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SaveDiscovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells
Bozdag, Murat; Mroweh, Nabil; Raucci, Alessia; Angeli, Andrea; Peppicelli, Silvia; Biagioni, Alessio; Calorini, Lido; Trisciuoglio, Daniela; Ragno, Rino; Astolfi, Roberta; Giuliani, Lidia; Zwergel, Clemens; Valente, Sergio; Andreucci, Elena; Carta, Fabrizio; Mai, Antonello; Supuran, Claudiu T.
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SaveEssential Oils as Antimicrobials against Acinetobacter baumannii: Experimental and Literature Data to Definite Predictive Quantitative Composition-Activity Relationship Models Using Machine Learning Algorithms
Astolfi, Roberta; Oliva, Alessandra; Raffo, Antonio; Sapienza, Filippo; Ragno, Alessio; Proia, Eleonora; Mastroianni, Claudio M.; Luceri, Cristina; Bozovic, Mijat; Mladenovic, Milan; Papa, Rosanna; Bottoni, Patrizia; Mazzinelli, Elena; Nocca, Giuseppina; Ragno, Rino
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Save(Heteroarylmethyl)benzoic Acids as a New Class of Bacterial Cystathionine γ-Lyase Inhibitors: Synthesis, Biological Evaluation, and Molecular Modeling
Golovina, Anastasia; Proia, Eleonora; Fiorentino, Francesco; Yunin, Maxim; Kasatkina, Maria; Zigangirova, Nailya; Soloveva, Anna; Sysolyatina, Elena; Ermolaeva, Svetlana; Novikov, Roman; Silonov, Sergei; Pushkin, Sergei; Mladenovic, Milan; Isakova, Julia; Belik, Albina; Nawrozkij, Maxim; Rotili, Dante; Ragno, Rino; Ivanov, Roman
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SaveScreening of the activity of sixty essential oils against plasmodium early mosquito stages in vitro and machine learning analysis reveals new putative inhibitors of malaria parasites
Deligianni, Elena; Pizzi, Elisabetta; Kavelaki, Ioanna; Siden-Kiamos, Inga; Sapienza, Filippo Umberto; Fioravanti, Rossella; Garzoli, Stefania; Pace, Tomasino; Ponzi, Marta; Ragno, Rino; Curra, Chiara
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SaveRETRACTION: Dissecting the role of novel EZH2 inhibitors in primary glioblastoma cell cultures: effects on proliferation, epithelialmesenchymal transition, migration, and on the pro-inflammatory phenotype (Retraction of Vol 11, art no 173, 2019)
Stazi, Giulia; Taglieri, Ludovica; Nicolai, Alice; Romanelli, Annalisa; Fioravanti, Rossella; Morrone, Stefania; Sabatino, Manuela; Ragno, Rino; Taurone, Samanta; Nebbioso, Marcella; Carletti, Raffaella; Artico, Marco; Valente, Sergio; Scarpa, Susanna; Mai, Antonello
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SaveChemical Composition and Anti-Candida Activity of Mentha suaveolens Ehrh. Essential Oils Obtained by Different Distillation Processes
Tadic, Vanja; Bozovic, Mijat; Sapienza, Filippo; Astolfi, Roberta; Mladenovic, Milan; Zaka, Maria Cristina; Del Bove, Fabiana; Borzacchi, Francesca; Fraschetti, Caterina; Rossi, Caterina; Vertuani, Silvia; Baldisserotto, Anna; Manfredini, Stefano; Ragno, Rino
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SaveMolecular Docking Assessment of Cathinones as 5-HT2AR Ligands: Developing of Predictive Structure-Based Bioactive Conformations and Three-Dimensional Structure-Activity Relationships Models for Future Recognition of Abuse Drugs
Tomasevic, Nevena; Vujovic, Maja; Kostic, Emilija; Ragavendran, Venkatesan; Arsic, Biljana; Matic, Sanja Lj.; Bozovic, Mijat; Fioravanti, Rossella; Proia, Eleonora; Ragno, Rino; Mladenovic, Milan
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SaveEffect of Different Soil Treatments on Production and Chemical Composition of Essential Oils Extracted from Foeniculum vulgare Mill., Origanum vulgare L. and Thymus vulgaris L.
Raffo, Antonio; Sapienza, Filippo Umberto; Astolfi, Roberta; Lombardi, Gabriele; Fraschetti, Caterina; Bozovic, Mijat; Artini, Marco; Papa, Rosanna; Trecca, Marika; Fiorentino, Simona; Vecchiarelli, Valerio; Papalini, Claudia; Selan, Laura; Ragno, Rino
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SaveBcl-2 family inhibitors sensitize human cancer models to therapy
Valentini, Elisabetta; Di Martile, Marta; Brignone, Matteo; Di Caprio, Marica; Manni, Isabella; Chiappa, Michela; Sergio, Ilaria; Chiacchiarini, Martina; Bazzichetto, Chiara; Conciatori, Fabiana; D'Aguanno, Simona; D'Angelo, Carmen; Ragno, Rino; Russillo, Michelangelo; Colotti, Gianni; Marchesi, Francesco; Bellone, Maria Laura; Dal Piaz, Fabrizio; Felli, Maria Pia; Damia, Giovanna; Del Bufalo, Donatella
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SaveIn Vivo Antiphytoviral and Aphid Repellency Activity of Essential Oils and Hydrosols from Mentha suaveolens and Foeniculum vulgare to Control Zucchini Yellow Mosaic Virus and Its Vector Aphis gossypii
Taglienti, Anna; Donati, Livia; Dragone, Immacolata; Ferretti, Luca; Gentili, Andrea; Araniti, Fabrizio; Sapienza, Filippo; Astolfi, Roberta; Fiorentino, Simona; Vecchiarelli, Valerio; Papalini, Claudia; Ragno, Rino; Bertin, Sabrina
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SavePyrimidine thioethers: A novel class of antidepressant agents, endowed with anxiolytic, performance enhancing and nootropic activity
Fioravanti, Rossella; Proia, Eleonora; Tyurenkov, Ivan N.; V. Kurkin, Denis; Bakulin, Dmitry A.; Kovalev, Nikolay S.; Sheikin, Dmitry S.; Kirillov, Ivan A.; Nawrozkij, Maxim B.; Vernigora, Andrey A.; Brunilina, Leila L.; Fiorentino, Francesco; Mladenovic, Milan; Rotili, Dante; Ragno, Rino
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