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The Concise Guide to PHARMACOLOGY 2025/26: G protein-coupled receptors Alexander, Stephen P. H.; Davenport, Anthony P.; Kelly, Eamonn; Gibb, Alasdair J.; Mathie, Alistair A.; Peach, Chloe J.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Southan, Christopher; Davies, Jamie A.; Abbracchio, Maria Pia; Abraham, George R.; Agoulnik, Alexander; Alexander, Wayne; Al-hosaini, Khaled; Back, Magnus; Baker, Jillian G.; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Beck-Sickinger, Annette G.; Behrens, Maik; Bennett, Kirstie A.; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria A.; Bonaventure, Pascal; Boulay, Francois; Bousquet, Corinne; Brauner-Osborne, Hans; Brown, Andrew J.; Burnstock, Geoffrey; Busnelli, Marta; Calo, Girolamo; Caruso, Vanni; Castano, Justo P.; Catt, Kevin J.; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Christopoulos, Arthur; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Cox, Helen M.; Csaba, Zsolt; Dahlgren, Claes; Dautzenberg, Frank M.; Dent, Gordon; Douglas, Steven D.; Dournaud, Pascal; Dubocovich, Margarita L.; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Forsman, Huamei Fu; Fumagalli, Marta; Gainetdinov, Raul R.; Garelja, Michael L.; de Gasparo, Marc; Gbahou, Florence; Gerard, Craig; Gershengorn, Marvin; Glass, Michelle; Gloriam, David E.; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gratz, Lukas; Gregory, Karen J.; Gruber, Christian; Gundlach, Andrew L.; Hamann, Jorg; Hanson, Julien; Hartman, Deborah S.; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Heitman, Laura; Herr, Deron R.; Hollenberg, Morley D.; Holliday, Nicholas D.; Holst, Birgitte; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; IJzerman, Adriaan P.; Inagami, Tadashi; Insel, Paul A.; Jacobson, Kenneth A.; Jacobson, Laura H.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kinsolving, Julia; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Laishram, Luxmichan; Langenhan, Tobias; Langmead, Christopher J.; Larhammar, Dan; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Leurs, Rob; Li, Xaria X.; Liebscher, Ines; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet J.; Malfacini, Davide; Manning, Maurice; Marangon, Davide; Martemyanov, Kirill; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip M.; Nahon, Jean-Louis; Neubig, Richard R.; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; O'Carroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Perry-Hauser, Nicole; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Qin, Helena Chengxue; Quinn, Mark; Raffaele, Stefano; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Buzon, Alejandro Romeral; Rondard, Philippe; Rosenkilde, Mette M.; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Scholz, Nicole; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Shukla, Arun K.; Singh, Khuraijam Dhanachandra; Smith, Craig M.; Smith, Nicola J.; Staeubert, Claudia; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David M.; Thomas, Walter (Wally); Timmermans, Pieter B. M. W. M.; Tirupula, Kalyan; Toll, Lawrence; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Verbalis, Joseph G.; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Williams, Tom Lloyd; Woodruff, Trent M.; Wu, Huixian; Yang, Cheng; Yao, Chengcan; Ye, Richard D.; Zaidman, Nathan Share Save
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Characterization of [3H]AZ12464237 as a high affinity, non-nucleotide antagonist radioligand for the P2Y12 receptor Steen, E. Johanna L.; Tousiaki, Efthalia-Natalia; Kingston, Lee; van der Wildt, Berend; Lenart, Nikolett; Beaino, Wissam; Verlaan, Mariska; Zarzycka, Barbara; Zinnhardt, Bastian; Denes, Adam; Gobbi, Luca; de Esch, Iwan J. P.; Elmore, Charles S.; Windhorst, Albert D.; Honer, Michael; Leurs, Rob Share Save
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Structural visualization of small molecule recognition by CXCR3 uncovers dual-agonism in the CXCR3-CXCR7 system Saha, Shirsha; Sano, Fumiya K.; Sharma, Saloni; Ganguly, Manisankar; Dalal, Annu; Mishra, Sudha; Tiwari, Divyanshu; Akasaka, Hiroaki; Kobayashi, Takaaki A.; Roy, Nabarun; Zaidi, Nashrah; Itoh, Yuzuru; Leurs, Rob; Banerjee, Ramanuj; Shihoya, Wataru; Nureki, Osamu Share Save
Design, Synthesis and Pharmacological Characterization of the First Photoswitchable Small-Molecule Agonist for the Atypical Chemokine Receptor 3 Berenger, Sophie; Adamska, Justyna M.; Deflorian, Francesca; de Graaf, Chris; Palmer, Christie B.; Szpakowska, Martyna; Chevigne, Andy; de Esch, Iwan J. P.; Zarzycka, Barbara; Vischer, Henry F.; Wijtmans, Maikel; Leurs, Rob Share Save
Probing the Histamine H1 Receptor Binding Site to Explore Ligand Binding Kinetics Kuhne, Sebastiaan; Bosma, Reggie; Kooistra, Albert J.; Riemens, Rick; Stroet, Marc C. M.; Vischer, Henry F.; de Graaf, Chris; Wijtmans, Maikel; Leurs, Rob; de Esch, Iwan J. P. Share Save
Inhibitors of malaria parasite cyclic nucleotide phosphodiesterases block asexual blood-stage development and mosquito transmission Gomez-Gonzalez, Paula-Josefina; Gupta, Antima; Drought, Laura G.; Patel, Avnish; Okombo, John; van der Watt, Mariette; Walker-Gray, Ryan; Schindler, Kyra A.; Burkhard, Anna Y.; Yeo, Tomas; Narwal, Sunil K.; Bloxham, Talia S.; Flueck, Christian; Walker, Eloise M.; Rey, Joshua A.; Fairhurst, Kate J.; Reader, Janette; Park, Heekuk; Pollard, Harry G.; Stewart, Lindsay B.; Brandner-Garrod, Luke; Kristan, Mojca; Sterk, Geert-Jan; van Nuland, Youri M.; Manko, Emilia; van Schalkwyk, Donelly A.; Zheng, Yang; Leurs, Rob; Dechering, Koen J.; Aguiar, Anna Caroline C.; Guido, Rafael V. C.; Pereira, Dhelio B.; Tumwebaze, Patrick K.; Nosbya, Samuel L.; Rosenthal, Philip J.; Cooper, Roland A.; Palmer, Mike; Parkinson, Tanya; Burrows, Jeremy N.; Uhlemann, Anne-Catrin; Birkholtz, Lyn-Marie; Small-Saunders, Jennifer L.; Duffy, James; Fidock, David A.; Brown, Alan; Gardner, Mark; Baker, David A. Share Save
Adhesion of Crithidia fasciculata promotes a rapid change in developmental fate driven by cAMP signaling Denecke, Shane; Malfara, Madeline F.; Hodges, Kelly R.; Holmes, Nikki A.; Williams, Andre R.; Gallagher-Teske, Julia H.; Pascarella, Julia M.; Daniels, Abigail M.; Sterk, Geert Jan; Leurs, Rob; Ruthel, Gordon; Hoang, Rachel; Povelones, Megan L.; Povelones, Michael Share Save
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The Role of Water Networks in Phosphodiesterase Inhibitor Dissociation and Kinetic Selectivity Blaazer, Antoni R.; Singh, Abhimanyu K.; Zara, Lorena; Boronat, Pierre; Bautista, Lady J.; Irving, Steve; Majewski, Maciej; Barril, Xavier; Wijtmans, Maikel; Danielson, U. Helena; Sterk, Geert Jan; Leurs, Rob; van Muijlwijk-Koezen, Jacqueline E.; Brown, David G.; de Esch, Iwan J. P. Share Save
A high-affinity, cis-on photoswitchable beta blocker to optically control β2-adrenergic receptors in vitro and in vivo Shi, Shuang; Zheng, Yang; Goulding, Joelle; Marri, Silvia; Lucarini, Laura; Konecny, Benjamin; Sgambellone, Silvia; Villano, Serafina; Bosma, Reggie; Wijtmans, Maikel; Briddon, Stephen J.; Zarzycka, Barbara A.; Vischer, Henry F.; Leurs, Rob Share Save
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Structural basis of ligand recognition and design of antihistamines targeting histamine H4 receptor Xia, Ruixue; Shi, Shuang; Xu, Zhenmei; Vischer, Henry F.; Windhorst, Albert D.; Qian, Yu; Duan, Yaning; Liang, Jiale; Chen, Kai; Zhang, Anqi; Guo, Changyou; Leurs, Rob; He, Yuanzheng Share Save
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