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SaveDiscovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells
Bozdag, Murat; Mroweh, Nabil; Raucci, Alessia; Angeli, Andrea; Peppicelli, Silvia; Biagioni, Alessio; Calorini, Lido; Trisciuoglio, Daniela; Ragno, Rino; Astolfi, Roberta; Giuliani, Lidia; Zwergel, Clemens; Valente, Sergio; Andreucci, Elena; Carta, Fabrizio; Mai, Antonello; Supuran, Claudiu T.
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SaveA Xanthine Derivative With Novel Heat Shock Protein 90-Alpha Inhibitory and Senolytic Properties
Atlante, Sandra; Cis, Luca; Pirolli, Davide; Zamperla, Michela Gottardi; Barbi, Veronica; Mai, Antonello; Zwergel, Clemens; Marcozzi, Serena; Giuliani, Maria Elisa; Bigossi, Giorgia; Lai, Giovanni; Orlando, Fiorenza; Giacconi, Robertina; Lattanzio, Fabrizia; Matacchione, Giulia; Giordani, Chiara; Bracci, Massimo; Olivieri, Fabiola; Boschi, Federico; De Fatis, Paola Tabarelli; Ivaldi, Giovanni Battista; Malavolta, Marco; Farsetti, Antonella; De Rosa, Maria Cristina; Gaetano, Carlo
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SaveProcognitive Potential of Neuroprotective Triazine 5-HT6 Receptor Antagonists Tested on Chronic Activity In Vivo in Rats: Computer-Aided Insight into the Role of Chalcogen-Differences on the Pharmacological Profile
Jastrzebska-Wiesek, M; Garbo, S; Cios, A; Wilczynska-Zawal, N; Partyka, A; Honkisz-Orzechowska, E; Zeslawska, E; Handzlik, J; Mordyl, B; Gluch-Lutwin, M; Raucci, A; Hittinger, M; Starek, M; Dabrowska, M; Nitek, W; Karcz, T; Skórkowska, A; Joanna, A; Czarnota-Lydka, K; Pyka, P; Szymanska, E; Kucwaj-Brysz, K; Zwergel, C; Wesolowska, A; Battistelli, C; Handzlik, J
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SaveHDAC3 genetic and pharmacologic inhibition radiosensitizes fusion positive rhabdomyosarcoma by promoting DNA double-strand breaks
Cassandri, Matteo; Porrazzo, Antonella; Pomella, Silvia; Noce, Beatrice; Zwergel, Clemens; Aiello, Francesca Antonella; Vulcano, Francesca; Milazzo, Luisa; Camero, Simona; Pajalunga, Deborah; Spada, Massimo; Manzi, Valeria; Gravina, Giovanni Luca; Codenotti, Silvia; Piccione, Michela; Tomaciello, Miriam; Signore, Michele; Barillari, Giovanni; Marchese, Cinzia; Fanzani, Alessandro; De Angelis, Biagio; Quintarelli, Concetta; Vakoc, Christopher R.; Chen, Eleanor Y.; Megiorni, Francesca; Locatelli, Franco; Valente, Sergio; Mai, Antonello; Rota, Rossella; Marampon, Francesco
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SaveHDAC3 sustains resistance to hypofractionated radiotherapy in fusion positve rhabdomyosarcoma cells
Cassandri, Matteo; Porrazzo, Antonella; Pomella, Silvia; Camero, Simona; Aiello, Francesca A.; D'Archivio, Lucrezia; Zwergel, Clemens; Noce, Beatrice; Tomaciello, Miriam; Vulcano, Francesca; Milazzo, Luisa; Pedini, Francesca; Signore, Michele; Fanzani, Alessandro; Marchese, Cinzia; Minniti, Giuseppe; Valente, Sergio; Mai, Antonello; Megiorni, Francesca; Rota, Rossella; Marampon, Francesco
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SaveHDAC1/2 control mesothelium/ovarian cancer adhesive interactions impacting on Talin-1-α5β1-integrin-mediated actin cytoskeleton and extracellular matrix protein remodeling
Terri, Michela; Sandoval, Pilar; Bontempi, Giulio; Montaldo, Claudia; Tomero-Sanz, Henar; de Turris, Valeria; Trionfetti, Flavia; Pascual-Anton, Lucia; Clares-Pedrero, Irene; Battistelli, Cecilia; Valente, Sergio; Zwergel, Clemens; Mai, Antonello; Rosano, Laura; del Pozo, Miguel angel; Sanchez-Alvarez, Miguel; Cabanas, Carlos; Tripodi, Marco; Lopez-Cabrera, Manuel; Strippoli, Raffaele
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SaveFirst-in-Class Selenium-Containing Potent Serotonin Receptor 5-HT6 Agents with a Beneficial Neuroprotective Profile against Alzheimer's Disease
Pyka, Patryk; Haberek, Wawrzyniec; Wiecek, Malgorzata; Szymanska, Ewa; Ali, Wesam; Cios, Agnieszka; Jastrzebska-Wiesek, Magdalena; Satala, Grzegorz; Podlewska, Sabina; Di Giacomo, Silvia; Di Sotto, Antonella; Garbo, Sabrina; Karcz, Tadeusz; Lambona, Chiara; Marocco, Francesco; Latacz, Gniewomir; Sudol-Talaj, Sylwia; Mordyl, Barbara; Gluch-Lutwin, Monika; Siwek, Agata; Czarnota-Lydka, Kinga; Gogola, Dawid; Olejarz-Maciej, Agnieszka; Wilczynska-Zawal, Natalia; Honkisz-Orzechowska, Ewelina; Starek, Malgorzata; Dabrowska, Monika; Kucwaj-Brysz, Katarzyna; Fioravanti, Rossella; Nasim, Muhammad Jawad; Hittinger, Marius; Partyka, Anna; Wesolowska, Anna; Battistelli, Cecilia; Zwergel, Clemens; Handzlik, Jadwiga
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