Not logged inSynthesis, Anti-HBV, and Anti-HIV Activities of 3′-Halogenated Bis(hydroxymethyl)-cyclopentenyladenines
Kumamoto, Hiroki; Imoto, Shuhei; Amano, Masayuki; Kuwata-Higashi, Nobuyo; Baba, Masanori; Mitsuya, Hiroaki; Odanaka, Yuki; Matsubayashi, Satoko Shimbara; Tanaka, Hiromichi; Haraguchi, Kazuhiro
Share
Save
Share
SaveSynthesis of 3′,4′-difluoro-3′-deoxyribonucleosides and its evaluation of the biological activities: Discovery of a novel type of anti-HCV agent 3′,4′-difluorocordycepin
Shimada, Hisashi; Haraguchi, Kazuhiro; Hotta, Kumi; Miyaike, Tomoko; Kitagawa, Yasuyuki; Tanaka, Hiromichi; Kaneda, Ryutaro; Abe, Hiroshi; Shuto, Satoshi; Mori, Kyoko; Ueda, Youki; Kato, Nobuyuki; Snoeck, Robert; Andrei, Graciela; Balzarini, Jan
Share
SaveTuning efficiency of the 4-exo-trig cyclization by the electronic effect: ring closure of 3,3-difluoro-4-pentenyl carbon radicals and synthesis of a gem-difluorocyclobutane nucleoside
Kumamoto, Hiroki; Kawahigashi, Sachiko; Wakabayashi, Hiromi; Nakano, Tomohiko; Miyaike, Tomoko; Kitagawa, Yasuyuki; Abe, Hiroshi; Ito, Mika; Haraguchi, Kazuhiro; Balzarini, Jan; Baba, Masanori; Tanaka, Hiromichi
Share
Save
Share
Save
Share
SaveSynthesis of 4′-Ethynyl-2′-deoxy-4′-thioribonucleosides and Discovery of a Highly Potent and Less Toxic NRTI
Haraguchi, Kazuhiro; Shimada, Hisashi; Kimura, Keigo; Akutsu, Genta; Tanaka, Hiromichi; Abe, Hiroshi; Hamasaki, Takayuki; Baba, Masanori; Gullen, Elizabeth A.; Dutschman, Ginger E.; Cheng, Yung-Chi; Balzarini, Jan
Share
Save
Share
SaveImpact of Novel Human Immunodeficiency Virus Type 1 Reverse Transcriptase Mutations P119S and T165A on 4′-Ethynylthymidine Analog Resistance Profile
Yang, Guangwei; Paintsil, Elijah; Dutschman, Ginger E.; Grill, Susan P.; Wang, Chuan-Jen; Wang, Jimin; Tanaka, Hiromichi; Hamasaki, Takayuki; Baba, Masanori; Cheng, Yung-Chi
Share
Save
Share
Save
Share
Save
Share
Save
Share
Save
Share
SaveIntracellular metabolism and persistence of the anti-human immunodeficiency virus activity of 2',3'-didehydro-3'-deoxy-4'-ethynylthymidine, a novel thymidine analog
Paintsil, Elijah; Dutschman, Ginger E.; Hu, Rong; Grill, Susan P.; Lam, Wing; Baba, Masanori; Tanaka, Hiromichi; Cheng, Yung-Chi
Share
Save
Share
Save
Share
Save
Share
Save
Share
Save
Share
Save