Not logged in Share Save
Kronopolitides A-F, a Family of 36-Membered Polyol Macrolides with Antiparasitic Activity against Chagas Disease Perez-Bonilla, Mercedes; Sanchez-Hidalgo, Marina; Gonzalez, Ignacio; Martin, Jesus; Tormo, Jose R.; Cho, Ahreum; Byun, Soo Young; Shum, David; Ioset, Jean-Robert; Reyes, Fernando; Genilloud, Olga Share Save
Efficient constitution of a library of rotenoid analogs active against Trypanosoma cruzi from a digitalized plant extract collection Gaudry, Arnaud; Marcourt, Laurence; Kaiser, Marcel; Fluckiger, Julien; David, Bruno; Grondin, Antonio; Ioset, Jean-Robert; Maser, Pascal; Queiroz, Emerson Ferreira; Allard, Pierre-Marie; Wolfender, Jean-Luc Share Save
A Sample-Centric and Knowledge-Driven Computational Framework for Natural Products Drug Discovery Gaudry, Arnaud; Pagni, Marco; Mehl, Florence; Moretti, Sebastien; Quiros-Guerrero, Luis-Manuel; Cappelletti, Luca; Rutz, Adriano; Kaiser, Marcel; Marcourt, Laurence; Queiroz, Emerson Ferreira; Ioset, Jean-Robert; Grondin, Antonio; David, Bruno; Wolfender, Jean-Luc; Allard, Pierre-Marie Share Save
Need for a Standardized Translational Drug Development Platform: Lessons Learned from the Repurposing of Drugs for COVID-19 Assmus, Frauke; Driouich, Jean-Selim; Abdelnabi, Rana; Vangeel, Laura; Touret, Franck; Adehin, Ayorinde; Chotsiri, Palang; Cochin, Maxime; Foo, Caroline S.; Jochmans, Dirk; Kim, Seungtaek; Luciani, Lea; Moureau, Gregory; Park, Soonju; Petit, Paul-Remi; Shum, David; Wattanakul, Thanaporn; Weynand, Birgit; Fraisse, Laurent; Ioset, Jean-Robert; Mowbray, Charles E.; Owen, Andrew; Hoglund, Richard M.; Tarning, Joel; de Lamballerie, Xavier; Nougairede, Antoine; Neyts, Johan; Sjo, Peter; Escudie, Fanny; Scandale, Ivan; Chatelain, Eric Share Save
Novel benzoxaborole, nitroimidazole and aminopyrazoles with activity against experimental cutaneous leishmaniasis Van Bocxlaer, Katrien; Caridha, Diana; Black, Chad; Vesely, Brian; Leed, Susan; Sciotti, Richard J.; Wijnant, Gert-Jan; Yardley, Vanessa; Braillard, Stephanie; Mowbray, Charles E.; Ioset, Jean-Robert; Croft, Simon L. Share Save
Share Save
Share Save
Share Save
Synthesis and evaluation of analogs of the phenylpyridazinone NPD-001 as potent trypanosomal TbrPDEB1 phosphodiesterase inhibitors and in vitro trypanocidals Veerman, Johan; van den Bergh, Toine; Orrling, Kristina M.; Jansen, Chimed; Cos, Paul; Maes, Louis; Chatelain, Eric; Ioset, Jean-Robert; Edink, Ewald E.; Tenor, Hermann; Seebeck, Thomas; de Esch, Iwan; Leurs, Rob; Sterk, Geert Jan Share Save
Share Save
Share Save
Share Save
Share Save
Selection and optimization of hits from a high-throughput phenotypic screen against Trypanosoma cruzi Keenan, Martine; Alexander, Paul W.; Chaplin, Jason H.; Abbott, Michael J.; Diao, Hugo; Wang, Zhisen; Best, Wayne M.; Perez, Catherine J.; Cornwall, Scott M. J.; Keatley, Sarah K.; Thompson, R. C. Andrew; Charman, Susan A.; White, Karen L.; Ryan, Eileen; Chen, Gong; Ioset, Jean-Robert; von Geldern, Thomas W.; Chatelain, Eric Share Save
Share Save
Catechol Pyrazolinones as Trypanocidals: Fragment-Based Design, Synthesis, and Pharmacological Evaluation of Nanomolar Inhibitors of Trypanosomal Phosphodiesterase B1 Orrling, Kristina M.; Jansen, Chimed; Vu, Xuan Lan; Balmer, Vreni; Bregy, Patrick; Shanmugham, Anitha; England, Paul; Bailey, David; Cos, Paul; Maes, Louis; Adams, Emily; van den Bogaart, Erika; Chatelain, Eric; Ioset, Jean-Robert; van de Stolpe, Andrea; Zorg, Stephanie; Veerman, Johan; Seebeck, Thomas; Sterk, Geert Jan; de Esch, Iwan J. P.; Leurs, Rob Share Save
Novel 3-Nitro-1H-1,2,4-triazole-Based Amides and Sulfonamides as Potential Antitrypanosomal Agents Papadopoulou, Maria V.; Bloomer, William D.; Rosenzweig, Howard S.; Chatelain, Eric; Kaiser, Marcel; Wilkinson, Shane R.; McKenzie, Caroline; Ioset, Jean-Robert Share Save
Share Save
Share Save