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Andrea Scozzafava

university of florence

115H-index
827Paper Count
4.6WCitation Count
Published Papers 300
Publication Date
Dioxygen, an unexpected carbonic anhydrase ligand
err2018-05-28
err14
errOAAI
errFerraroni, Marta; Gaspari, Roberto; Scozzafava, Andrea; Cavalli, Andrea; Supuran, Claudiu T.
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Discovery of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Management of Rheumatoid Arthritis
err2018-05-10
err48
PREAI
errAkgul, Ozlem; Mannelli, Lorenzo Di Cesare; Vullo, Daniela; Angeli, Andrea; Ghelardini, Carla; Bartolucci, Gianluca; Altamimi, Abdulmalik Saleh Alfawaz; Scozzafava, Andrea; Supuran, Claudiu T.; Carta, Fabrizio
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Sulphonamide inhibition studies of the β-carbonic anhydrase from the bacterial pathogen Clostridium perfringens
err2017-11-03
err20
errOAAI
errVullo, Daniela; Kumar, R. Siva Sai; Scozzafava, Andrea; Ferry, James G.; Supuran, Claudiu T.
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1,3-Oxazole-based selective picomolar inhibitors of cytosolic human carbonic anhydrase II alleviate ocular hypertension in rabbits: Potency is supported by X-ray crystallography of two leads
err2017-09-01
err12
PREAI
errFerraroni, Marta; Lucarini, Laura; Masini, Emanuela; Korsakov, Mikhail; Scozzafava, Andrea; Supuran, Claudiu T.; Krasavin, Mikhail
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Design and Synthesis of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Treatment of Rheumatoid Arthritis
err2017-01-23
err111
PREAI
errBua, Silvia; Mannelli, Lorenzo Di Cesare; Vullo, Daniela; Ghelardini, Carla; Bartolucci, Gianluca; Scozzafava, Andrea; Supuran, Claudiu T.; Carta, Fabrizio
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Polyamines and α-Carbonic Anhydrases
err2016-12-15
err10
errOAAI
errScozzafava, Andrea; Supuran, Claudiu T.; Carta, Fabrizio
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Kinetic and X-ray crystallographic investigations of substituted 2-thio-6-oxo-1,6-dihydropyrimidine-benzenesulfonamides acting as carbonic anhydrase inhibitors
err2016-08-01
err18
PREAI
errVullo, Daniela; Supuran, Claudiu T.; Scozzafava, Andrea; De Simone, Giuseppina; Monti, Simona Maria; Alterio, Vincenzo; Carta, Fabrizio
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Monothiocarbamates Strongly Inhibit Carbonic Anhydrases in Vitro and Possess Intraocular Pressure Lowering Activity in an Animal Model of Glaucoma
err2016-06-13
err52
PREAI
errVullo, Daniela; Durante, Mariaconcetta; Di Leva, Francesco Saverio; Cosconati, Sandro; Masini, Emanuela; Scozzafava, Andrea; Novellino, Ettore; Supuran, Claudiu T.; Carta, Fabrizio
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Rosmarinic acid inhibits some metabolic enzymes including glutathione S-transferase, lactoperoxidase, acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase isoenzymes
err2016-02-10
err173
errOAAI
errGulcin, Ilhami; Scozzafava, Andrea; Supuran, Claudiu T.; Koksal, Zeynep; Turkan, Fikret; Cetinkaya, Songul; Bingol, Zeynebe; Huyut, Zubeyir; Alwasel, Saleh H.
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Thioxocoumarins Show an Alternative Carbonic Anhydrase Inhibition Mechanism Compared to Coumarins
err2015-12-29
err76
PREAI
errFerraroni, Marta; Carta, Fabrizio; Scozzafava, Andrea; Supuran, Claudiu T.
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Benzenesulfonamides incorporating bulky aromatic/heterocyclic tails with potent carbonic anhydrase inhibitory activity
err2015-12-01
err18
PREAI
errBozdag, Murat; Alafeefy, Ahmed M.; Vullo, Daniela; Carta, Fabrizio; Dedeoglu, Nurcan; Al-Tamimi, Abdul-Malek S.; Al-Jaber, Nabila A.; Scozzafava, Andrea; Supuran, Claudiu T.
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Development and ex vivo evaluation of 5-aminolevulinic acid-loaded niosomal formulations for topical photodynamic therapy
err2015-10-01
err28
PREAI
errBragagni, Marco; Scozzafava, Andrea; Mastrolorenzo, Antonio; Supura, Claudiu T.; Mura, Paola
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Cyclodextrin complexation highly enhances efficacy of arylsulfonylureido benzenesulfonamide carbonic anhydrase inhibitors as a topical antiglaucoma agents
err2015-09-01
err21
PREAI
errBragagni, Marco; Bozdag, Murat; Carta, Fabrizio; Scozzafava, Andrea; Lanzi, Cecilia; Masini, Emanuela; Mura, Paola; Supuran, Claudiu T.
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Cloning, characterization and anion inhibition studies of a new γ-carbonic anhydrase from the Antarctic bacterium Pseudoalteromonas haloplanktis
err2015-08-01
err24
PREAI
errDe Luca, Viviana; Vullo, Daniela; Del Prete, Sonia; Carginale, Vincenzo; Scozzafava, Andrea; Osman, Sameh M.; AlOthman, Zeid; Supuran, Claudiu T.; Capasso, Clemente
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Deciphering the Mechanism of Carbonic Anhydrase Inhibition with Coumarins and Thiocoumarins (vol 53, pg 335, 2010)
err2015-06-30
err4
PREAI
errMaresca, Alfonso; Temperini, Claudia; Pochet, Lionel; Masereel, Bernard; Scozzafava, Andrea; Supuran, Claudiu T.
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Synthesis of a new series of dithiocarbamates with effective human carbonic anhydrase inhibitory activity and antiglaucoma action
err2015-05-01
err41
PREAI
errBozdag, Murat; Carta, Fabrizio; Vullo, Daniela; Akdemir, Atilla; Isik, Semra; Lanzi, Cecilia; Scozzafava, Andrea; Masini, Emanuela; Supuran, Claudiu T.
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A class of sulfonamide carbonic anhydrase inhibitors with neuropathic pain modulating effects
err2015-04-01
err133
PREAI
errCarta, Fabrizio; Mannelli, Lorenzo Di Cesare; Pinard, Melissa; Ghelardini, Carla; Scozzafava, Andrea; McKenna, Robert; Supuran, Claudiu T.
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Sulfonamide inhibition studies of the γ-carbonic anhydrase from the Antarctic cyanobacterium Nostoc commune
err2015-04-01
err32
PREAI
errVullo, Daniela; De Luca, Viviana; Del Prete, Sonia; Carginale, Vincenzo; Scozzafava, Andrea; Capasso, Clemente; Supuran, Claudiu T.
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