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Synthesis, in vitro and in vivo biological evaluation of novel dual compounds targeting both acetylcholinesterase and serotonergic 5-HT4 receptors with potential interest in the treatment of Alzheimer's disease Rochais, Christophe; Lecoutey, Cedric; Lalut, Julien; Davis, Audrey; Duval, Emilie; Gaven, Florence; Largilliere, Stacy; Nee, Gerald; Corvaisier, Sophie; Santos, Jana Sopkova de Oliveira; Since, Marc; Freret, Thomas; Legrand, Romain; Callizot, Noelle; Claeysen, Sylvie; Boulouard, Michel; Dallemagne, Patrick Share Save
Towards New Anti-Inflammatory Agents: Design, Synthesis and Evaluation of Molecules Targeting XIAP-BIR2 Farag, Marc; Guedeney, Nicolas; Schwalen, Florian; Zadoroznyj, Aymeric; Barczyk, Amelie; Giret, Martin; Antraygues, Kevin; Wang, Alice; Cornu, Marie; Suzanne, Peggy; Since, Marc; Voisin-Chiret, Anne Sophie; Dubrez, Laurence; Leleu-Chavain, Natascha; Kieffer, Charline; Santos, Jana Sopkova-de Oliveira Share Save
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Synthesis of Nitrostyrylthiazolidine-2,4-dione Derivatives Displaying Antileishmanial Potential Khoumeri, Omar; Hutter, Sebastien; Primas, Nicolas; Castera-Ducros, Caroline; Carvalho, Sandra; Wyllie, Susan; Efrit, Mohamed Lotfi; Fayolle, Dimitri; Since, Marc; Vanelle, Patrice; Verhaeghe, Pierre; Azas, Nadine; El-Kashef, Hussein Share Save
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Novel thienopyrimidones targeting hepatic and erythrocytic stages of Plasmodium parasites with increased microsomal stability Lagardere, Prisca; Mustiere, Romain; Amanzougaghene, Nadia; Hutter, Sebastien; Casanova, Marion; Franetich, Jean-Francois; Tajeri, Shahin; Malzert-Freon, Aurelie; Corvaisier, Sophie; Since, Marc; Azas, Nadine; Vanelle, Patrice; Verhaeghe, Pierre; Primas, Nicolas; Mazier, Dominique; Masurier, Nicolas; Lisowski, Vincent Share Save
Design, synthesis and biological characterization of novel activators of the TrkB neurotrophin receptor Antonijevic, Mirjana; Charou, Despoina; Ramos, Isbaal; Valcarcel, Maria; Gravanis, Achille; Villace, Patricia; Callizot, Noelle; Since, Marc; Dallemagne, Patrick; Charalampopoulos, Ioannis; Rochais, Christophe Share Save
Synthesis of antiplasmodial 2-aminothieno[3,2-d]pyrimidin-4(3H)-one analogues using the scaffold hopping strategy Mustiere, Romain; Lagardere, Prisca; Hutter, Sebastien; Dell'Orco, Viviana; Amanzougaghene, Nadia; Tajeri, Shahin; Franetich, Jean-Francois; Corvaisier, Sophie; Since, Marc; Malzert-Freon, Aurelie; Masurier, Nicolas; Lisowski, Vincent; Verhaeghe, Pierre; Mazier, Dominique; Azas, Nadine; Vanelle, Patrice; Primas, Nicolas Share Save
Improving Aqueous Solubility and In Vitro Pharmacokinetic Properties of the 3-Nitroimidazo[1,2-a]pyridine Antileishmanial Pharmacophore Paoli-Lombardo, Romain; Primas, Nicolas; Bourgeade-Delmas, Sandra; Hutter, Sebastien; Sournia-Saquet, Alix; Boudot, Clotilde; Brenot, Emilie; Castera-Ducros, Caroline; Corvaisier, Sophie; Since, Marc; Malzert-Freon, Aurelie; Courtioux, Bertrand; Valentin, Alexis; Verhaeghe, Pierre; Azas, Nadine; Rathelot, Pascal; Vanelle, Patrice Share Save
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Cyclic Poly(α-peptoid)s by Lithium bis(trimethylsilyl)amide (LiHMDS)-Mediated Ring-Expansion Polymerization: Simple Access to Bioactive Backbones Salas-Ambrosio, Pedro; Tronnet, Antoine; Since, Marc; Bourgeade-Delmas, Sandra; Stigliani, Jean-Luc; Vax, Amelie; Lecommandoux, Sebastien; Dupuy, Bruno; Verhaeghe, Pierre; Bonduelle, Colin Share Save
Pleiotropic prodrugs: Design of a dual butyrylcholinesterase inhibitor and 5-HT6 receptor antagonist with therapeutic interest in Alzheimer's disease Toublet, Francois-Xavier; Lalut, Julien; Hatat, Berenice; Lecoutey, Cedric; Davis, Audrey; Since, Marc; Corvaisier, Sophie; Freret, Thomas; Santos, Jana Sopkova-de Oliveira; Claeysen, Sylvie; Boulouard, Michel; Dallemagne, Patrick; Rochais, Christophe Share Save
Antikinetoplastid SAR study in 3-nitroimidazopyridine series: Identification of a novel non-genotoxic and potent anti-T.b. brucei hitcompound with improved pharmacokinetic properties Fersing, Cyril; Boudot, Clotilde; Paoli-Lombardo, Romain; Primas, Nicolas; Pinault, Emilie; Hutter, Sebastien; Castera-Ducros, Caroline; Kabri, Youssef; Pedron, Julien; Bourgeade-Delmas, Sandra; Sournia-Saquet, Alix; Stigliani, Jean-Luc; Valentin, Alexis; Azqueta, Amaya; Muruzabal, Damian; Destere, Alexandre; Wyllie, Susan; Fairlamb, Alan H.; Corvaisier, Sophie; Since, Marc; Malzert-Freon, Aurelie; Di Giorgio, Carole; Rathelot, Pascal; Azas, Nadine; Courtioux, Bertrand; Vanelle, Patrice; Verhaeghe, Pierre Share Save
Pyridoclax-loaded nanoemulsion for enhanced anticancer effect on ovarian cancer Groo, A. C.; Hedir, S.; Since, M.; Brotin, E.; Weiswald, L. -B.; Paysant, H.; Nee, G.; Coolzaet, M.; Goux, D.; Delepee, R.; Freret, T.; Poulain, L.; Voisin-Chiret, A. S.; Malzert-Freon, A. Share Save
8-Alkynyl-3-nitroimidazopyridines display potent antitrypanosomal activity against both T. b. brucei and cruzi Fersing, Cyril; Boudot, Clotilde; Castera-Ducros, Caroline; Pinault, Emilie; Hutter, Sebastien; Paoli-Lombardo, Romain; Primas, Nicolas; Pedron, Julien; Seguy, Line; Bourgeade-Delmas, Sandra; Sournia-Saquet, Alix; Stigliani, Jean-Luc; Brossas, Jean-Yves; Paris, Luc; Valentin, Alexis; Wyllie, Susan; Fairlamb, Alan H.; Boutet-Robinet, Elisa; Corvaisier, Sophie; Since, Marc; Malzert-Freon, Aurelie; Destere, Alexandre; Mazier, Dominique; Rathelot, Pascal; Courtioux, Bertrand; Azas, Nadine; Verhaeghe, Pierre; Vanelle, Patrice Share Save
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