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Yan Fan

nanjing drum tower hospital group suqian hospital

21H-index
85Paper Count
1.9KCitation Count
Published Papers 31
Publication Date
Discovery of a Novel EGFR PROTAC Degrader against C797S Resistance Mutation with Potent Antitumor Efficacy in NSCLC Treatment
err2025-07-10
err0
PREAI
errXiaoxue Wang; Cheng Wang; Yakun Ma; Yongjun Piao; Yi Shi; Shuang Yang; Jia Li; Yan Fan
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Discovery of (E)-2-cyano-N-(2,3-dihydrobenzo[b][1,4] dioxin-6-yl)-3-(1H-indol-3-yl)acrylamide as a novel TDO inhibitor for cancer treatment
err2025-07-01
err0
PREAI
errWang, Xiang; Wang, Xiaoshuang; Wang, Xiaoxue; Xu, Kejia; Long, Jie; Chen, Yanan; Liu, Yanhua; Niu, Haiying; Zeng, Beilei; Fan, Yan
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Amelioration of immunoglobulin A vasculitis by suppression of the pathological expansion of T follicular helper 17 cells
err2024-12-01
err0
PREAI
errJiang, Qinglian; Chi, Xuyang; Wei, Tong; Nakayamada, Shingo; Shan, Yu; Sun, Yini; Zhao, Xing; Zhou, Jieqing; Fan, Yan; Gu, Jia; Jiang, Hong; Ma, Xiaoxue
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Novel EGFR inhibitors against resistant L858R/T790M/C797S mutant for intervention of non-small cell lung cancer
err2024-11-01
err3
PREAI
errWang, Xiaoxue; Qin, Zhongxiang; Qiu, Wenrui; Xu, Kejia; Bai, Yuting; Zeng, Beilei; Ma, Yakun; Yang, Shuang; Shi, Yi; Fan, Yan
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CDK9 inhibitors in cancer research
err2022-01-01
err15
errOAAI
errHuang, Zhi; Wang, Tianqi; Wang, Cheng; Fan, Yan
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Discovery of a potent and selective inhibitor of histone lysine demethylase KDM4D
err2021-11-01
err10
PREAI
errFang, Zhen; Liu, Yang; Zhang, Rong; Chen, Qiang; Wang, Tianqi; Yang, Wei; Fan, Yan; Yu, Chundong; Xiang, Rong; Yang, Shengyong
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Discovery of 12O-A Novel Oral Multi-Kinase Inhibitor for the Treatment of Solid Tumor
err2020-11-09
err4
errOAAI
errFan, Yan; Huang, Zhi; Wang, Xiaoshuang; Ma, Yakun; Li, Yongtao; Yang, Shengyong; Shi, Yi
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Novel CDKs inhibitors for the treatment of solid tumour by simultaneously regulating the cell cycle and transcription control
err2020-01-03
err17
errOAAI
errWang, Xin; Deng, Kaiyuan; Wang, Cheng; Li, Yao; Wang, Tianqi; Huang, Zhi; Ma, Yakun; Sun, Peiqing; Shi, Yi; Yang, Shengyong; Fan, Yan; Xiang, Rong
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Novel dual inhibitors targeting CDK4 and VEGFR2 synergistically suppressed cancer progression and angiogenesis
err2019-11-01
err28
PREAI
errHuang, Zhi; Zhao, Borui; Qin, Zhongxiang; Li, Yongtao; Wang, Tianqi; Zhou, Wei; Zheng, Jianyu; Yang, Shengyong; Shi, Yi; Fan, Yan; Xiang, Rong
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Novel cyclin-dependent kinase 9 (CDK9) inhibitor with suppression of cancer sternness activity against non-small-cell lung cancer
err2019-11-01
err40
PREAI
errWang, Xin; Yu, Chenhua; Wang, Cheng; Ma, Yakun; Wang, Tianqi; Li, Yao; Huang, Zhi; Zhou, Mangian; Sun, Peiqing; Zheng, Jianyu; Yang, Shengyong; Fan, Yan; Xiang, Rong
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Memory stem T cells generated by Wnt signaling from blood of human renal clear cell carcinoma patients
err2019-01-01
err19
errOAAI
errYan, Cihui; Chang, Jingjing; Song, Xinmiao; Yan, Fan; Yu, Wenwen; An, Yang; Wei, Feng; Yang, Lili; Ren, Xiubao
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Mangosteen ethanol extract alleviated the severity of collagen-induced arthritis in rats and produced synergistic effects with methotrexate
err2018-12-04
err20
errOAAI
errZuo, Jian; Yin, Qin; Wang, Lin; Zhang, Wen; Fan, Yan; Zho, Yu-Yan; Li, Yan; Wang, Guo-Dong
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A highly potent and selective inhibitor Roxyl-WL targeting IDO1 promotes immune response against melanoma
err2018-06-22
err10
errOAAI
errXu, Guangwei; Wang, Tianqi; Li, Yongtao; Huang, Zhi; Wang, Xin; Zheng, Jianyu; Yang, Shengyong; Fan, Yan; Xiang, Rong
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Discovery of &ITN&IT1-(4-((7-Cyclopentyl-6-(dimethylcarbamoyl)-7&ITH&IT-pyrrolo[2,3-&ITd&IT]pyrimidin-2-yl)amino)phenyl)-&ITN&IT8-hydroxyoctanediamide as a Novel Inhibitor Targeting Cyclin-dependent Kinase 4/9 (CDK4/9) and Histone Deacetlyase 1 (HDAC1) against Malignant Cancer
err2018-03-08
err73
PREAI
errLi, Yongtao; Luo, Xiaohe; Guo, Qingxiang; Nie, Yongwei; Wang, Tianqi; Zhang, Chao; Huang, Zhi; Wang, Xin; Liu, Yanhua; Chen, Yanan; Zheng, Jianyu; Yang, Shengyong; Fan, Yan; Xiang, Rong
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Highly Selective, Potent, and Oral mTOR Inhibitor for Treatment of Cancer as Autophagy Inducer
err2018-01-27
err18
PREAI
errGuo, Qingxiang; Yu, Chenhua; Zhang, Chao; Li, Yongtao; Wang, Tianqi; Huang, Zhi; Wang, Xin; Zhou, Wei; Li, Yao; Qin, Zhongxiang; Wang, Cheng; Gao, Ruifang; Nie, Yongwei; Ma, Yakun; Shi, Yi; Zheng, Jianyu; Yang, Shengyong; Fan, Yan; Xiang, Rong
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