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J

Jef Rozenski

rega institute

40H-index
284Paper Count
7.2KCitation Count
Published Papers 95
Publication Date
An automated dual-mode platform for affinity-based screening of natural products using a pressure-driven strategy
err2026-06-20
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PREAI
errJingyi Jian; Kris Wolfs; Francesco Ciacci; Hao Tian; Jef Rozenski; Ivo F.J. Vankelecom; Zhengjin Jiang; Erwin Adams; Ann Van Schepdael
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Monocyte-hitchhiking system for the targeted delivery of paclitaxel-loaded PLGA nanoparticles to glioblastoma in mice
err2026-04-22
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errOAAI
errXanthippi Koutsoumpou; Vincent Lenders; Akshaya Lakshmi Krishnamoorthy; Ine Vlaeminck; Jef Rozenski; Floriana De Marco; Carla Rios Luci; Filipa Roque Goncalves; Hermon Girmatsion; Marta Ciwinksa; Max Nobis; Colinda L. G. J. Scheele; Stefaan J. Soenen; Steven De Vleeschouwer; Bella B. Manshian
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Tuning i-motif folding and stability with acyclic phosphonate-linked (ZNA) cytidine residues
err2025-10-07
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errOAAI
errMarlies Derden †; Sten Reynders †; Jérôme Rihon; Xinlu Li; Frédérick Coosemans; Jef Rozenski; Piet Herdewijn; Elisabetta Groaz †; Eveline Lescrinier †
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Structure–Activity Relationship Study of 3-Alkynyl-6-aryl-isothiazolo[4,3-b]pyridines as Dual Inhibitors of the Lipid Kinases PIKfyve and PIP4K2C
err2025-09-21
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errOAAI
errDemian Kalebic; Ling-Jie Gao; Belén Martinez-Gualda; Marwah Karim; Sirle Saul; Do Hoang Nhu Tran; Jef Rozenski; Leentje Persoons; Dominique Schols; Wim Dehaen; Shirit Einav; Steven De Jonghe
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Discovery and exploration of disubstituted [1,2,5]oxadiazolo-[3,4-b]pyrazines as novel C-C chemokine receptor type 5 signaling inhibitors targeting the intracellular allosteric binding pocket
err2025-07-01
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PREAI
errBillen, Margaux; Reynders, Sten; Claes, Sandra; Kleinboelting, Silke; Rozenski, Jef; Bulai, Radu-George; Rocca, Edoardo; Homer, Natalie Z. M.; Webster, Scott P.; Kaminski, Tim P.; Lescrinier, Eveline; Schols, Dominique; Verwilst, Peter
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A guanidine-based coronavirus replication inhibitor which targets the nsp15 endoribonuclease and selects for interferon-susceptible mutant viruses
err2025-02-11
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errOAAI
errVan Loy, Benjamin; Pujol, Eugenia; Kamata, Kenichi; Lee, Xiao Yin; Bakirtzoglou, Nikolai; Van Berwaer, Ria; Vandeput, Julie; Mestdagh, Cato; Persoons, Leentje; De Wijngaert, Brent; Goovaerts, Quinten; Noppen, Sam; Jacquemyn, Maarten; Ahmadzadeh, Kourosh; Bernaerts, Eline; Martin-Lopez, Juan; Escriche, Celia; Vanmechelen, Bert; Krasniqi, Besir; Singh, Abhimanyu K.; Daelemans, Dirk; Maes, Piet; Matthys, Patrick; Dehaen, Wim; Rozenski, Jef; Das, Kalyan; Voet, Arnout; Vazquez, Santiago; Naesens, Lieve; Stevaert, Annelies
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Assessment of in vitro antimicrobial activity of clindamycin metabolites against Staphylococcus species
err2023-10-01
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errOAAI
errVan De Sijpe, Greet; Mylemans, Marnix; Alvarez, Laura Armengol; Ozbey, Agustos Cetin; Allegaert, Karel; Rozenski, Jef; Annaert, Pieter; Desmet, Stefanie; Spriet, Isabel
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Nucleoside Derivatives of 2,6-Diaminopurine Antivirals: Base-Modified Nucleosides with Broad-Spectrum Antimicrobial Properties
err2023-06-02
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PREAI
errMartina, Maria Grazia; Giammarino, Federica; Vicenti, Ilaria; Groaz, Elisabetta; Rozenski, Jef; Incerti, Matteo; Sannio, Filomena; Docquier, Jean Denis; Zazzi, Maurizio; Radi, Marco
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Modularity of RBC hitchhiking with polymeric nanoparticles: testing the limits of non-covalent adsorption
err2022-07-16
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errOAAI
errLenders, Vincent; Escudero, Remei; Koutsoumpou, Xanthippi; Alvarez, Laura Armengol; Rozenski, Jef; Soenen, Stefaan J.; Zhao, Zongmin; Mitragotri, Samir; Baatsen, Pieter; Allegaert, Karel; Toelen, Jaan; Manshian, Bella B.
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Ways to Improve Insights into Clindamycin Pharmacology and Pharmacokinetics Tailored to Practice
err2022-05-21
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errOAAI
errArmengol Alvarez, Laura; van de Sijpe, Greet; Desmet, Stefanie; Metsemakers, Willem-Jan; Spriet, Isabel; Allegaert, Karel; Rozenski, Jef
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Exploring the dNTP -binding site of HIV-1 reverse transcriptase for inhibitor design
err2021-12-01
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PREAI
errGu, Weijie; Martinez, Sergio; Singh, Abhimanyu K.; Nguyen, Hoai; Rozenski, Jef; Schols, Dominique; Herdewijn, Piet; Das, Kalyan; De Jonghe, Steven
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Overview of in-capillary enzymatic reactions using capillary electrophoresis
err2021-09-23
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errOAAI
errRozenski, Jef; Asfaw, Adissu Alemayehu; Van Schepdael, Ann
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Synthesis and structure-activity studies of novel anhydrohexitol-based Leucyl-tRNA synthetase inhibitors
err2021-02-01
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errOAAI
errDe Ruysscher, Dries; Pang, Luping; Lenders, Stijn M. G.; Cappoen, Davie; Cos, Paul; Rozenski, Jef; Strelkov, Sergei, V; Weeks, Stephen D.; Van Aerschot, Arthur
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Recent progress in the LC-MS/MS analysis of oxidative stress biomarkers
err2020-12-28
err19
errOAAI
errAndries, Asmin; Rozenski, Jef; Vermeersch, Pieter; Mekahli, Djalila; Van Schepdael, Ann
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Synthesis and Biological Evaluation of 1,3-Dideazapurine-Like 7-Amino-5-Hydroxymethyl-Benzimidazole Ribonucleoside Analogues as Aminoacyl-tRNA Synthetase Inhibitors
err2020-10-16
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errOAAI
errZhang, Baole; Pang, Luping; Nautiyal, Manesh; De Graef, Steff; Gadakh, Bharat; Lescrinier, Eveline; Rozenski, Jef; Strelkov, Sergei V.; Weeks, Stephen D.; Van Aerschot, Arthur
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Phenyltriazole-functionalized sulfamate inhibitors targeting tyrosyl- or isoleucyl-tRNA synthetase
err2020-08-01
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errOAAI
errDe Ruysscher, Dries; Pang, Luping; Mattelaer, Charles-Alexandre; Nautiyal, Manesh; De Graef, Steff; Rozenski, Jef; Strelkov, Sergei, V; Lescrinier, Eveline; Weeks, Stephen D.; Van Aerschot, Arthur
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Rational design of an XNA ligase through docking of unbound nucleic acids to toroidal proteins (vol 47, pg 7130, 2019)
err2019-11-12
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errOAAI
errVanmeert, Michiel; Razzokov, Jamoliddin; Mirza, Muhammad Usman; Weeks, Stephen D.; Schepers, Guy; Bogaerts, Annemie; Rozenski, Jef; Froeyen, Mathy; Herdewijn, Piet; Pinheiro, Vitor B.; Lescrinier, Eveline
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Synthesis and Biological Evaluation of Lipophilic Nucleoside Analogues as Inhibitors of Aminoacyl-tRNA Synthetases
err2019-10-09
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errOAAI
errNautiyal, Manesh; Gadakh, Bharat; De Graef, Steff; Pang, Luping; Khan, Masroor; Xun, Yi; Rozenski, Jef; Van Aerschot, Arthur
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Acylated sulfonamide adenosines as potent inhibitors of the adenylate-forming enzyme superfamily
err2019-07-01
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errOAAI
errDe Ruysscher, Dries; Pang, Luping; De Graef, Steff; Nautiyal, Manesh; De Borggraeve, Wim M.; Rozenski, Jef; Strelkov, Sergei V.; Weeks, Stephen D.; Van Aerschot, Arthur
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Invading Escherichia coli Genetics with a Xenobiotic Nucleic Acid Carrying an Acyclic Phosphonate Backbone (ZNA)
err2019-06-28
err28
errOAAI
errLuo, Min; Groaz, Elisabetta; Froeyen, Mathy; Pezo, Valerie; Jaziri, Faten; Leonczak, Piotr; Schepers, Guy; Rozenski, Jef; Marliere, Philippe; Herdewijn, Piet
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