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Michael Kassiou

Faculty of Science

63H-index
411Paper Count
1.4WCitation Count
Published Papers 189
Publication Date
Investigation of reported small molecule P2Y6 receptor antagonists
err2026-07-11
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errChianna Dane; André D.J. McKenzie; Andrew P. Montgomery; Jonathan Du; Eryn L. Werry; Michael Kassiou
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Flash Assembloids: A Rapid Biofabrication of a Platform for Modeling Early Glioblastoma Invasion at the Glioblastoma–Brain Organoid Interfaces
err2026-05-11
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errChao Liang; Henry Robert Howard; Shihui Chen; Won-Young Choi; Summer Cao; Arthur Chien; Kevin Zou; Michael Kassiou; Fabien Delerue; Ho Sang Jung; Yeonju Park; Young Mee Jung; Yong-Dae Kwon; Karrie M. Kiang; Gilberto Ka-Kit Leung; Ryohichi Sugimura; Ann-Na Cho; Sang Jin Lee
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Stability of the translocator protein 18 kDa density within cognitive circuits in brains of virally-suppressed people with HIV
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IF3.1
err2026-05-01
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PREAI
errRubin, Leah H.; Maki, Pauline M.; Du, Yong; Dastgheyb, Raha M.; Nam, Hwanhee; Rowe, Steven P.; Lesniak, Wojciech G.; Minn, Il; Hall, Andrew W.; Mathews, William B.; Kassiou, Michael; Dannals, Robert F.; Kassaye, Seble G.; Brown, Todd T.; Pomper, Martin G.; Coughlin, Jennifer M.
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Decreased functional connectivity in post-COVID syndrome patients with high neuroinflammatory activity
err2026-04-23
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errDenise Visser; Leo Pieperhoff; Luigi Lorenzini; Sandeep S.V. Golla; Sander C.J. Verfaillie; Anouk Verveen; Elsmarieke van de Giessen; Marijke E. den Hollander; Janneke Horn; Caroline M. van Heugten; Menno D. de Jong; Cees C. van den Wijngaard; Tessa van der Maaden; Maria Prins; Patrick Schober; Robert C. Schuit; Michael Kassiou; Albert D. Windhorst; Brent Appelman; Michele van Vugt
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Histone methyltransferase PRDM9 promotes survival of drug-tolerant persister cells in glioblastoma
err2025-12-15
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errGeorge L. Joun; Emma G. Kempe; Brianna Chen; Jayden R. Sterling; Ramzi H. Abbassi; Dana Friess; Matthew Singleton; Chandra Choudhury; Oana C. Marian; W. Daniel du Preez; Ariadna Recasens; Teleri Clark; Tian Y. Du; Jason K. K. Low; Hani Kim; Pengyi Yang; Jasmine Khor; Monira Hoque; Dinesh C. Indurthi; Mani Kuchibhotla; Ranjith Palanisamy; William T. Jorgensen; Andrew P. Montgomery; Jennifer R. Baker; Sarah L. Higginbottom; Eva Tomaskovic-Crook; Jeremy M. Crook; Lipin Loo; Bryan W. Day; G. Gregory Neely; Ernesto Guccione; Terrance G. Johns; Michael Kassiou; Yuchen Feng; Lachlan Harris; Anthony S. Don; Lenka Munoz
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The adamantane scaffold: Beyond a lipophilic moiety
err2025-07-01
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errDane, Chianna; Montgomery, Andrew P.; Kassiou, Michael
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PK 11195 derivatives: exploring the influence of amide and heterocyclic substitution on A147T TSPO discrimination
err2025-01-01
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PREAI
errSokias, Renee; Zhao, Andrea; Werry, Eryn L.; Montgomery, Andrew P.; Hibbs, David E.; Sullivan, Michael A.; Mckenzie, Andre D. J.; Cumbers, Grace A.; Allen, Beau M.; Danon, Jonathan J.; Kassiou, Michael
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P2X 7-receptor binding in new-onset and secondary progressive MS - a [11C]SMW139 PET study
err2024-12-05
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errLehto, Jussi; Aarnio, Richard; Tuisku, Jouni; Sucksdorff, Marcus; Koivumaeki, Esa Mikko; Nylund, Marjo; Helin, Semi; Rajander, Johan; Danon, Jonathan; Gilchrist, Jayson; Kassiou, Michael; Oikonen, Vesa; Airas, Laura
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Enhancing CNS mitophagy: drug development and disease-relevant models
err2024-11-01
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PREAI
errDhar, Krishayant S.; Townsend, Brendan; Montgomery, Andrew P.; Danon, Jonathan J.; Pagan, Julia K.; Kassiou, Michael
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Imaging the translocator protein 18 kDa within cognitive control and declarative memory circuits in virally suppressed people with HIV
errAIDS
IF3.1
err2024-10-10
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PREAI
errRubin, Leah H.; Maki, Pauline M.; Du, Yong; Sweeney, Shannon Eileen; O'Toole, Riley; Nam, Hwanhee; Lee, Hannah; Soule, Ana R.; Rowe, Steven P.; Lesniak, Wojciech G.; Minn, Il; Dastgheyb, Raha; Shorer, Eran F.; Wugalter, Katrina A.; Severson, Joan; Wu, Yunkou; Hall, Andrew W.; Mathews, William B.; Kassiou, Michael; Dannals, Robert F.; Kassaye, Seble G.; Brown, Todd T.; Bakker, Arnold; Pomper, Martin G.; Coughlin, Jennifer M.
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Structure-based drug design for TSPO: Challenges and opportunities
err2024-09-01
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errGiladi, Mia; Montgomery, Andrew P.; Kassiou, Michael; Danon, Jonathan J.
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Synthesis and Antitumour Evaluation of Tricyclic Indole-2-Carboxamides against Paediatric Brain Cancer Cells
err2024-08-08
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errHamilton, Alexander John; Lane, Samuel; Werry, Eryn L.; Suri, Amreena; Bailey, Anders W.; Merce, Clementine; Kadolsky, Ulrich; Payne, Alan D.; Kassiou, Michael; Sredni, Simone Treiger; Saxena, Alka; Gunosewoyo, Hendra
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An Investigation on Linker Modifications of Cyanoguanidine-Based P2X7 Receptor Antagonists
err2024-07-12
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errGarrett, Taylor R.; Gilchrist, Jayson; Mckenzie, Andre D. J.; Larik, Fayaz Ali; Danon, Jonathan J.; Werry, Eryn L.; Kassiou, Michael
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Structure-Activity Relationships, Deuteration, and Fluorination of Synthetic Cannabinoid Receptor Agonists Related to AKB48, 5F-AKB-48, and AFUBIATA
err2024-05-20
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PREAI
errSparkes, Eric; Maloney, Callan J.; Markham, Jack W.; Dane, Chianna; Boyd, Rochelle; Gilchrist, Jayson; Moir, Michael; Gordon, Rebecca; Luo, Jia Lin; Pike, Edward; Walker, Katelyn A.; Kassiou, Michael; Mcgregor, Iain S.; Kevin, Richard C.; Hibbs, David E.; Jorgensen, William T.; Banister, Samuel D.; Cairns, Elizabeth A.; Ametovski, Adam
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Glial reactivity in a mouse model of beta-amyloid deposition assessed by PET imaging of P2X7 receptor and TSPO using [11C]SMW139 and [18F]F-DPA (vol 14, 25, 2024)
err2024-05-03
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errAlzghool, Obada M.; Aarnio, Richard; Helin, Jatta S.; Wahlroos, Saara; Keller, Thomas; Matilainen, Markus; Solis, Junel; Danon, Jonathan J.; Kassiou, Michael; Snellman, Anniina; Solin, Olof; Rinne, Juha O.; Haaparanta-Solin, Merja
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Fragment-based drug discovery for disorders of the central nervous system: designing better drugs piece by piece
err2024-04-18
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errChan, Bill W. G. L.; Lynch, Nicholas B.; Tran, Wendy; Joyce, Jack M.; Savage, G. Paul; Meutermans, Wim; Montgomery, Andrew P.; Kassiou, Michael
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Glial reactivity in a mouse model of beta-amyloid deposition assessed by PET imaging of P2X7 receptor and TSPO using [11C]SMW139 and [18F]F-DPA
err2024-03-06
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errOAAI
errAlzghool, Obada M.; Aarnio, Richard; Helin, Jatta S.; Wahlroos, Saara; Keller, Thomas; Matilainen, Markus; Solis, Junel; Danon, Jonathan J.; Kassiou, Michael; Snellman, Anniina; Solin, Olof; Rinne, Juha O.; Haaparanta-Solin, Merja
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Efficacy of DYRK1A inhibitors in novel models of Down syndrome acute lymphoblastic leukemia
err2024-02-29
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errCarey-Smith, Shannon L.; Simad, Maryam H.; Panchal, Kunjal; Aya-Bonilla, Carlos; Smolders, Hannah; Lin, Sang; Armitage, Jesse D.; Nguyen, Vivien T.; Bentley, Kathryn; Ford, Jette; Singh, Sajla; Oommen, Joyce; Laurent, Anouchka P.; Mercher, Thomas; Crispino, John D.; Montgomery, Andrew P.; Kassiou, Michael; Besson, Thierry; Deau, Emmanuel; Meijer, Laurent; Cheung, Laurence C.; Kotecha, Rishi S.; Malinge, Sebastien
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Brain 11β-Hydroxysteroid Dehydrogenase Type 1 Occupancy by XanamemT Assessed by PET in Alzheimer's Disease and Cognitively Normal Individuals
err2024-01-30
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errVillemagne, Victor L.; Dore, Vincent; Chong, Lee; Kassiou, Michael; Mulligan, Rachel; Feizpour, Azadeh; Taylor, Jack; Roesner, Miriam; Miller, Tamara; Rowe, Christopher C.
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