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SaveLead Optimization of Positive Allosteric KV7.2/3 Channel Modulators toward Improved Balance of Lipophilicity and Aqueous Solubility
Lemke, Jana; Mengers, Nadine; Schmidt, Louis; Schulig, Lukas; Koenig, Stefanie; Rosendahl, Pascal; Bartz, Frieda-Marie; Garscha, Ulrike; Bednarski, Patrick J.; Link, Andreas
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SaveStructure-Guided Engineering of a Versatile Urethanase Improves Its Polyurethane Depolymerization Activity
Li, ZS; Han, X; Cong, L; Singh, P; Paiva, P; Branson, Y; Li, WS; Chen, YY; Jaradat, DMM; Lennartz, F; Bayer, T; Schmidt, L; Garscha, U; You, S; Fernandes, PA; Ramos, MJ; Bornscheuer, UT; Weber, G; Wei, R; Liu, WD
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SaveStructural Elucidation of a Metagenomic Urethanase and Its Engineering Towards Enhanced Hydrolysis Profiles
Bayer, Thomas; Palm, Gottfried J.; Berndt, Leona; Meinert, Hannes; Branson, Yannick; Schmidt, Louis; Cziegler, Clemens; Somvilla, Ina; Zurr, Celine; Graf, Leonie G.; Janke, Una; Badenhorst, Christoffel P. S.; Koenig, Stefanie; Delcea, Mihaela; Garscha, Ulrike; Wei, Ren; Lammers, Michael; Bornscheuer, Uwe T.
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SaveIdentification of 2,4-Dinitro-Biphenyl-Based Compounds as MAPEG Inhibitors
Di Micco, Simone; Terracciano, Stefania; Pierri, Martina; Cantone, Vincenza; Liening, Stefanie; Koenig, Stefanie; Garscha, Ulrike; Hofstetter, Robert Klaus; Koeberle, Andreas; Werz, Oliver; Bruno, Ines; Bifulco, Giuseppe
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SaveSynthesis and structure-activity relationships for some novel diflapolin derivatives with benzimidazole subunit
Vieider, Lisa; Zoeller, Eva; Romp, Erik; Schoenthaler, Martin; Hernandez-Olmos, Victor; Temml, Veronika; Hasenoehrl, Thomas; Schuster, Daniela; Werz, Oliver; Garscha, Ulrike; Matuszczak, Barbara
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SaveExploration of Long-Chain Vitamin E Metabolites for the Discovery of a Highly Potent, Orally Effective, and Metabolically Stable 5-LOX Inhibitor that Limits Inflammation
Neukirch, Konstantin; Alsabil, Khaled; Dinh, Chau-Phi; Bilancia, Rossella; Raasch, Martin; Ville, Alexia; Cerqua, Ida; Viault, Guillaume; Breard, Dimitri; Pace, Simona; Temml, Veronika; Brunner, Elena; Jordan, Paul M.; Marques, Marta C.; Loeser, Konstantin; Gollowitzer, Andre; Permann, Stephan; Gerstmeier, Jana; Lorkowski, Stefan; Stuppner, Hermann; Garscha, Ulrike; Rodrigues, Tiago; Bernardes, Goncalo J. L.; Schuster, Daniela; Seraphin, Denis; Richomme, Pascal; Rossi, Antonietta; Mosig, Alexander S.; Roviezzo, Fiorentina; Werz, Oliver; Helesbeux, Jean-Jacques; Koeberle, Andreas
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SaveModulation of microRNA processing by 5-lipoxygenase
Uebbing, Stella; Kreiss, Marius; Scholl, Friederike; Haefner, Ann-Kathrin; Sueruen, Duran; Garscha, Ulrike; Werz, Oliver; Basavarajappa, Devaraj; Samuelsson, Bengt; Radmark, Olof; Suess, Beatrix; Steinhilber, Dieter
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SaveTargeting biosynthetic networks of the proinflammatory and proresolving lipid metabolome
Werner, Markus; Jordan, Paul M.; Romp, Erik; Czapka, Anna; Rao, Zhigang; Kretzer, Christian; Koeberle, Andreas; Garscha, Ulrike; Pace, Simona; Claesson, Hans-Erik; Serhan, Charles N.; Werz, Oliver; Gerstmeier, Jana
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SaveMelleolides from Honey Mushroom Inhibit 5-Lipoxygenase via Cys159
Koenig, Stefanie; Romp, Erik; Krauth, Verena; Ruehl, Michael; Doerfer, Maximilian; Liening, Stefanie; Hofmann, Bettina; Haefner, Ann-Kathrin; Steinhilber, Dieter; Karas, Michael; Garscha, Ulrike; Hoffmeister, Dirk; Werz, Oliver
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