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SaveDesign, synthesis, selection, and evaluation of a potent multi-kinase targeting N4-phenylsubstituted-7H-pyrrolo[2,3-d]pyrimidin-4-amine derivative with significant anticancer activity in P53 mutant and wild type models of upper gastrointestinal cancers
Samant, Amruta; Visal, Tanvi; Pancholi, Priya; Kansara, Dhvanir; Dichwalkar, Tanmay; Senones, Robert; Kurup, Sonali; Sehdev, Vikas
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SaveDesign, synthesis and biological activity of N4-phenylsubstituted-7H-pyrrolo[2,3-d]pyrimidin-4-amines as dual inhibitors of aurora kinase A and epidermal growth factor receptor kinase
Kurup, Sonali; McAllister, Bradley; Liskova, Pavlina; Mistry, Trusha; Fanizza, Anthony; Stanford, Dan; Slawska, Jolanta; Keller, Ulrich; Hoellein, Alexander
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SaveRS-41, a multi-targeted kinase inhibitor, induces cell cycle arrest and apoptosis in p53 mutant and wild type models of upper gastrointestinal cancers
Visal, Tanvi; Patel, Shraddha; Pancholi, Priya; Bapat, Samhita; Samant, Amruta; Kansara, Dhvanir; Kurup, Sonali; Sehdev, Vikas
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