arrow
Back
J

Jean‐Robert Ioset

drugs for neglected diseases initiative

35H-index
78Paper Count
2.8KCitation Count
Published Papers 22
Publication Date
Kronopolitides A-F, a Family of 36-Membered Polyol Macrolides with Antiparasitic Activity against Chagas Disease
err2025-12-01
err0
PREAI
errPerez-Bonilla, Mercedes; Sanchez-Hidalgo, Marina; Gonzalez, Ignacio; Martin, Jesus; Tormo, Jose R.; Cho, Ahreum; Byun, Soo Young; Shum, David; Ioset, Jean-Robert; Reyes, Fernando; Genilloud, Olga
errShare
errSave
Efficient constitution of a library of rotenoid analogs active against Trypanosoma cruzi from a digitalized plant extract collection
err2025-01-01
err0
errOAAI
errGaudry, Arnaud; Marcourt, Laurence; Kaiser, Marcel; Fluckiger, Julien; David, Bruno; Grondin, Antonio; Ioset, Jean-Robert; Maser, Pascal; Queiroz, Emerson Ferreira; Allard, Pierre-Marie; Wolfender, Jean-Luc
errShare
errSave
A Sample-Centric and Knowledge-Driven Computational Framework for Natural Products Drug Discovery
err2024-02-20
err5
errOAAI
errGaudry, Arnaud; Pagni, Marco; Mehl, Florence; Moretti, Sebastien; Quiros-Guerrero, Luis-Manuel; Cappelletti, Luca; Rutz, Adriano; Kaiser, Marcel; Marcourt, Laurence; Queiroz, Emerson Ferreira; Ioset, Jean-Robert; Grondin, Antonio; David, Bruno; Wolfender, Jean-Luc; Allard, Pierre-Marie
errShare
errSave
Need for a Standardized Translational Drug Development Platform: Lessons Learned from the Repurposing of Drugs for COVID-19
err2022-08-12
err4
errOAAI
errAssmus, Frauke; Driouich, Jean-Selim; Abdelnabi, Rana; Vangeel, Laura; Touret, Franck; Adehin, Ayorinde; Chotsiri, Palang; Cochin, Maxime; Foo, Caroline S.; Jochmans, Dirk; Kim, Seungtaek; Luciani, Lea; Moureau, Gregory; Park, Soonju; Petit, Paul-Remi; Shum, David; Wattanakul, Thanaporn; Weynand, Birgit; Fraisse, Laurent; Ioset, Jean-Robert; Mowbray, Charles E.; Owen, Andrew; Hoglund, Richard M.; Tarning, Joel; de Lamballerie, Xavier; Nougairede, Antoine; Neyts, Johan; Sjo, Peter; Escudie, Fanny; Scandale, Ivan; Chatelain, Eric
errShare
errSave
Novel benzoxaborole, nitroimidazole and aminopyrazoles with activity against experimental cutaneous leishmaniasis
err2019-12-01
err55
errOAAI
errVan Bocxlaer, Katrien; Caridha, Diana; Black, Chad; Vesely, Brian; Leed, Susan; Sciotti, Richard J.; Wijnant, Gert-Jan; Yardley, Vanessa; Braillard, Stephanie; Mowbray, Charles E.; Ioset, Jean-Robert; Croft, Simon L.
errShare
errSave
Addressing the most neglected diseases through an open research model: The discovery of fenarimols as novel drug candidates for eumycetoma
err2018-04-26
err30
errOAAI
errLim, Wilson; Melse, Youri; Konings, Mickey; Hung Phat Duong; Eadie, Kimberly; Laleu, Benoit; Perry, Benjamin; Todd, Matthew H.; Ioset, Jean-Robert; van de Sande, Wendy W. J.
errShare
errSave
errShare
errSave
Assessing anti-T. cruzi candidates in vitro for sterile cidality
err2016-12-01
err37
errOAAI
errCal, Monica; Ioset, Jean-Robert; Fugi, Matthia A.; Maser, Pascal; Kaiser, Marcel
errShare
errSave
Synthesis and evaluation of analogs of the phenylpyridazinone NPD-001 as potent trypanosomal TbrPDEB1 phosphodiesterase inhibitors and in vitro trypanocidals
err2016-04-01
err36
errOAAI
errVeerman, Johan; van den Bergh, Toine; Orrling, Kristina M.; Jansen, Chimed; Cos, Paul; Maes, Louis; Chatelain, Eric; Ioset, Jean-Robert; Edink, Ewald E.; Tenor, Hermann; Seebeck, Thomas; de Esch, Iwan; Leurs, Rob; Sterk, Geert Jan
errShare
errSave
Discovery of potent nitrotriazole-based antitrypanosomal agents: In vitro and in vivo evaluation
err2015-10-01
err44
errOAAI
errPapadopoulou, Maria V.; Bloomer, William D.; Rosenzweig, Howard S.; O'Shea, Ivan P.; Wilkinson, Shane R.; Kaiser, Marcel; Chatelain, Eric; Ioset, Jean-Robert
errShare
errSave
Development and Validation of a Novel Leishmania donovani Screening Cascade for High-Throughput Screening Using a Novel Axenic Assay with High Predictivity of Leishmanicidal Intracellular Activity
err2015-09-25
err29
errOAAI
errNuehs, Andrea; De Rycker, Manu; Manthri, Sujatha; Comer, Eamon; Scherer, Christina A.; Schreiber, Stuart L.; Ioset, Jean-Robert; Gray, David W.
errShare
errSave
Novel 3-Nitrotriazole-Based Amides and Carbinols as Bifunctional Antichagasic Agents
err2015-01-23
err54
errOAAI
errPapadopoulou, Maria V.; Bloomer, William D.; Lepesheva, Galina I.; Rosenzweig, Howard S.; Kaiser, Marcel; Aguilera-Venegas, Benjamin; Wilkinson, Shane R.; Chatelain, Eric; Ioset, Jean-Robert
errShare
errSave
Novel 3-nitro-1H-1,2,4-triazole-based piperazines and 2-amino-1,3-benzothiazoles as antichagasic agents
err2013-11-01
err42
errOAAI
errPapadopoulou, Maria V.; Bloomer, William D.; Rosenzweig, Howard S.; Kaiser, Marcel; Chatelain, Eric; Ioset, Jean-Robert
errShare
errSave
Selection and optimization of hits from a high-throughput phenotypic screen against Trypanosoma cruzi
err2013-10-21
err21
PREAI
errKeenan, Martine; Alexander, Paul W.; Chaplin, Jason H.; Abbott, Michael J.; Diao, Hugo; Wang, Zhisen; Best, Wayne M.; Perez, Catherine J.; Cornwall, Scott M. J.; Keatley, Sarah K.; Thompson, R. C. Andrew; Charman, Susan A.; White, Karen L.; Ryan, Eileen; Chen, Gong; Ioset, Jean-Robert; von Geldern, Thomas W.; Chatelain, Eric
errShare
errSave
Identification of Compounds with Anti-Proliferative Activity against Trypanosoma brucei brucei Strain 427 by a Whole Cell Viability Based HTS Campaign
err2012-11-29
err83
errOAAI
errSykes, Melissa L.; Baell, Jonathan B.; Kaiser, Marcel; Chatelain, Eric; Moawad, Sarah R.; Ganame, Danny; Ioset, Jean-Robert; Avery, Vicky M.
errShare
errSave
Catechol Pyrazolinones as Trypanocidals: Fragment-Based Design, Synthesis, and Pharmacological Evaluation of Nanomolar Inhibitors of Trypanosomal Phosphodiesterase B1
err2012-10-08
err56
PREAI
errOrrling, Kristina M.; Jansen, Chimed; Vu, Xuan Lan; Balmer, Vreni; Bregy, Patrick; Shanmugham, Anitha; England, Paul; Bailey, David; Cos, Paul; Maes, Louis; Adams, Emily; van den Bogaart, Erika; Chatelain, Eric; Ioset, Jean-Robert; van de Stolpe, Andrea; Zorg, Stephanie; Veerman, Johan; Seebeck, Thomas; Sterk, Geert Jan; de Esch, Iwan J. P.; Leurs, Rob
errShare
errSave
Novel 3-Nitro-1H-1,2,4-triazole-Based Amides and Sulfonamides as Potential Antitrypanosomal Agents
err2012-05-23
err104
errOAAI
errPapadopoulou, Maria V.; Bloomer, William D.; Rosenzweig, Howard S.; Chatelain, Eric; Kaiser, Marcel; Wilkinson, Shane R.; McKenzie, Caroline; Ioset, Jean-Robert
errShare
errSave
errShare
errSave