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Different chemical scaffolds bind to L-phe site in Mycobacterium tuberculosis Phe-tRNA synthetase Gade, Priyanka; Chang, Changsoo; Pryde, Denise S.; Fletcher, Daniel; Niven, Sarah; Magalhaes, Luma Godoy; Robinson, David; Saini, Jagmohan; Ibrahim, Peter E. G. F.; Forte, Barbara; Wower, Jacek; Bodkin, Michael J.; Baragana, Beatriz; Gilbert, Ian H.; Michalska, Karolina; Joachimiak, Andrzej Share Save
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A Structurally Diverse Compound Screening Library to Identify Substrates for Diamine, Polyamine, and Related Acetyltransferases Leiva, Hazel; De Silva, Pamela L. Caro; Painter, Ron; Le, Van Thi Bich; Uychoco, Patricia; Paniagua, Daniel Figueroa; Endres, Michael; Maltseva, Natalia; Joachimiak, Andrzej; Kuhn, Misty L. Share Save
Nα -acetyl-L-ornithine deacetylase from Escherichia coli and a ninhydrin-based assay to enable inhibitor identification (vol 12, 1415644, 2024) Kelley, Emma H.; Osipiuk, Jerzy; Korbas, Malgorzata; Endres, Michael; Bland, Alayna; Ehrman, Victoria; Joachimiak, Andrzej; Olsen, Kenneth W.; Becker, Daniel P. Share Save
Revealing reaction intermediates in one-carbon elongation by thiamine diphosphate/CoA-dependent enzyme family Kim, Youngchang; Lee, Seung Hwan; Gade, Priyanka; Nattermann, Maren; Maltseva, Natalia; Endres, Michael; Chen, Jing; Wichmann, Philipp; Hu, Yang; Marchal, Daniel G.; Yoshikuni, Yasuo; Erb, Tobias J.; Gonzalez, Ramon; Michalska, Karolina; Joachimiak, Andrzej Share Save
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Outcomes of the EMDataResource cryo-EM Ligand Modeling Challenge Lawson, Catherine L.; Kryshtafovych, Andriy; Pintilie, Grigore D.; Burley, Stephen K.; Cerny, Jiri; Chen, Vincent B.; Emsley, Paul; Gobbi, Alberto; Joachimiak, Andrzej; Noreng, Sigrid; Prisant, Michael G.; Read, Randy J.; Richardson, Jane S.; Rohou, Alexis L.; Schneider, Bohdan; Sellers, Benjamin D.; Shao, Chenghua; Sourial, Elizabeth; Williams, Chris I.; Williams, Christopher J.; Yang, Ying; Abbaraju, Venkat; Afonine, Pavel V.; Baker, Matthew L.; Bond, Paul S.; Blundell, Tom L.; Burnley, Tom; Campbell, Arthur; Cao, Renzhi; Cheng, Jianlin; Chojnowski, Grzegorz; Cowtan, K. D.; DiMaio, Frank; Esmaeeli, Reza; Giri, Nabin; Grubmueller, Helmut; Hoh, Soon Wen; Hou, Jie; Hryc, Corey F.; Hunte, Carola; Igaev, Maxim; Joseph, Agnel P.; Kao, Wei-Chun; Kihara, Daisuke; Kumar, Dilip; Lang, Lijun; Lin, Sean; Subramaniya, Sai R. Maddhuri Venkata; Mittal, Sumit; Mondal, Arup; Moriarty, Nigel W.; Muenks, Andrew; Murshudov, Garib N.; Nicholls, Robert A.; Olek, Mateusz; Palmer, Colin M.; Perez, Alberto; Pohjolainen, Emmi; Pothula, Karunakar R.; Rowley, Christopher N.; Sarkar, Daipayan; Schaefer, Luisa U.; Schlicksup, Christopher J.; Schroeder, Gunnar F.; Shekhar, Mrinal; Si, Dong; Singharoy, Abhishek; Sobolev, Oleg V.; Terashi, Genki; Vaiana, Andrea C.; Vedithi, Sundeep C.; Verburgt, Jacob; Wang, Xiao; Warshamanage, Rangana; Winn, Martyn D.; Weyand, Simone; Yamashita, Keitaro; Zhao, Minglei; Schmid, Michael F.; Berman, Helen M.; Chiu, Wah Share Save
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Native Mass Spectrometry Dissects the Structural Dynamics of an Allosteric Heterodimer of SARS-CoV-2 Nonstructural Proteins Thibert, Stephanie M.; Reid, Deseree J.; Wilson, Jesse W.; Varikoti, Rohith; Maltseva, Natalia; Schultz, Katherine J.; Kruel, Agustin; Babnigg, Gyorgy; Joachimiak, Andrzej; Kumar, Neeraj; Zhou, Mowei Share Save
Structure-based design of SARS-CoV-2 papain-like protease inhibitors Jadhav, Prakash; Huang, Bo; Osipiuk, Jerzy; Zhang, Xiaoming; Tan, Haozhou; Tesar, Christine; Endres, Michael; Jedrzejczak, Robert; Tan, Bin; Deng, Xufang; Joachimiak, Andrzej; Cai, Jianfeng; Wang, Jun Share Save
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Sel1-like proteins and peptides are the major Oxalobacter formigenes-derived factors stimulating oxalate transport by human intestinal epithelial cells Arvans, Donna; Chang, Changsoo; Alshaikh, Altayeb; Tesar, Christine; Babnigg, Gyorgy; Wolfgeher, Don; Kron, Stephen; Antonopoulos, Dionysios; Bashir, Mohamed; Cham, Candace; Musch, Mark; Chang, Eugene; Joachimiak, Andrzej; Hassan, Hatim Share Save
Dual domain recognition determines SARS-CoV-2 PLpro selectivity for human ISG15 and K48-linked di-ubiquitin Wydorski, Pawel M. M.; Osipiuk, Jerzy; Lanham, Benjamin T. T.; Tesar, Christine; Endres, Michael; Engle, Elizabeth; Jedrzejczak, Robert; Mullapudi, Vishruth; Michalska, Karolina; Fidelis, Krzysztof; Fushman, David; Joachimiak, Andrzej; Joachimiak, Lukasz A. A. Share Save
Potent and selective covalent inhibition of the papain-like protease from SARS-CoV-2 Sanders, Brian C.; Pokhrel, Suman; Labbe, Audrey D.; Mathews, Irimpan I.; Cooper, Connor J.; Davidson, Russell B.; Phillips, Gwyndalyn; Weiss, Kevin L.; Zhang, Qiu; O'Neill, Hugh; Kaur, Manat; Schmidt, Jurgen G.; Reichard, Walter; Surendranathan, Surekha; Parvathareddy, Jyothi; Phillips, Lexi; Rainville, Christopher; Sterner, David E.; Kumaran, Desigan; Andi, Babak; Babnigg, Gyorgy; Moriarty, Nigel W.; Adams, Paul D.; Joachimiak, Andrzej; Hurst, Brett L.; Kumar, Suresh; Butt, Tauseef R.; Jonsson, Colleen B.; Ferrins, Lori; Wakatsuki, Soichi; Galanie, Stephanie; Head, Martha S.; Parks, Jerry M. Share Save
Raf Kinase Inhibitory Protein Function Is Regulated via a Flexible Pocket and Novel Phosphorylation-Dependent Mechanism Granovsky, Alexey E.; Clark, Matthew C.; McElheny, Dan; Heil, Gary; Hong, Jia; Liu, Xuedong; Kim, Youngchang; Joachimiak, Grazyna; Joachimiak, Andrzej; Koide, Shohei; Rosner, Marsha Rich Share Save
A cryptic oxidoreductase safeguards oxidative protein folding in Corynebacterium diphtheriae Reardon-Robinson, Melissa E.; Nguyen, Minh Tan; Sanchez, Belkys C.; Osipiuk, Jerzy; Ruckert, Christian; Chang, Chungyu; Chen, Bo; Nagvekar, Rahul; Joachimiak, Andrzej; Tauch, Andreas; Das, Asis; Ton-That, Hung Share Save