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Dante Rotili

roma tre university

52H-index
274Paper Count
8.8KCitation Count
Published Papers 156
Publication Date
Development of High-Affinity CHD1 Chromodomain Inhibitors
err2026-05-05
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errHolger Greschik; Florian Friedrich; Ludwig Seifert; Farnoush Mousavizadeh; Francesco Fiorentino; Johannes Walz; Lin Zhang; Jianyu Li; Emanuele Fabbrizi; Stefano Tomassi; Farhad Panahi; Niklas Papenkordt; Silas L. Wurnig; Johannes Osterroth; Anna M. Strasser; Jan Ruprecht; Aurélien F. A. Moumbock; Martin Hügle; Manuela Sum; Ling Peng; Sheng Wang; Adina A. Baniahmad; Laura Pulido-Cortés; H. Th. Marc Timmers; Ralf Flaig; Eric Metzger; Bernhard Breit; Oliver Einsle; Stefan Günther; Dante Rotili; Antonello Mai; Roland Schüle; Manfred Jung
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Development of Biphenyl-Substituted Uracil-Based Hydroxamic Acids (UBHAs) as Potent HDAC Inhibitors with Pro-Apoptotic Activity in Leukemia and Prostate Cancer Cells
err2026-04-30
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errFrancesco Fiorentino; Giulio Bontempi; Federica Michetti; Valeria Pecci; Emanuele Fabbrizi; Daniela Passeri; Letizia Corsetti; Valentina Farini; Fabrizio Casano; Antimo Gioiello; Antonella Di Sotto; Roberto Pellicciari; Donatella Del Bufalo; Daniela Trisciuoglio; Simona Nanni; Raffaele Strippoli; Antonello Mai; Dante Rotili
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Structural snapshots of Pseudomonas aeruginosa LptB2FG and LptB2FGC reveal insights into lipopolysaccharide recognition and transport
err2025-12-17
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errFrancesco Fiorentino; Matteo Cervoni; Yi Wang; Leonhard H. Urner; Joshua B. Sauer; Anh Tran; Robin A. Corey; Dante Rotili; Antonello Mai; Phillip J. Stansfeld; Francesco Imperi; Edward W. Yu; Chih-Chia Su; Carol V. Robinson; Jani R. Bolla
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Correction: Sennato et al. Optimization of Lipoplexes Functionalized with a Sialic Acid Mimetic (F9-PEG) to Target the C1858T PTPN22 Variant for Preclinical Assessment of a Novel Immunotherapy in Endocrine Autoimmunity. Pharmaceutics 2025, 17, 710
err2025-12-12
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errSimona Sennato; Giorgia Paldino; Cecilia Bombelli; Irene Mezzani; Stefania Petrini; Eugenia Belcastro; Domenico Vittorio Delfino; Francesco Fiorentino; Carlotta Marianecci; Alessia Ciogli; Dante Rotili; Francesca Ceccacci; Alessandra Fierabracci
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A Feasibility Study of Co-Established Patient-Derived Subcutaneous Xenograft and Organotypic Slice Cultures in Hormone-Naive Primary Prostate Cancer Preclinical Modeling: A Single-Institution Experience
err2025-11-06
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errValeria Pecci; Melissa Borsa; Aurora Aiello; Sara De Martino; Luca Cis; Francesco Pierconti; Domenico Varacalli; Martina Bracco; Cristian Ripoli; Francesco Pinto; Dante Rotili; Claudio Grassi; Carlo Gaetano; Alfredo Pontecorvi; Antonella Farsetti; Simona Nanni
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Sirtuin modulators: a review of patents from 2020 to 2024
err2025-11-06
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PREAI
errEmanuele Fabbrizi; Francesco Fiorentino; Antonello Mai; Dante Rotili
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Unraveling the Roles of Epigenetic Regulators During the Embryonic Development of Rhipicephalus microplus
err2025-09-21
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errAnderson Mendonça Amarante; Daniel Martins de Oliveira; Marcos Paulo Nicolich Camargo de Souza; Manoel Fonseca-Oliveira; Antonio Galina; Serena Rosignoli; Angélica Fernandes Arcanjo; Bruno Moraes; Alessandro Paiardini; Dante Rotili; Juan Diego de Paula Li Yasumura; Sarah Henaut-Jacobs; Thiago Motta Venancio; Marcelle Uhl; Rodrigo Nunes-da-Fonseca; Luis Fernando Parizi; Itabajara da Silva Vaz Junior; Claudia dos Santos Mermelstein; Thamara Rios; Lucas Tirloni; Carlos Logullo; Marcelo Rosado Fantappié
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A C3-Symmetric Diphenylethylendiamine-Based Catalyst in the Asymmetric Michael Addition of α,β-Unsaturated Ketones with 4-Hydroxycoumarin and 4-Hydroxyquinolin-2-One
err2025-08-13
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PREAI
errShilashi Badasa Oljira; Martina De Angelis; Simone Manetto; Francesco Fiorentino; Dante Rotili; Luciana Mosca; Daniel Di Risola; Roberto Mattioli; Marco Pierini; Giulia Mazzoccanti; Alessia Ciogli
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Bromodomain and Extra-Terminal Family Proteins BRD2, BRD3, and BRD4 Contribute to H19-Dependent Transcriptional Regulation of Cell Adhesion Molecules, Modulating Metastatic Dissemination Program in Prostate Cancer
err2025-08-09
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errValeria Pecci; Melissa Borsa; Aurora Aiello; Sara De Martino; Luca Cis; Cristian Ripoli; Dante Rotili; Francesco Pierconti; Francesco Pinto; Claudio Grassi; Carlo Gaetano; Antonella Farsetti; Simona Nanni
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1,2,4-Oxadiazoles in medicinal chemistry: trends of the last years
err2025-07-05
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errAnastasia Cherkasova; Roberta Astolfi; Maxim Nawrozkij; Boris Gladkikh; Eleonora Proia; Lidia Giuliani; Dante Rotili; Rino Ragno; Roman Ivanov
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Tranylcypromine-Based LSD1 Inhibitors as Useful Agents to Reduce Viability of Schistosoma mansoni
err2025-07-02
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errEmanuele Fabbrizi; Gebremedhin Solomon Hailu; A. Ganesan; Rossella Fioravanti; Clemens Zwergel; Chiara Lambona; Sergio Valente; Giulia Fianco; Angela Iuzzolino; Daniela Trisciuoglio; Jonatan Caroli; Andrea Mattevi; Cécile Häberli; Jennifer Keiser; Dante Rotili; Antonello Mai
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Development of C646-Based Proteolysis Targeting Chimeras Degraders of the Lysine Acetyltransferases CBP and p300
err2025-04-01
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PREAI
errFiorentino, Francesco; Spriano, Filippo; Tomaselli, Daniela; Risi, Giorgia; Fabbrizi, Emanuele; Pecci, Valeria; Nanni, Simona; Bertoni, Francesco; Rotili, Dante; Mai, Antonello
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Quinoline-based compounds can inhibit diverse enzymes that act on DNA
err2024-12-01
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errZhou, Jujun; Chen, Qin; Ren, Ren; Yang, Jie; Liu, Bigang; Horton, John R.; Chang, Caleb; Li, Chuxuan; Maksoud, Leora; Yang, Yifei; Rotili, Dante; Jain, Abhinav K.; Zhang, Xing; Blumenthal, Robert M.; Chen, Taiping; Gao, Yang; Valente, Sergio; Mai, Antonello; Cheng, Xiaodong
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Epigenetic modulation of sirt1 and sirt6 in cardiovascular diseases: unraveling autophagy regulation and endothelial function
err2024-10-28
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PREAI
errBordin, A.; Cozzolino, C.; Floris, E.; Valente, S.; Cavarretta, E.; Picchio, V; Chimenti, I; Rotili, D.; Frati, G.; Mai, A.; De Falco, E.
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Prognostic Impact of H19/Cell Adhesion Molecules Circuitry on Prostate Cancer Biopsy
err2024-10-12
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errPecci, Valeria; Pierconti, Francesco; Carlino, Angela; Pinto, Francesco; Gradilone, Ugo; De Martino, Sara; Rotili, Dante; Grassi, Claudio; Pontecorvi, Alfredo; Gaetano, Carlo; Strigari, Lidia; Farsetti, Antonella; Nanni, Simona
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The bromodomain and extraterminal domain family proteins, BRD2, BRD3 and BRD4, are enrolled in H19-dependent transcriptional regulation of cell adhesion molecules and modulate metastatic dissemination program in prostate cancer
err2024-10-01
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PREAI
errPecci, V.; Borsa, M.; Aiello, A.; De Martino, S.; Cis, L.; Ripoli, C.; Rotili, D.; Pierconti, F.; Pinto, F.; Grassi, C.; Alfredo, P.; Gaetano, C.; Antonella, F.; Nanni, S.
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Activation and inhibition of sirtuins: From bench to bedside
err2024-08-31
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errFiorentino, Francesco; Fabbrizi, Emanuele; Mai, Antonello; Rotili, Dante
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Transmission-Blocking Strategies for Malaria Eradication: Recent Advances in Small-Molecule Drug Development
err2024-07-19
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errAppetecchia, Federico; Fabbrizi, Emanuele; Fiorentino, Francesco; Consalvi, Sara; Biava, Mariangela; Poce, Giovanna; Rotili, Dante
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Structure-based mechanism of riboregulation of the metabolic enzyme SHMT1
err2024-07-01
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errSpizzichino, Sharon; Di Fonzo, Federica; Marabelli, Chiara; Tramonti, Angela; Chaves-Sanjuan, Antonio; Parroni, Alessia; Boumis, Giovanna; Liberati, Francesca Romana; Paone, Alessio; Montemiglio, Linda Celeste; Ardini, Matteo; Jakobi, Arjen J.; Bharadwaj, Alok; Swuec, Paolo; Tartaglia, Gian Gaetano; Paiardini, Alessandro; Contestabile, Roberto; Mai, Antonello; Rotili, Dante; Fiorentino, Francesco; Macone, Alberto; Giorgi, Alessandra; Tria, Giancarlo; Rinaldo, Serena; Bolognesi, Martino; Giardina, Giorgio; Cutruzzola, Francesca
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M6A reduction relieves FUS-associated ALS granules
err2024-06-12
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errDi Timoteo, Gaia; Giuliani, Andrea; Setti, Adriano; Biagi, Martina C.; Lisi, Michela; Santini, Tiziana; Grandioso, Alessia; Mariani, Davide; Castagnetti, Francesco; Perego, Eleonora; Zappone, Sabrina; Lattante, Serena; Sabatelli, Mario; Rotili, Dante; Vicidomini, Giuseppe; Bozzoni, Irene
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