Not logged inMonitoring drug-target interactions through target engagement-mediated amplification on arrays and in situ
Al-Amin, Rasel A.; Johansson, Lars; Abdurakhmanov, Eldar; Landegren, Nils; Lof, Liza; Arngarden, Linda; Blokzijl, Andries; Svensson, Richard; Hammond, Maria; Lonn, Peter; Haybaeck, Johannes; Kamali-Moghaddam, Masood; Jensen, Annika Jenmalm; Danielson, U. Helena; Artursson, Per; Lundback, Thomas; Landegren, Ulf
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SavePharmacological targeting of MTHFD2 suppresses acute myeloid leukemia by inducing thymidine depletion and replication stress
Bonagas, Nadilly; Gustafsson, Nina M. S.; Henriksson, Martin; Marttila, Petra; Gustafsson, Robert; Wiita, Elisee; Borhade, Sanjay; Green, Alanna C.; Vallin, Karl S. A.; Sarno, Antonio; Svensson, Richard; Gokturk, Camilla; Pham, Therese; Jemth, Ann-Sofie; Loseva, Olga; Cookson, Victoria; Kiweler, Nicole; Sandberg, Lars; Rasti, Azita; Unterlass, Judith E.; Haraldsson, Martin; Andersson, Yasmin; Scaletti, Emma R.; Bengtsson, Christoffer; Paulin, Cynthia B. J.; Sanjiv, Kumar; Abdurakhmanov, Eldar; Pudelko, Linda; Kunz, Ben; Desroses, Matthieu; Iliev, Petar; Farnegardh, Katarina; Kramer, Andreas; Garg, Neeraj; Michel, Maurice; Haggblad, Sara; Jarvius, Malin; Kalderen, Christina; Jensen, Amanda Bogedahl; Almlof, Ingrid; Karsten, Stella; Zhang, Si Min; Haggblad, Maria; Eriksson, Anders; Liu, Jianping; Glinghammar, Bjorn; Nekhotiaeva, Natalia; Klingegard, Fredrik; Koolmeister, Tobias; Martens, Ulf; Llona-Minguez, Sabin; Moulson, Ruth; Nordstrom, Helena; Parrow, Vendela; Dahllund, Leif; Sjoberg, Birger; Vargas, Irene L.; Vo, Duy Duc; Wannberg, Johan; Knapp, Stefan; Krokan, Hans E.; Arvidsson, Per, I; Scobie, Martin; Meiser, Johannes; Stenmark, Pal; Berglund, Ulrika Warpman; Homan, Evert J.; Helleday, Thomas
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SaveUltralarge Virtual Screening Identifies SARS-CoV-2 Main Protease Inhibitors with Broad-Spectrum Activity against Coronaviruses
Luttens, Andreas; Gullberg, Hjalmar; Abdurakhmanov, Eldar; Duy Duc Vo; Akaberi, Dario; Talibov, Vladimir O.; Nekhotiaeva, Natalia; Vangeel, Laura; De Jonghe, Steven; Jochmans, Dirk; Krambrich, Janina; Tas, Ali; Lundgren, Bo; Gravenfors, Ylva; Craig, Alexander J.; Atilaw, Yoseph; Sandstrom, Anja; Moodie, Lindon W. K.; Lundkvist, Ake; van Hemert, Martijn J.; Neyts, Johan; Lennerstrand, Johan; Kihlberg, Jan; Sandberg, Kristian; Danielson, U. Helena; Carlsson, Jens
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SaveDiscovery of pyrazinone based compounds that potently inhibit the drug-resistant enzyme variant R155K of the hepatitis C virus NS3 protease
Belfrage, Anna Karin; Abdurakhmanov, Eldar; Akerblom, Eva; Brandt, Peter; Oshalim, Anna; Gising, Johan; Skogh, Anna; Neyts, Johan; Danielson, U. Helena; Sandstrom, Anja
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