maria-Jesus; Bryant-Friedrich, Amanda; Georg, Gunda; Ali, Amjad; Ornstein, Paul L. L.; Ferrins, Lori; Trippier, Paul C. C.
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Novel Trifluoromethyl Pyrimidinone Compounds With Activity Against Mycobacterium tuberculosis
err2021-04-29
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errOAAI
errHembre, Erik; Early, Julie V.; Odingo, Joshua; Shelton, Catherine; Anoshchenko, Olena; Guzman, Junitta; Flint, Lindsay; Dennison, Devon; McNeil, Matthew B.; Korkegian, Aaron; Ovechkina, Yulia; Ornstein, Paul; Masquelin, Thierry; Hipskind, Philip A.; Parish, Tanya
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Modulation of TARP γ8-Containing AMPA Receptors as a Novel Therapeutic Approach for Chronic Pains
err2019-06-01
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errKnopp, Kelly L.; Simmons, Rosa Maria A.; Guo, Wenhong; Adams, Benjamin L.; Gardinier, Kevin M.; Gernert, Douglas L.; Ornstein, Paul L.; Porter, Warren; Reel, Jon; Ding, Chunjin; Wang, He; Qian, Yuewei; Burris, Kevin D.; Need, Anne; Barth, Vanessa; Swanson, Steven; Catlow, John; Witkin, Jeffrey M.; Zwart, Ruud; Sher, Emanuele; Choong, Kar-Chan; Wall, Theron M.; Schober, Douglas; Felder, Christian C.; Kato, Akihiko S.; Bredt, David S.; Nisenbaum, Eric S.
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The synthesis and evaluation of triazolopyrimidines as anti-tubercular agents三唑并嘧啶类抗结核药物的合成与评价
err2017-08-01
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errOAAI
errZuniga, Edison S.; Korkegian, Aaron; Mullen, Steven; Hembre, Erik J.; Ornstein, Paul L.; Cortez, Guillermo; Biswas, Kallolmay; Kumar, Naresh; Cramer, Jeffrey; Masquelin, Thierry; Hipskind, Philip A.; Odingo, Joshua; Parish, Tanya
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Comparative Effects of LY3020371, a Potent and Selective Metabotropic Glutamate (mGlu) 2/3 Receptor Antagonist, and Ketamine, a Noncompetitive N-Methyl-D-Aspartate Receptor Antagonist in Rodents: Evidence Supporting the Use of mGlu2/3 Antagonists, for the Treatment of Depression.
err2017-04-01
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errWitkin, J. M.; Mitchell, S. N.; Wafford, K. A.; Carter, G.; Gilmour, G.; Li, J.; Eastwood, B. J.; Overshiner, C.; Li, X.; Rorick-Kehn, L.; Rasmussen, K.; Anderson, W. H.; Nikolayev, A.; Tolstikov, V. V.; Kuo, M. -S.; Catlow, J. T.; Li, R.; Smith, S. C.; Mitch, C. H.; Ornstein, P. L.; Swanson, S.; Monn, J. A.
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Preclinical predictors that the orthosteric mGlu2/3 receptor antagonist LY3020371 will not engender ketamine-associated neurotoxic, motor, cognitive, subjective, or abuse-liability-related effects
err2017-04-01
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PREAI
errWitkin, J. M.; Monn, J. A.; Li, J.; Johnson, B.; McKinzie, D. L.; Wang, X-S; Heinz, B. A.; Li, R.; Ornstein, P. L.; Smith, S. C.; Mitch, C. H.; Calligaro, D. O.; Swanson, S.; Allen, D.; Phillips, K.; Gilmour, G.
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Discovery of (1S,2R,3S,4S,5R,6R)-2-Amino-3-[(3,4-difluorophenyl)sulfanylmethyl]-4-hydroxy-bicyclo[3.1.0]hexane-2,6-dicarboxylic Acid Hydrochloride (LY3020371•HCl): A Potent, Metabotropic Glutamate 2/3 Receptor Antagonist with Antidepressant-Like Activity
err2016-12-06
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errChappell, Mark D.; Li, Renhua; Smith, Stephon C.; Dressman, Bruce A.; Tromiczak, Eric G.; Tripp, Allie E.; Blanco, Maria-Jesus; Vetman, Tatiana; Quimby, Steven J.; Matt, James; Britton, Thomas C.; Fivush, Adam M.; Schkeryantz, Jeffrey M.; Mayhugh, Daniel; Erickson, Jon A.; Bures, Mark G.; Jaramillo, Carlos; Carpintero, Mercedes; Eugenio de Diego, Jose; Barberis, Mario; Garcia-Cerrada, Susana; Soriano, Jose F.; Antonysamy, Stephen; Atwell, Shane; MacEwan, Lain; Condon, Bradley; Sougias, Christine; Wang, Jing; Zhang, Aiping; Conners, Kris; Groshong, Chris; Wasserman, Stephen R.; Koss, John W.; Witkin, Jeffrey M.; Li, Xia; Overshiner, Carl; Wafford, Keith A.; Seidel, Wesley; Wang, Xu-Shan; Heinz, Beverly A.; Swanson, Steven; Catlow, John T.; Bedwell, David W.; Monn, James A.; Mitch, Charles H.; Ornstein, Paul L.
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Forebrain-selective AMPA-receptor antagonism guided by TARP γ-8 as an antiepileptic mechanism
err2016-11-07
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PREAI
errKato, Akihiko S.; Burris, Kevin D.; Gardinier, Kevin M.; Gernert, Douglas L.; Porter, Warren J.; Reel, Jon; Ding, Chunjin; Tu, Yuan; Schober, Douglas A.; Lee, Matthew R.; Heinz, Beverly A.; Fitch, Thomas E.; Gleason, Scott D.; Catlow, John T.; Yu, Hong; Fitzjohn, Stephen M.; Pasqui, Francesca; Wang, He; Qian, Yuewei; Sher, Emanuele; Zwart, Ruud; Wafford, Keith A.; Rasmussen, Kurt; Ornstein, Paul L.; Isaac, John T. R.; Nisenbaum, Eric S.; Bredt, David S.; Witkin, Jeffrey M.
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Discovery of the First α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor Antagonist Dependent upon Transmembrane AMPA Receptor Regulatory Protein (TARP) γ-8
err2016-04-29
err53
PREAI
errGardinier, Kevin M.; Gernert, Douglas L.; Porter, Warren J.; Reel, Jon K.; Ornstein, Paul L.; Spinazze, Patrick; Stevens, F. Craig; Hahn, Patric; Hollinshead, Sean P.; Mayhugh, Daniel; Schkeryantz, Jeff; Khilevich, Albert; De Frutos, Oscar; Gleason, Scott D.; Kato, Akihiko S.; Luffer-Atlas, Debra; Desai, Prashant V.; Swanson, Steven; Burris, Kevin D.; Ding, Chunjin; Heinz, Beverly A.; Need, Anne B.; Barth, Vanessa N.; Stephenson, Gregory A.; Diseroad, Benjamin A.; Woods, Tim A.; Yu, Hong; Bredt, David; Witkin, Jeffrey M.
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Transmembrane AMPA Receptor Regulatory Proteins and Cornichon-2 Allosterically Regulate AMPA Receptor Antagonists and Potentiators
err2011-04-01
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errSchober, Douglas A.; Gill, Martin B.; Yu, Hong; Gernert, Douglas L.; Jeffries, Matthew W.; Ornstein, Paul L.; Kato, Akihiko S.; Felder, Christian C.; Bredt, David S.
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A novel, competitive mGlu5 receptor antagonist (LY344545) blocks DHPG-induced potentiation of NMDA responses but not the induction of LTP in rat hippocampal slices
err2009-01-29
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errOAAI
errDoherty, AJ; Palmer, MJ; Bortolotto, ZA; Hargreaves, A; Kingston, AE; Ornstein, PL; Schoepp, DD; Lodge, D; Collingridge, GL
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Antiallodynic and antihyperalgesic effects of selective competitive GLUK5 (GluR5) ionotropic glutamate receptor antagonists in the capsaicin and carrageenan models in rats
err2006-10-01
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PREAI
errJones, Carrie K.; Alt, Andrew; Ogden, Ann Marie; Bleakman, David; Simmons, Rosa M. A.; Iyengar, Smriti; Dominguez, Esteban; Ornstein, Paul L.; Shannon, Harlan E.
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Pharmacological characterization of the competitive GLUK5 receptor antagonist decahydroisoquinoline LY466195 in vitro and in vivo
err2006-08-01
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PREAI
errWeiss, Brianne; Alt, Andrew; Ogden, Ann Marie; Gates, Mary; Dieckman, Donna K.; Clemens-Smith, Amy; Ho, Ken H.; Jarvie, Keith; Rizkalla, Geihan; Wright, Rebecca A.; Calligaro, David O.; Schoepp, Darryle; Mattiuz, Edward L.; Stratford, Robert E.; Johnson, Bryan; Salhoff, Craig; Katofiasc, Mary; Phebus, Lee A.; Schenck, Kathryn; Cohen, Marlene; Filla, Sandra A.; Ornstein, Paul L.; Johnson, Kirk W.; Bleakman, David
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Two prodrugs of potent and selective GluR5 kainate receptor antagonists actives in three animal models of pain
err2005-05-21
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PREAI
errDominguez, E; Iyengar, S; Shannon, HE; Bleakman, D; Alt, A; Arnold, BM; Bell, MG; Bleisch, TJ; Buckmaster, JL; Castano, AM; Del Prado, M; Escribano, A; Filla, SA; Ho, KH; Hudziak, KJ; Jones, CK; Martinez-Perez, JA; Mateo, A; Mathes, BM; Mattiuz, EL; Ogden, AML; Simmons, RMA; Stack, DR; Stratford, RE; Winter, MA; Wu, ZP; Ornstein, PL
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LY293558, a novel AMPA/GluR5 antagonist, is efficacious and well-tolerated in acute migraine
err2004-07-01
err143
PREAI
errSang, CN; Ramadan, NM; Wallihan, RG; Chappell, AS; Freitag, FG; Smith, TR; Silberstein, SD; Johnson, KW; Phebus, LA; Bleakman, D; Ornstein, PL; Arnold, B; Tepper, SJ; Vandenhende, F
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Synthesis and structure-activity relationships of novel arylpiperazines as potent and selective agonists of the melanocortin subtype-4 receptor
err2004-01-06
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PREAI
errRichardson, TI; Ornstein, PL; Briner, K; Fisher, MJ; Backer, RT; Biggers, CK; Clay, MP; Emmerson, PJ; Hertel, LW; Hsiung, HM; Husain, S; Kahl, SD; Lee, JA; Lindstrom, TD; Martinelli, MJ; Mayer, JP; Mullaney, JT; O'Brien, TP; Pawlak, JM; Revell, KD; Shah, J; Zgombick, JM; Herr, RJ; Melekhov, A; Sampson, PB; King, CHR
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A role for Ca2+ stores in kainate receptor-dependent synaptic facilitation and LTP at mossy fiber synapses in the hippocampus
errNEURON
IF15
err2003-07-01
err183
errOAAI
errLauri, SE; Bortolotto, ZA; Nistico, R; Bleakman, D; Ornstein, PL; Lodge, D; Isaac, JTR; Collingridge, GL
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