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Claudiu T. Supuran

sezione di chimica farmaceutica

152H-index
4.2KPaper Count
13.0WCitation Count
Published Papers 1394
Publication Date
Multi-target pyrazolopyrimidine-coumarin derivatives as potent CA IX/XII and tubulin polymerization inhibitors: Design, synthesis, and biological evaluation
err2026-03-20
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PREAI
errMahmoud S. Elkotamy; Mohamed A. Abdelrahman; Simone Giovannuzzi; Mahmoud Abdelrahman Alkabbani; Alessio Nocentini; Claudiu T. Supuran; Wagdy M. Eldehna; Hatem A. Abdel-Aziz; Sahar M. Abou-Seri
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Hybridization Approach Applied to Umbelliferon and Vanilloids toward New Inhibitors of Carbonic Anhydrases IX and XII with In Vitro Antiproliferative and Anti-inflammatory Activities
err2026-01-01
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PREAI
errMelfi, Francesco; Mencarelli, Noemi; Carradori, Simone; Gallorini, Marialucia; Angeli, Andrea; Poli, Giulio; Cataldi, Amelia; D'Agostino, Ilaria; Di Credico, Andrea; Di Baldassarre, Angela; Tuccinardi, Tiziano; Supuran, Claudiu T.
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Targeting microbial β-CAs: bridging in silico screening with in vitro validation
err2025-12-01
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errOAAI
errTondo, Anna Rita; Fantacuzzi, Marialuigia; Carradori, Simone; D'Agostino, Ilaria; Angeli, Andrea; Supuran, Claudiu T.; Capasso, Clemente; Gambacorta, Nicola; Piemontese, Luca; Laghezza, Antonio; Nicolotti, Orazio; Tortorella, Paolo; Agamennone, Mariangela
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Design; synthesis; molecular modelling investigation and biological studies of novel human carbonic anhydrase inhibitors based on coumalic acid
err2025-08-14
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errOAAI
errVirginia Pontecorvi; Andrea Angeli; Luigi Cutarella; Mattia Mori; Daniela Secci; Michele Coluccia; Simone Carradori; Anna Troiani; Federico Pepi; Chiara Salvitti; Alessia Di Noi; Mattia Spano; Francesca Arrighi; Elena De Falco; Antonella Bordin; Emanuela Berrino; Arianna Granese; Paola Chimenti; Paolo Guglielmi; Claudiu T. Supuran
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Redesigning oxazolidinones as carbonic anhydrase inhibitors against vancomycin-resistant enterococci
err2025-07-01
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errOAAI
errAmmara, Andrea; Giovannuzzi, Simone; Bonardi, Alessandro; Abutaleb, Nader S.; Abouelkhair, Ahmed A.; Flaherty, Daniel P.; Seleem, Mohamed N.; Capasso, Clemente; Gratteri, Paola; Supuran, Claudiu T.
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Exploration of 3-Substituted Benzofuran-Tethered Sulfamoyl Triazoles as Carbonic Anhydrase Inhibitors: Design, Synthesis, and Biological Evaluation
err2025-05-20
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PREAI
errAnuradha Singampalli; Rani Bandela; Bulti Bakchi; Simone Giovannuzzi; Karol Biernacki; Puja Kumari Agnivesh; Srinivas Nanduri; Nitin Pal Kalia; Claudiu T. Supuran; Venkata Madhavi Yaddanapudi
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Selective Inhibition of Carbonic Anhydrase IX and XII by Natural Coumarin Coladonin and Its Derivatives: Promising Antimelanoma and Antiglioblastoma Agents
err2025-05-19
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PREAI
errMustafa, M; Baccari, W; Nocentini, A; Massardi, ML; Smietana, M; Abbass, EM; Saidi, I; Znati, M; Ben Jannet, H; Ronca, R; Supuran, CT; Winum, JY
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Discovery of Trypanosoma cruzi Carbonic Anhydrase Inhibitors by a Combination of Ligand- and Structure-Based Virtual Screening
err2025-05-12
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PREAI
errGori, Denis N. Prada; Barrionuevo, Emilia M.; Alberca, Lucas N.; Sbaraglini, Maria L.; Llanos, Manuel A.; Giovannuzzi, Simone; Carta, Fabrizio; Marchetto, Matias I.; Supuran, Claudiu T.; Soto, Catalina D. Alba; Gavernet, Luciana; Talevi, Alan
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Repositioning FDA-Approved Sulfonamide-Based Drugs as Potential Carbonic Anhydrase Inhibitors in Trypanosoma cruzi: Virtual Screening and In Vitro Studies
err2025-05-01
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errOrtiz-Perez, Eyra; Moreno-Rodriguez, Adriana; Delgado-Maldonado, Timoteo; Ortega-Balleza, Jessica L.; Gonzalez-Gonzalez, Alonzo; Paz-Gonzalez, Alma D.; Vazquez, Karina; Avalos-Navarro, Guadalupe; Giovannuzzi, Simone; Supuran, Claudiu T.; Rivera, Gildardo
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Discover the Power of Lithospermic Acid as Human Carbonic Anhydrase VA and Pancreatic Lipase Inhibitor Through In Silico and In Vitro Studies
err2025-04-21
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errCitriniti, Emanuele Liborio; Rocca, Roberta; Costa, Giosue; Sciacca, Claudia; Cardullo, Nunzio; Muccilli, Vera; Karioti, Anastasia; Carta, Fabrizio; Supuran, Claudiu T.; Alcaro, Stefano; Ortuso, Francesco
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4-Substituted Pyridine-3-Sulfonamides as Carbonic Anhydrase Inhibitors Modified by Click Tailing: Synthesis, Activity, and Docking Studies
err2025-04-17
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errSzafranski, Krzysztof; Slawinski, Jaroslaw; Kawiak, Anna; Chojnacki, Jaroslaw; Kosno, Michal; Ammara, Andrea; Supuran, Claudiu T.
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Exploring nutritional supplement use for countering respiratory tract infections through an X (formerly Twitter)-based survey
err2025-04-15
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errRajeev K. Singla; Himel Mondal; Shailja Singla; Ronita De; Sahar Behzad; Mihnea-Alexandru Găman; Siva Sai Chandragiri; Merisa Cenanovic; Jayanta Kumar Patra; Jennifer R. Depew; Hemanth Kumar Boyina; Abdulkadir Yusif Maigoro; Soojin Lee; Omar M. Atrooz; Gitishree Das; Fabien Schultz; Emad Mohamed Abdallah; Hitesh Chopra; Jamil Ahmad; Rupesh K. Gautam; Sourav S. Patnaik; Bey Hing Goh; Smith B. Babiaka; Sharad Vats; Michael P. Okoh; Atallah F. Ahmed; Ankit Kumar Dubey; Ronan Lordan; Parasuraman Aiya Subramani; Amit Kumar Singh; José M. Alvarez-Suarez; Dinesh Kumar Chellappan; Shravan Kumar Paswan; Prabhakar Semwal; Johra Khan; Sadeeq Sheshe; Neeraj Kumar Sethiya; Tomasz M. Karpiński; Muhammad Riaz; Zahra Emam-Djomeh; Girish Kumar Gupta; Reecha Madaan; Suresh Kumar; Neeraj Choudhary; Salvatore Parisi; Harald Willschke; Vasil Pirgozliev; Rehab A. Rayan; Valentin Ritschl; Shaikat Mondal; Gokhan Zengin; Pritt Verma; Bhupinder Kapoor; Monica Gulati; Gareeballah Osman Adam Balla; Dan Khoa Le; Valeria Pittalà; Amr El-Demerdash; Garba M. Khalid; Jesus Simal-Gandara; Qushmua E. Alzahrani; Gian Luigi Russo; Kiran R. Kharat; Anupam Bishayee; Dongdong Wang; Ilkay Erdogan Orhan; Hammad Ullah; Michael Heinrich; Bikash Baral; Nikolay T. Tzvetkov; Andy Wai Kan Yeung; João M.L. Dias-Ferreira; Scarlett Perez Olea; Yugal Kishore Mohanta; Azazahemad A. Kureshi; Claudiu T. Supuran; Neeraj Rani; Rohit Gundamaraju; Eoghan Joseph Mulholland; Sara Di Lonardo; Albena T. Dinkova-Kostova; Elena González-Burgos; Lucian Hritcu; Pravin Badhe; Abhilasha Singh; Fuad Al-Rimawi; Antoni Sureda; Rambod Abiri; Nady Braidy; Lorenz Kapral; A.N. Abdullahi; Christhian Delfino Villanueva Medina; Helen Sheridan; Massimo Lucarini; Alessandra Durazzo; Francesca Giampieri; Davide Barreca; Witkowska Anna Maria; José Carlos Andrade; Carmela Fimognari; Faizan Akram; Aleksei Tikhonov; Maurizio Battino; Akolade R. Oladipupo; Mila Emerald; Thomas Efferth; Said Amrani; Javier Echeverría; Anna Maria Louka; Surya Kant Tripathi; Bernd L. Fiebich; Nour Eddine Es-Safi; Shafaat Yar Khan; Vivek P. Chavda; Muhammad Asim Masoom Zubair; Samrina Hussain; Muhammad Fasih Ur Rahman; Joy Odimegwu; Jaroslaw Olav Horbanczuk; Hari Prasad Devkota; Alejandro Cifuentes; Rupinder Sodhi; Antonello Santini; Ourlad Alzeus G. Tantengco; Sandeep Ramchandra Pai; Ananda Kumar Chettupalli; Sebastian Granica; Nikola M. Stojanović; Devesh Tewari; Vineet Mittal; Vandana Garg; Mohammad Akhlaquer Rahman; Rajan Logesh; Ioana Berindan-Neagoe; Rohit Sharma; Artur Jóźwik; Maima Matin; Emil D. Parvanov; Nina Strzałkowska; Farhan Bin Matin; Olena Litvinova; Jivko Stoyanov; Monika Michalczuk; Bogumila Zima-Kulisiewicz; Okyaz Eminaga; Awanish Mishra; Nishat Jahan; Joanna Bensz; Tanuj Joshi; Aman Upaganlawar; Kiran Patni; Aleksandra Zielińska; Dalibor Hrg; Artur Stolarczyk; Olga Adamska; George Perry; Michał Ławiński; Agnieszka Kamińska; Mario Štefanović; Bodrun Naher Siddiquea; Sara Frazzini; Luciana Rossi; Marek Wieczorek; Michel Edwar Mickael; Leif-Alexander Garbe; Atanas G. Atanasov; Bairong Shen
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Exploration of Aromatic Hydrazides as Inhibitors of Human Carbonic Anhydrases
err2025-04-01
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errOAAI
errMenendez, German Benito; Giovannuzzi, Simone; Bonardi, Alessandro; Nocentini, Alessio; Gratteri, Paola; Supuran, Claudiu T.
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Investigation on Human Carbonic Anhydrase IX and XII Inhibitory Activity and A549 Antiproliferative Activity of a New Class of Coumarinamides
err2025-03-05
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errMoi, Davide; Carradori, Simone; Gallorini, Marialucia; Mencarelli, Noemi; Deplano, Alberto; Angeli, Andrea; Vittorio, Serena; Supuran, Claudiu T.; Onnis, Valentina
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Synthesis and Evaluation of Thiazolidinone-Isatin Hybrids for Selective Inhibition of Cancer-Related Carbonic Anhydrases
err2025-03-01
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errOnali, Alessia; Sanna, Erica; Lupia, Antonio; Secci, Daniela; Atzeni, Giulia; Demuru, Laura; Angeli, Andrea; Cottiglia, Filippo; Meleddu, Rita; Emmolo, Roberta; Corona, Angela; Maccioni, Elias; Supuran, Claudiu T.; Distinto, Simona
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Kinetic and structural studies of gamma-carbonic anhydrase from the oral pathogen Porphyromonas gingivalis
err2025-03-01
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PREAI
errFerraroni, Marta; Angeli, Andrea; De Luca, Viviana; Capasso, Clemente; Supuran, Claudiu T.
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