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Amy Hauck Newman

national institutes of health

63H-index
414Paper Count
1.4WCitation Count
Published Papers 219
Publication Date
The structure of the dopamine D3 receptor bound to cariprazine reveals principles for partial agonists with designed pharmacology
err2026-08-28
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errEliane Hadas Yardeni; Dóra Judit Kiss; Julie Sanchez; Keshet Shavit; Dénes Szepesi Kovács; Attila Egyed; Caleb D. Vogt; Supriya A. Gaitonde; Jacqueline Glenn; Meritxell Canals; Michel Bouvier; Amy Hauck Newman; J. Robert Lane; György M. Keserű; Moran Shalev-Benami
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Tailoring cariprazine for dual disorders via secondary pharmacophore optimization
err2026-02-10
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errCaleb D. Vogt; Julie Sanchez; Alessandro Bonifazi; Elizabeth Saab; Arina Ranjit; Rana Rais; J. Robert Lane; Amy Hauck Newman
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Structure–Function Activity Relationships of Cariprazine Analogues with Distinct G Protein versus β-Arrestin Activities at the Dopamine D3 Receptor
err2025-11-28
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PREAI
errBradley M. Keegan; Caleb D. Vogt; Li Chen; Renee J. Nosko; Elizabeth Saab; Alessandro Bonifazi; Emma S. Gogarnoiu; Anver Basha Shaik; Amy Hauck Newman; Lei Shi
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Acai Berry Extracts Can Mitigate the L-Glutamate-Induced Neurotoxicity Mediated by N-Methyl-D-Aspartate Receptors
err2025-10-01
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errMaryam N. ALNasser; Nirmal Malik; Abrar Ahmed; Amy Newman; Ian R. Mellor; Wayne G. Carter
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Development of a HiBiT Peptide-Based NanoBRET Ligand Binding Assay for Galanin Receptor 1 in Live Cells
err2025-07-04
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PREAI
errHu Zhu; Harrison C. Daly; Tae Gyun Yang; Josh Born; Gisela Andrea Camacho-Hernandez; Mingyang Yuan; Mari Inglese; Vinoth Kumar Chenniappan; Kris Zimmerman; Robin Hurst; Xin Hu; Amy Hauck Newman; Sergi Ferré; Rachel Friedman Ohana; Matthew D. Hall; Samarjit Patnaik
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Monoamine transporter ubiquitination and inward-open conformation synergistically maximize transporter endocytosis
err2024-11-22
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errSorkina, Tatiana; Bagalkot, Tarique; Cheng, Mary Hongying; Guthrie, Daryl A.; Newman, Amy Hauck; Watkins, Simon C.; Sorkin, Alexander
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Presynaptic and Postsynaptic Mesolimbic Dopamine D3 Receptors Play Distinct Roles in Cocaine Versus Opioid Reward in Mice
err2024-11-01
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PREAI
errXi, Zheng-Xiong; Bocarsly, Miriam E.; Galaj, Ewa; Hempel, Briana; Teresi, Catherine; Shaw, Marlisa; Bi, Guo-Hua; Jordan, Chloe; Linz, Emily; Alton, Hannah; Tanda, Gianluigi; Freyberg, Zachary; Alvarez, Veronica A.; Newman, Amy Hauck
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Development of Novel Tools for Dissection of Central Versus Peripheral Dopamine D2-Like Receptor Signaling in Dysglycemia
err2024-06-13
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errBonifazi, Alessandro; Ellenberger, Michael; Farino, Zachary J.; Aslanoglou, Despoina; Rais, Rana; Pereira, Sandra; Mantilla-Rivas, Jose O.; Boateng, Comfort A.; Eshleman, Amy J.; Janowsky, Aaron; Hahn, Margaret K.; Schwartz, Gary J.; Slusher, Barbara S.; Newman, Amy Hauck; Freyberg, Zachary
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Empowering Voices: Inspiring Women in Medicinal Chemistry
err2024-03-08
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errBlanco, Maria-Jesus; Bronson, Joanne J.; Dimauro, Erin F.; Dzierba, Carolyn; Eggen, Marijean; Garner, Amanda L.; Georg, Gunda; Giarolla, Jeanine; Goodwin, Nicole C.; Grenier-Davies, Melissa C.; Haskell-Luevano, Carrie; Holzgrabe, Ulrike; Huang, Rong; Lagiakos, H. Rachel; Leftheris, Katerina; Martin, Yvonne; Matos, Maria Joao; May-Dracka, Tricia L.; Muller, Christa E.; Newman, Amy H.; Parmee, Emma; Petter, Jennifer C.; Tamayo, Nuria A.; Wexler, Ruth R.; Bolognesi, Maria Laura; Ripka, Amy; Young, Wendy
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Empowering Voices: Inspiring Women in Medicinal Chemistry
err2024-03-08
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errBlanco, Maria-Jesus; Bronson, Joanne J.; DiMauro, Erin F.; Dzierba, Carolyn; Eggen, Marijean; Garner, Amanda L.; Georg, Gunda; Giarolla, Jeanine; Goodwin, Nicole C.; Grenier-Davies, Melissa C.; Haskell-Luevano, Carrie; Holzgrabe, Ulrike; Huang, Rong; Lagiakos, H. Rachel; Leftheris, Katerina; Martin, Yvonne; Matos, Maria Joao; May-Dracka, Tricia L.; Muller, Christa E.; Newman, Amy H.; Parmee, Emma; Petter, Jennifer C.; Tamayo, Nuria A.; Wexler, Ruth R.; Bolognesi, Maria Laura; Ripka, Amy; Young, Wendy
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Development of a Fluorescently Labeled Ligand for Rapid Detection of DAT in Human and Mouse Peripheral Blood Monocytes
errJACS AU
IF8.7
err2024-01-24
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errCamacho-Hernandez, Gisela Andrea; Gopinath, Adithya; Okorom, Amarachi V.; Khoshbouei, Habibeh; Newman, Amy Hauck
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Modifications to 1-(4-(2-Bis(4-fluorophenyl)methyl)sulfinyl)alkyl Alicyclic Amines That Improve Metabolic Stability and Retain an Atypical DAT Inhibitor Profile
err2023-12-20
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PREAI
errOkorom, Amarachi V.; Camacho-Hernandez, Gisela Andrea; Salomon, Kristine; Lee, Kuo Hao; Ku, Therese C.; Cao, Jianjing; Won, Sung Joon; Friedman, Jacob; Lam, Jenny; Paule, James; Rais, Rana; Klein, Benjamin; Xi, Zheng-Xiong; Shi, Lei; Loland, Claus J.; Newman, Amy Hauck
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Pharmacology and Therapeutic Potential of Benzothiazole Analogues for Cocaine Use Disorder
err2023-08-30
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errBoateng, Comfort A.; Nilson, Ashley N.; Placide, Rebekah; Pham, Mimi L.; Jakobs, Franziska M.; Boldizsar, Noelia; Mcintosh, Scot; Stallings, Leia S.; Korankyi, Ivana V.; Kelshikar, Shreya; Shah, Nisha; Panasis, Diandra; Muccilli, Abigail; Ladik, Maria; Maslonka, Brianna; McBride, Connor; Sanchez, Moises Ximello; Akca, Ebrar; Alkhatib, Mohammad; Saez, Julianna; Nguyen, Catherine; Kurtyan, Emily; DePierro, Jacquelyn; Crowthers, Raymond; Brunt, Dylan; Bonifazi, Alessandro; Newman, Amy Hauck; Rais, Rana; Slusher, Barbara S.; Free, R. Benjamin; Sibley, David R.; Stewart, Kent D.; Wu, Chun; Hemby, Scott E.; Keck, Thomas M.
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Pharmacological and Physicochemical Properties Optimization for Dual-Target Dopamine D3 (D3R) and μ-Opioid (MOR) Receptor Ligands as Potentially Safer Analgesics
err2023-07-19
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errBonifazi, Alessandro; Saab, Elizabeth; Sanchez, Julie; Nazarova, Antonina L.; Zaidi, Saheem A.; Jahan, Khorshada; Katritch, Vsevolod; Canals, Meritxell; Lane, J. Robert; Newman, Amy Hauck
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An FSCV Study on the Effects of Targeted Typical and Atypical DAT Inhibition on Dopamine Dynamics in the Nucleus Accumbens Shell of Male and Female Mice
err2023-07-19
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PREAI
errHersey, Melinda; Chen, Andy Y.; Bartole, Mattingly K.; Anand, Jayati; Newman, Amy Hauck; Tanda, Gianluigi
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Evaluating Serotonin 2C and Dopamine D3 Receptor Ligands, Alone and in Mixtures, as Candidate Medications for Substance Use Disorders
err2023-06-01
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errMason, Briana; Thomas, Anona; Shi, Yonggong; George, Christina; Cao, Jianjing; Newman, Amy; Collins, Gregory T.
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Effects of selective dopamine D3 receptor partial agonist/antagonists on oxycodone self-administration and antinociception in monkeys
err2023-04-28
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PREAI
errWoodlief, Kendall; Allen, Mia I.; Cornelissen, Jeremy C.; Banks, Matthew L.; Newman, Amy Hauck; Nader, Michael A.
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The Effects of the Dopamine Transporter Ligands JJC8-088 and JJC8-091 on Cocaine versus Food Choice in Rhesus MonkeysS
err2023-03-01
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errOAAI
errRahimi, Omeed; Cao, Jianjing; Lam, Jenny; Childers, Steven R.; Rais, Rana; Porrino, Linda J.; Newman, Amy Hauck; Nader, Michael A.
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3,4-Methylenedioxypyrovalerone High-Responder Phenotype as a Tool to Evaluate Candidate Medications for Stimulant Use Disorder
err2023-03-01
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errOAAI
errDoyle, Michelle R.; Peng, Lindsey N.; Cao, Jianjing; Rice, Kenner C.; Newman, Amy Hauck; Collins, Gregory T.
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