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Scholars864
Papers293
Citations0
Related Papers (291)
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Identification of the Piperidyl Urea Derivative BAY-439 as a Potent and Selective Inhibitor of Human Phospholipase A2 Group V (hPLA2-G5) for the Treatment of Inflammatory Pain
errJournal of Medicinal Chemistry
IF6.8
err2026-05-19
err0
PREAI
errGernot Langer; Nico Bräuer; Daryl Walter; Stuart Flanagan; Olivier Rémi Barbeau; Wei Tsung Yau; James Jenkins; Dennis Wegener; Daren Fearon; Anne-Marie Coelho; Benjamin Bader; Anders Friberg; Hartmut Beck; Vera Pütter; Frank Sacher
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PIP4K2A/2B inhibitor suppresses tumor growth in a xenograft model of NSCLC
erriScience
IF4.1
err2026-04-30
err0
errOAAI
errZunyu He; Song Chen; Marcus Bosenberg; Viswanathan Muthusamy; Yibo Xi; He Wang; Fabrizio Micheli; Agostino Cianciulli; Claudia Beato; Michael Van Zandt; Jonathan Ellman; Ya Ha
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Density-adjusted analysis of cell interactions to decipher tissue landscape changes
erriScience
IF4.1
err2026-04-21
err0
errOAAI
errMisha Siddiqui; Azam Hamidinekoo; Jennifer Y. Tan; Renata Leke; Bader Zarrouki; Nick Trahearn; Yeman Brhane Hagos; Chirine Sakr; Andrea Lampis; Christopher Bagnall; Giovanni Pellegrini; Simon P. Castillo; Benjamin Challis; Yinyin Yuan; Marco Bezzi; Stephanie Ling
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The magnitude of the pharmacodynamic index for NOSO-502: pathogen clearance, emergence of resistance and human dose predictions
errJournal of Antimicrobial Chemotherapy
IF3.6
err2026-04-01
err0
PREAI
errvan den Berg, Sanne; Attwood, Marie; Griffin, Pippa; Noel, Alan; Das, Shampa; Zeitlinger, Markus; Racine, Emilie; Boulenc, Xavier; Muller, Anouk E.; Sassen, Sebastiaan D. T.; Bahmany, Soma; ten Kate, Marian T.; MacGowan, Alasdair; Meletiadis, Joseph
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Repurposing drugs for treating the neurobehavioral manifestations of PTEN hamartoma tumor syndrome
erriScience
IF4.1
err2026-03-20
err0
errOAAI
errTim Fieblinger; Judith Rudolph; Kerstin Müller; Petra Friess; Nicole Weigelt; Christina Thiede; Simone Modolo; Denise Federico; Malik Majandinow; Federico Tinarelli; Vivian J.A. Costantini; Pier P. Marrese; Annalisa Mercuri; Nikisha Carty; Ana Christina Gomes; Maria A. Whitehead; Philip A. Gerrard; Chrisovalantis Papadopoulos; Paul Elvin
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Modulation of VHL binding affinity improves selectivity of PROTACs targeting BRM (SMARCA2) over BRG1 (SMARCA4)
errResults in Chemistry
IF4.2
err2026-03-01
err1
PREAI
errBerlin, Michael; Cantley, Jennifer; Broccatelli, Fabio; Cao, Lin; Chen, Huifen; Cheung, Tommy K.; Crew, Andrew P.; DiNicola, Dean; Dong, Hanqing; Grimmer, Matthew; Hamman, Brian D.; Harbin, Alicia; He, Mingtao; Hu, Xiuxian; Hole, Alison J.; Januario, Thomas; Kerry, Philip S.; Liu, Xiangjia; Quinn, Connor; Rose, Christopher M.; Rousseau, Emma; Snyder, Lawrence B.; Staben, Leanna R.; Wang, Gan; Wang, Jing; Ye, Xiaofen; Yauch, Robert L.; Dragovich, Peter S.
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Discovery of Potent PDE4 Inhibitors with 3(2H)-Pyridazinone Scaffold: Synthesis, In Silico Studies and In Vitro/Vivo Evaluation
errMolecules
IF4.6
err2026-02-17
err0
errOAAI
errVergelli, Claudia; Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Gracia, Jordi; Buil, Maria Antonia; Garrido, Yolanda; Pages, Lluis; Taltavull, Joan; Gavalda, Amadeu; Calama, Elena; Giovannoni, Maria Paola
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Discovery of Potent; Selective; and Brain-Penetrant Small Molecule CD38 Inhibitors
errACS Medicinal Chemistry Letters
IF4
err2026-01-29
err0
PREAI
errAndrew J. Stott; Roland W. Bürli; Kevin J. Doyle; Louise Dickson; Richard C. Hewer; Philip Pickford; Maxine J. Roberts; Rosie Waters-Hall; Yiming Wu; Matthias Zebisch; Victor Rangel; Matthis Geitmann; Kim Matthews; Nicola L. Brice; Mark Carlton; Lee A. Dawson; Jenna R. M. Harvey
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The COMBINE pneumonia model: a multicenter study to standardize a mouse pneumonia model with Pseudomonas aeruginosa and Klebsiella pneumoniae for antibiotic development
errMicrobiology Spectrum
IF3.8
err2026-01-01
err0
PREAI
errHansen, Jon U.; Arrazuria, Rakel; Hoover, Jennifer L.; Kerscher, Bernhard; Huseby, Douglas L.; Sordello, Sylvie; Gribbon, Philip; Gadiya, Yojana; Berlin, Leonie Von; Witt, Gesa; Tassi, Natalia; Rosenborg, Frederikke; Cao, Sha; Bekeredjian-Ding, Isabelle; Lindahl, Otto; Hughes, Diarmaid; Friberg, Lena E.; Vingsbo Lundberg, Carina
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Corrigendum to “Chronic cholesterol administration to the brain supports complete and long-lasting cognitive and motor amelioration in Huntington’s disease” [Pharmacol. Res. 194 (2023) 106823]
errPharmacological Research
IF10.5
err2025-10-21
err0
errOAAI
errGiulia Birolini; Marta Valenza; Ilaria Ottonelli; Francesca Talpo; Lucia Minoli; Andrea Cappelleri; Mauro Bombaci; Claudio Caccia; Caterina Canevari; Arianna Trucco; Valerio Leoni; Alice Passoni; Monica Favagrossa; Maria Rosaria Nucera; Laura Colombo; Saverio Paltrinieri; Renzo Bagnati; Jason Thomas Duskey; Riccardo Caraffi; Maria Angela Vandelli; Franco Taroni; Mario Salmona; Eugenio Scanziani; Gerardo Biella; Barbara Ruozi; Giovanni Tosi; Elena Cattaneo
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Every Compound a Candidate: experience-led risk-taking approaches to accelerate small-molecule drug discovery
errDRUG DISCOVERY TODAY
IF7.5
err2025-05-01
err0
PREAI
errMcginnity, Dermot F.; Meneyrol, Jerome; Boldron, Christophe; Johnstone, Craig
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Human cone photoreceptor transplantation stimulates remodeling and restores function in AIPL1 model of end-stage Leber congenital amaurosis
errSTEM CELL REPORTS
IF5.1
err2025-04-01
err0
errOAAI
errProcyk, Christopher A.; Melati, Anna; Ribeiro, Joana; Liu, Jingshu; Branch, Matthew J.; Delicata, Jamie D.; Tariq, Menahil; Kalarygrou, Aikaterini A.; Kapadia, Jessica; Khorsani, Majid Moshtagh; West, Emma L.; Smith, Alexander J.; Gonzalez-Cordero, Anai; Ali, Robin R.; Pearson, Rachael A.
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Mefloquine reduces the bacterial membrane fluidity of Acinetobacter baumannii and distorts the bacterial membrane when combined with polymyxin B
errMBIO
IF4.7
err2025-02-25
err0
errOAAI
errTharmalingam, Nagendran; Jayanthan, Harikrishna Sekar; Port, Jenna; Rossatto, Fernanda Cristina Possamai; Mylonakis, Eleftherios
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Quantum Mechanics-Based Ranking of Predicted Proteolysis Targeting Chimeras-Mediated Ternary Complexes
errACS MEDICINAL CHEMISTRY LETTERS
IF4
err2025-02-06
err1
PREAI
errMonteleone, Stefania; Morao, Inaki; Fedorov, Dmitri G.; Kellici, Tahsin F.
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Patients With Immunoglobulin A Nephropathy Show Abnormal Frequencies of B Cell Subsets , Unconventional T Cells, and High Levels of Galactose-Deficient IgA1-Coated Gut Bacteria
errKIDNEY INTERNATIONAL REPORTS
IF5.7
err2025-02-01
err1
errOAAI
errGentile, Micaela; Goerlich, Nina; Lo, I-Ju; Olson, N. Eric; Mcconnell, Mark; Pospiech, Johannes; Bohnenpoll, Tobias; Skroblin, Philipp; Radresa, Olivier; Andag, Uwe; Campbell, Kirk N.; Meliambro, Kristin; Sanchez-Russo, Luis; Verlato, Alberto; Fiaccadori, Enrico; Kim-Schulze, Seunghee; Lanau, Maria; Fernandez-Lorente, M. Loreto; Fribourg, Miguel; Manrique, Joaquin; Cravedi, Paolo
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Modeling Inflammatory Bowel Disease in mice with Humanized immune system
errJOURNAL OF CROHNS & COLITIS
IF8.7
err2025-01-22
err1
PREAI
errCoupe, B.; Charton, A.; Placide, F.; Machet, F.
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Validation framework for in vivo digital measures
errFRONTIERS IN TOXICOLOGY
IF4.6
err2025-01-08
err0
errOAAI
errBaran, Szczepan W.; Bolin, Susan E.; Gaburro, Stefano; van Gaalen, Marcel M.; La Follette, Megan R.; Liu, Chang-Ning; Maguire, Sean; Noldus, Lucas P. J. J.; Bratcher-Petersen, Natalie; Berridge, Brian R.
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Optimisation of a novel series of ENaC inhibitors, leading to the selection of the long-acting inhaled clinical candidate ETD001, a potential new treatment for cystic fibrosis
errEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
IF5.9
err2025-01-01
err0
PREAI
errDanahay, Henry; Gosling, Martin; Fox, Roy; Lilley, Sarah; Charlton, Holly; Hargrave, Jonathan D.; Schofield, Thomas B.; Hay, Duncan A.; Went, Naomi; McMahon, Pearl; Marlin, Frederic; Scott, John; Vile, Julia; Hewison, Steve; Ellam, Sarah; Brown, Samantha; Sabater, Juan; Kennet, Guy; Lightowler, Sean; Collingwood, Stephen P.
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ETD001: A novel inhaled ENaC blocker with an extended duration of action in vivo
errJOURNAL OF CYSTIC FIBROSIS
IF6
err2025-01-01
err2
PREAI
errDanahay, Henry; Mccarthy, Clive; Schofield, Thomas; Fox, Roy; Charlton, Holly; Lilley, Sarah; Sabater, Juan; Salathe, Matthias; Baumlin, Nathalie; Collingwood, Stephen P.; Gosling, Martin
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In Vivo Activity Profiling of Biosynthetic Darobactin D22 against Critical Gram-Negative Pathogens
errACS INFECTIOUS DISEASES
IF3.8
err2024-11-20
err1
errOAAI
errKany, Andreas M.; Fries, Franziska; Seyfert, Carsten E.; Porten, Christoph; Deckarm, Selina; Ortiz, Mariia Chacon; Dubarry, Nelly; Vaddi, Swapna; Grosse, Miriam; Bernecker, Steffen; Sandargo, Birthe; Muller, Alison V.; Bacque, Eric; Stadler, Marc; Herrmann, Jennifer; Muller, Rolf
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