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Vincenzo Summa

department of pharmacy

32H-index
158Paper Count
4.7KCitation Count
Published Papers 64
Publication Date
Efficient and scalable photochemical coupling of pinacol and aza-pinacol in continuous-flow
err2026-07-11
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errAntonella Ilenia Alfano; Luigi Maria Moreno Tufano; Vincenzo Summa; Margherita Brindisi
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F2F-202; a Selective Histone Deacetylase 6 (HDAC6) Inhibitor; Behaves as an Arrow with Multiple Tips against Azole-Resistant C. albicans: Modulation of Yeast-to-Hyphae Transition; Trailing Effect; and Oxidative Stress
err2026-05-22
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errSimona Barone; Baptiste Mateu; Marialuisa Piccolo; Anna Guadagni; Carlo Irace; Francesca Lembo; Vincenzo Summa; Elisabetta Buommino; Margherita Brindisi
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Fine-tuning the combination of novel spirocyclic capping moieties and heterocyclic zinc binding groups for selective HDAC6 inhibition: design, synthesis, kinetic and biological studies.
err2026-03-29
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errSimona Barone; Ivana Bello; Gessica Filocamo; Carmen Cerchia; Anna Guadagni; Mirko Brunetti; Emanuela Cosentino; Maria Hanl; Beate König; Camilla Esposito; Linda Schäker-Hübner; Vincenzo Summa; Elisabetta Panza; Finn K. Hansen; Margherita Brindisi
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Selective HDAC6 Inhibition by Mesinostat Impairs Tumor Growth and Stemness in Triple-Negative Breast Cancer
err2025-12-02
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errIvana Bello; Simona Barone; Anna Guadagni; Camilla Esposito; Morena D’Ariano; Martina Smimmo; Giuseppe Cirino; Vincenzo Summa; Margherita Brindisi; Elisabetta Panza
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The role of dopaminergic signalling from physiology to neuroprotection in acute and chronic disorders
err2025-11-15
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errMartina Di Nunzio; Maria Lidia Mignogna; Marco Bacigaluppi; Paola Panina-Bordignon; Paolo Ragonese; Luca Muzio; Vincenzo Summa; Gianvito Martino
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METTL16-mediated inhibition of MXD4 promotes leukemia through activation of the MYC-MAX axis
err2025-09-14
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errGuglielmo Bove; Mehrad Babaei; Alberto Bueno-Costa; Sajid Amin; Nicla Simonelli; Rosaria Benedetti; Carmela Dell’Aversana; Mariarosaria Conte; Liliana Montella; Vincenzo Summa; Margherita Brindisi; Maria Rosaria Del Sorbo; Marco Crepaldi; Gregorio Favale; Nuria Profitos-Peleja; Vincenzo Carafa; Gaël Roué; Fortunato Ciardiello; Annalisa Capuano; Hendrik G. Stunnenberg; Wouter L. Megchelenbrink; Angela Nebbioso; Manel Esteller; Lucia Altucci; Nunzio Del Gaudio
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Challenging triple negative breast cancer through HDAC6 selective inhibition: Novel cap-group identification, structure-activity relationships, computational and biological studies
err2025-05-10
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errBarone, Simona; Bello, Ivana; Guadagni, Anna; Cerchia, Carmen; Filocamo, Gessica; Cassese, Emilia; Alfano, Antonella Ilenia; Esposito, Camilla; Morel, Alvaro Javier Feliz; Brunetti, Mirko; Lavecchia, Antonio; Summa, Vincenzo; Panza, Elisabetta; Brindisi, Margherita
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Integrating Surface Plasmon Resonance and Docking Analysis for Mechanistic Insights of Tryptase Inhibitors
err2025-03-17
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errPorta, Alessia; Manelfi, Candida; Talarico, Carmine; Beccari, Andrea Rosario; Brindisi, Margherita; Summa, Vincenzo; Iaconis, Daniela; Gobbi, Marco; Beeg, Marten
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Tackling triple negative breast cancer with HDAC inhibitors: 6 is the isoform!
err2024-12-01
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errGuadagni, Anna; Barone, Simona; Alfano, Antonella Ilenia; Pelliccia, Sveva; Bello, Ivana; Panza, Elisabetta; Summa, Vincenzo; Brindisi, Margherita
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Nutraceutical formulation based on a synergic combination of melatonin and palmitoylethanolamide for the management of allergic events
err2024-08-27
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errMaisto, Maria; Piccolo, Vincenzo; Marzocchi, Adua; Maresca, Daniela Claudia; Romano, Benedetta; Summa, Vincenzo; Tenore, Gian Carlo; Ercolano, Giuseppe; Ianaro, Angela
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A Rapid and Reliable Spectrofluorimetric Method to Measure the Urinary Lactulose/Mannitol Ratio for Dysbiosis Assessment
err2024-07-13
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errCerrato, Lorenzo Marino; Schiano, Elisabetta; Iannuzzo, Fortuna; Tenore, Gian Carlo; Summa, Vincenzo; Daglia, Maria; Novellino, Ettore; Stornaiuolo, Mariano
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Optimization and Validation of Procyanidins Extraction and Phytochemical Profiling of Seven Herbal Matrices of Nutraceutical Interest
err2024-05-10
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errKeivani, Niloufar; Piccolo, Vincenzo; Marzocchi, Adua; Maisto, Maria; Tenore, Gian Carlo; Summa, Vincenzo
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Characterization and quantification of intact glucosinolates in Catozza rapeseeds: A promising food matrix for nutraceuticals development as a source of hydrogen sulfide
err2024-05-01
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errPiccolo, Vincenzo; Maisto, Maria; Cerrato, Lorenzo Marino; Esposito, Erika; Panza, Elisabetta; Sorrentino, Raffaella; Mitidieri, Emma; Bianca, Roberta d'Emmanuele di Villa; Tenore, Gian Carlo; Summa, Vincenzo
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Phytochemical investigation and antioxidant properties of unripe tomato cultivars (Solanum lycopersicum L.)
err2024-04-01
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errPiccolo, Vincenzo; Maisto, Maria; Schiano, Elisabetta; Iannuzzo, Fortuna; Keivani, Niloufar; Rigano, Maria Manuela; Santini, Antonello; Novellino, Ettore; Tenore, Gian Carlo; Summa, Vincenzo
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Unveiling the modulation of Pseudomonas aeruginosa virulence and biofilm formation by selective histone deacetylase 6 inhibitors
err2024-02-02
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errBarone, Simona; Mateu, Baptiste; Turco, Luigia; Pelliccia, Sveva; Lembo, Francesca; Summa, Vincenzo; Buommino, Elisabetta; Brindisi, Margherita
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The Urine Metabolome of R6/2 and zQ175DN Huntington's Disease Mouse Models
err2023-08-18
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errSpeziale, Roberto; Montesano, Camilla; Di Pietro, Giulia; Cicero, Daniel Oscar; Summa, Vincenzo; Monteagudo, Edith; Orsatti, Laura
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Broad-spectrum coronavirus 3C-like protease peptidomimetic inhibitors effectively block SARS-CoV-2 replication in cells: Design, synthesis, biological evaluation, and X-ray structure determination
err2023-05-01
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errStefanelli, Irina; Corona, Angela; Cerchia, Carmen; Cassese, Emilia; Improta, Salvatore; Costanzi, Elisa; Pelliccia, Sveva; Morasso, Stefano; Esposito, Francesca; Paulis, Annalaura; Scognamiglio, Sante; Leva, Francesco Saverio Di; Storici, Paola; Brindisi, Margherita; Tramontano, Enzo; Cannalire, Rolando; Summa, Vincenzo
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Photo-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds
err2023-04-12
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PREAI
errAlfano, Antonella Ilenia; Pelliccia, Sveva; Rossino, Giacomo; Chianese, Orazio; Summa, Vincenzo; Collina, Simona; Brindisi, Margherita
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Nirmatrelvir treatment of SARS-CoV-2-infected mice blunts antiviral adaptive immune responses
err2023-03-22
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errFumagalli, Valeria; Di Lucia, Pietro; Rava, Micol; Marotta, Davide; Bono, Elisa; Grassi, Stefano; Donnici, Lorena; Cannalire, Rolando; Stefanelli, Irina; Ferraro, Anastasia; Esposito, Francesca; Pariani, Elena; Inverso, Donato; Montesano, Camilla; Delbue, Serena; Perlman, Stanley; Tramontano, Enzo; De Francesco, Raffaele; Summa, Vincenzo; Guidotti, Luca G.; Iannacone, Matteo
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