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Philip Gribbon

Fraunhofer Institute for Translational Medicine and Pharmacology

31H-index
211Paper Count
3.6KCitation Count
Published Papers 47
Publication Date
Experimental and machine learning-based exploration of repurposed drugs reveals chemical features underlying phospholipidosis
err2026-02-06
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errMaria Kuzikov; Adelinn Kalman; Reagon Karki; Jeanette Reinshagen; Johanna Huchting; Kun Qian; Hanna Axelsson; Marianna Tampere; Päivi Östling; Brinton Seashore-Ludlow; Yojana Gadiya; Philip Gribbon; Andrea Zaliani
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2nd EUOS/SLAS Joint Challenge: Prediction of spectral properties of compounds
err2025-11-22
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errKatholiki Skopelitou; Federica Rossella; Rawdat Awuku Larbi; Philip Gribbon; Thalita Cirino; Igor V. Tetko
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The fast-dissociating D2 antagonist antipsychotic JNJ-37822681 is a neuronal Kv7 channel opener: Potential repurposing for epilepsy treatment
err2025-07-23
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errLidia Carotenuto; Oliver Keminer; Giusy Carleo; Andrea Zaliani; Antonio Leo; Rita Citraro; Giovambattista De Sarro; Nina Dirkx; Marcus Kaji; Sarah Weckhuysen; Jeanette Reinshagen; Vincenzo Barrese; Natascia Guida; Carmine Ostacolo; Francesco Miceli; Philip Gribbon; Maurizio Taglialatela
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Optimization and Evaluation of Complementary Degrader Discovery Assays for Application in Screening
err2025-07-20
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errJohanna Huchting; Arjen Weller; Moyra Schweizer; Mona Brandt; Jan Heering; Maria Kuzikov; Markus Wolf; Jeanette Reinshagen; Markus A. Queisser; Philip Gribbon; Andrea Zaliani; Ole Pless; Aimo Kannt
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Papaverine Targets STAT Signaling: A Dual-Action Therapy Option Against SARS-CoV-2
err2025-04-02
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errReus, Philipp; Torbica, Emma; Rothenburger, Tamara; Bechtel, Marco; Kandler, Joshua; Ciesek, Sandra; Gribbon, Philip; Kannt, Aimo; Cinatl, Jindrich; Bojkova, Denisa
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Predicting Antimicrobial Class Specificity of Small Molecules Using Machine Learning
err2025-02-23
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errGadiya, Yojana; Genilloud, Olga; Bilitewski, Ursula; Broenstrup, Mark; von Berlin, Leonie; Attwood, Marie; Gribbon, Philip; Zaliani, Andrea
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From library to landscape: integrative annotation workflows for compound libraries in drug repurposing
err2025-01-01
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errReinshagen, Jeanette; Seashore-Ludlow, Brinton; Gadiya, Yojana; Gustavsson, Anna-Lena; Tanoli, Ziaurrehman; Aittokallio, Tero; Huchting, Johanna; Jenmalm-Jensen, Annika; Gribbon, Philip; Zaliani, Andrea; Ballante, Flavio
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Design, quality and validation of the EU-OPENSCREEN fragment library poised to a high-throughput screening collection
err2024-01-01
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errJalencas, Xavier; Berg, Hannes; Espeland, Ludvik Olai; Sreeramulu, Sridhar; Kinnen, Franziska; Richter, Christian; Georgiou, Charis; Yadrykhinsky, Vladyslav; Specker, Edgar; Jaudzems, Kristaps; Miletic, Tanja; Harmel, Robert; Gribbon, Phil; Schwalbe, Harald; Brenk, Ruth; Jirgensons, Aigars; Zaliani, Andrea; Mestres, Jordi
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Limited high-throughput screening compatibility of the phenuivirus cap-binding domain
err2023-12-20
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errScherf, Janna; Vogel, Dominik; Gul, Sheraz; Reinshagen, Jeanette; Gribbon, Philip; Rosenthal, Maria
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Drug repurposing for the treatment of COVID-19: Targeting nafamostat to the lungs by a liposomal delivery system
err2023-12-01
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errReus, Philipp; Guthmann, Hadar; Uhlig, Nadja; Agbaria, Majd; Issmail, Leila; Eberlein, Valentina; Nordling-David, Mirjam M.; Jbara-Agbaria, Doaa; Ciesek, Sandra; Bojkova, Denisa; Cinatl, Jindrich; Burger-Kentischer, Anke; Rupp, Steffen; Zaliani, Andrea; Grunwald, Thomas; Gribbon, Philip; Kannt, Aimo; Golomb, Gershon
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Be sustainable: EOSC-Life recommendations for implementation of FAIR principles in life science data handling
err2023-11-15
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errDavid, Romain; Rybina, Arina; Burel, Jean-Marie; Heriche, Jean-Karim; Audergon, Pauline; Boiten, Jan-Willem; Coppens, Frederik; Crockett, Sara; Exter, Katrina; Fahrner, Sven; Fratelli, Maddalena; Goble, Carole; Gormanns, Philipp; Grantner, Tobias; Gruening, Bjoern; Gurwitz, Kim Tamara; Hancock, John M.; Harmse, Henriette; Holub, Petr; Juty, Nick; Karnbach, Geoffrey; Karoune, Emma; Keppler, Antje; Lancelotti, Carla; Klemeier, Jessica; Legras, Jean-Luc; Lister, Allyson L.; Longo, Dario Livio; Ludwig, Rebecca; Madon, Benedicte; Massimi, Marzia; Matser, Vera; Matteoni, Rafaele; Mayrhofer, Michaela Th; Ohmann, Christian; Panagiotopoulou, Maria; Parkinson, Helen; Perseil, Isabelle; Pfander, Claudia; Pieruschka, Roland; Raess, Michael; Rauber, Andreas; Richard, Audrey S.; Romano, Paolo; Rosato, Antonio; Sanchez-Pla, Alex; Sansone, Susanna-Assunta; Sarkans, Ugis; Serrano-Solano, Beatriz; Tang, Jing; Tanoli, Ziaurrehman; Tedds, Jonathan; Wagener, Harald; Weise, Martin; Westerhoff, Hans, V; Wittner, Rudolf; Ewbank, Jonathan; Blomberg, Niklas; Gribbon, Philip
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ADAMTS-7 Modulates Atherosclerotic Plaque Formation by Degradation of TIMP-1
err2023-09-29
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errSharifi, M. Amin; Wierer, Michael; Dang, Tan An; Milic, Jelena; Moggio, Aldo; Sachs, Nadja; von Scheidt, Moritz; Hinterdobler, Julia; Mueller, Philipp; Werner, Julia; Stiller, Barbara; Aherrahrou, Zouhair; Erdmann, Jeanette; Zaliani, Andrea; Graettinger, Mira; Reinshagen, Jeanette; Gul, Sheraz; Gribbon, Philip; Maegdefessel, Lars; Bernhagen, Juergen; Sager, Hendrik B.; Mann, Matthias; Schunkert, Heribert; Kessler, Thorsten
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Pharmacophore-Based Machine Learning Model To Predict Ligand Selectivity for E3 Ligase Binders
err2023-08-09
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errKarki, Reagon; Gadiya, Yojana; Gribbon, Philip; Zaliani, Andrea
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DHFR Inhibitors Display a Pleiotropic Anti-Viral Activity against SARS-CoV-2: Insights into the Mechanisms of Action
err2023-05-09
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errIaconis, Daniela; Caccuri, Francesca; Manelfi, Candida; Talarico, Carmine; Bugatti, Antonella; Filippini, Federica; Zani, Alberto; Novelli, Rubina; Kuzikov, Maria; Ellinger, Bernhard; Gribbon, Philip; Riecken, Kristoffer; Esposito, Francesca; Corona, Angela; Tramontano, Enzo; Beccari, Andrea Rosario; Caruso, Arnaldo; Allegretti, Marcello
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Easy access to α-ketoamides as SARS-CoV-2 and MERS Mpro inhibitors via the PADAM oxidation route
err2022-12-01
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errPelliccia, Sveva; Cerchia, Carmen; Esposito, Francesca; Cannalire, Rolando; Corona, Angela; Costanzi, Elisa; Kuzikov, Maria; Gribbon, Philip; Zaliani, Andrea; Brindisi, Margherita; Storici, Paola; Tramontano, Enzo; Summa, Vincenzo
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Comprehensive Fragment Screening of the SARS-CoV-2 Proteome Explores Novel Chemical Space for Drug Development
err2022-10-13
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errBerg, Hannes; Martin, Maria A. Wirtz; Altincekic, Nadide; Alshamleh, Islam; Bains, Jasleen Kaur; Blechar, Julius; Ceylan, Betul; de Jesus, Vanessa; Dhamotharan, Karthikeyan; Fuks, Christin; Gande, Santosh L.; Hargittay, Bruno; Hohmann, Katharina F.; Hutchison, Marie T.; Korn, Sophie Marianne; Krishnathas, Robin; Kutz, Felicitas; Linhard, Verena; Matzel, Tobias; Meiser, Nathalie; Niesteruk, Anna; Pyper, Dennis J.; Schulte, Linda; Trucks, Sven; Azzaoui, Kamal; Blommers, Marcel J. J.; Gadiya, Yojana; Karki, Reagon; Zaliani, Andrea; Gribbon, Philip; Almeida, Marcius da Silva; Anobom, Cristiane Dinis; Bula, Anna L.; Butikofer, Matthias; Caruso, Icaro Putinhon; Felli, Isabella Caterina; Da Poian, Andrea T.; de Amorim, Gisele Cardoso; Fourkiotis, Nikolaos K.; Gallo, Angelo; Ghosh, Dhiman; Gomes-Neto, Francisco; Gorbatyuk, Oksana; Hao, Bing; Kurauskas, Vilius; Lecoq, Lauriane; Li, Yunfeng; Mebus-Antunes, Nathane Cunha; Mompean, Miguel; Neves-Martins, Thais Cristtina; Ninot-Pedrosa, Marti; Pinheiro, Anderson S.; Pontoriero, Letizia; Pustovalova, Yulia; Riek, Roland; Robertson, Angus J.; Saad, Marie Jose Abi; Trevino, Miguel A.; Tsika, Aikaterini C.; Almeida, Fabio C. L.; Bax, Ad; Henzler-Wildman, Katherine; Hoch, Jeffrey C.; Jaudzems, Kristaps; Laurents, Douglas, V; Orts, Julien; Pierattelli, Roberta; Spyroulias, Georgios A.; Duchardt-Ferner, Elke; Ferner, Jan; Furtig, Boris; Hengesbach, Martin; Lohr, Frank; Qureshi, Nusrat; Richter, Christian; Saxena, Krishna; Schlundt, Andreas; Sreeramulu, Sridhar; Wacker, Anna; Weigand, Julia E.; Wirmer-Bartoschek, Julia; Wohnert, Jens; Schwalbe, Harald
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Variability of murine bacterial pneumonia models used to evaluate antimicrobial agents
err2022-09-08
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errArrazuria, Rakel; Kerscher, Bernhard; Huber, Karen E.; Hoover, Jennifer L.; Lundberg, Carina Vingsbo; Hansen, Jon Ulf; Sordello, Sylvie; Renard, Stephane; Aranzana-Climent, Vincent; Hughes, Diarmaid; Gribbon, Philip; Friberg, Lena E.; Bekeredjian-Ding, Isabelle
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Expert workshop summary: Advancing toward a standardized murine model to evaluate treatments for antimicrobial resistance lung infections
err2022-09-08
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errArrazuria, Rakel; Kerscher, Bernhard; Huber, Karen E.; Hoover, Jennifer L.; Lundberg, Carina Vingsbo; Hansen, Jon Ulf; Sordello, Sylvie; Renard, Stephane; Aranzana-Climent, Vincent; Hughes, Diarmaid; Gribbon, Philip; Friberg, Lena E.; Bekeredjian-Ding, Isabelle
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Selection of data sets for FAIRification in drug discovery and development: Which, why, and how?
err2022-08-01
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errAlharbi, Ebtisam; Gadiya, Yojana; Henderson, David; Zaliani, Andrea; Delfin-Rossaro, Alejandra; Cambon-Thomsen, Anne; Kohler, Manfred; Witt, Gesa; Welter, Danielle; Juty, Nick; Jay, Caroline; Engkvist, Ola; Goble, Carole; Reilly, Dorothy S.; Satagopam, Venkata; Ioannidis, Vassilios; Gu, Wei; Gribbon, Philip
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Drug Repurposing to Target Neuroinflammation and Sensory Neuron-Dependent Pain
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IF14.4
err2022-03-07
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errSisignano, Marco; Gribbon, Philip; Geisslinger, Gerd
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