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Pharmacological characterization of a clinical candidate, TG-0 054, a small molecule inverse agonist targeting CXCR4 Pan, Kylie S.; Wang, Ziming; Pfeil, Cy; Bergkamp, Nick D.; Mobach, Simon; Roth, Susanne; Rizk, Aurelien; Lohse, Martin J.; Annibale, Paolo; Siderius, Marco; Zimmermann, Mirjam; Smit, Martine J.; Bosma, Reggie Share Save
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Nanobody against SARS-CoV-2 non-structural protein Nsp9 inhibits viral replication in human airway epithelia Venit, Tomas; Blavier, Jeremy; Maseko, Sibusiso B.; Shu, Sam; Espada, Lilia; Breunig, Christopher; Holthoff, Hans-Peter; Desbordes, Sabrina C.; Lohse, Martin; Esposito, Gennaro; Twizere, Jean-Claude; Percipalle, Piergiorgio Share Save
ADAM19 cleaves the PTH receptor and associates with brachydactyly type E Aydin, Atakan; Klenk, Christoph; Nemec, Katarina; Isbilir, Ali; Martin, Lisa M.; Zauber, Henrik; Rrustemi, Trendelina; Toka, Hakan R.; Schuster, Herbert; Gong, Maolian; Stricker, Sigmar; Bock, Andreas; Baehring, Sylvia; Selbach, Matthias; Lohse, Martin J.; Luft, Friedrich C. Share Save
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Phosphodiesterase 3a Catalytic-domain Mutants Cause Hypertension With Brachydactyly Kayser, Charlotte; Bock, Andreas; Leeuwen, Lisette; Herkert, Johanna; Vos, Yvonne; Kidd, Alexa; Aydin, Atakan; Daumke, Oliver; Lohse, Martin; Luft, Friedrich C. Share Save
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Development of an Indole-Amide-Based Photoswitchable Cannabinoid Receptor Subtype 1 (CB1R) ?Cis-On? Agonist Rodriguez-Soacha, Diego A.; Steinmueller, Sophie A. M.; Isbilir, Ali; Fender, Julia; Deventer, Marie H.; Ramirez, Yesid A.; Tutov, Anna; Sotriffer, Christoph; Stove, Christophe P.; Lorenz, Kristina; Lohse, Martin J.; Hislop, James N.; Decker, Michael Share Save
Unraveling the hidden temporal range of fast β2-adrenergic receptor mobility by time-resolved fluorescence Balakrishnan, Ashwin; Hemmen, Katherina; Choudhury, Susobhan; Krohn, Jan-Hagen; Jansen, Kerstin; Friedrich, Mike; Beliu, Gerti; Sauer, Markus; Lohse, Martin J.; Heinze, Katrin G. Share Save
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A Versatile Sub-Nanomolar Fluorescent Ligand Enables NanoBRET Binding Studies and Single-Molecule Microscopy at the Histamine H3 Receptor Rosier, Niklas; Graetz, Lukas; Schihada, Hannes; Moeller, Jan; Isbilir, Ali; Humphrys, Laura J.; Nagl, Martin; Seibel, Ulla; Lohse, Martin J.; Pockes, Steffen Share Save
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Differences in interactions between transmembrane domains tune the activation of metabotropic glutamate receptors Thibado, Jordana K.; Tano, Jean-Yves; Lee, Joon; Salas-Estrada, Leslie; Provasi, Davide; Strauss, Alexa; Ribeiro, Joao Marcelo Lamim; Xiang, Guoqing; Broichhagen, Johannes; Filizola, Marta; Lohse, Martin J.; Levitz, Joshua Share Save
Determination of G-protein-coupled receptor oligomerization by molecular brightness analyses in single cells Isbilir, Ali; Serfling, Robert; Moeller, Jan; Thomas, Romy; De Faveri, Chiara; Zabel, Ulrike; Scarselli, Marco; Beck-Sickinger, Annette G.; Bock, Andreas; Coin, Irene; Lohse, Martin J.; Annibale, Paolo Share Save
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Advanced fluorescence microscopy reveals disruption of dynamic CXCR4 dimerization by subpocket-specific inverse agonists Isbilir, Ali; Moeller, Jan; Arimont, Marta; Bobkov, Vladimir; Perpina-Viciano, Cristina; Hoffmann, Carsten; Inoue, Asuka; Heukers, Raimond; de Graaf, Chris; Smit, Martine J.; Annibale, Paolo; Lohse, Martin J. Share Save
Establishing a sensitive fluorescence-based quantification method for cyclic nucleotides Gruteser, Nadine; Kohlhas, Viktoria; Balfanz, Sabine; Franzen, Arne; Guenther, Anne; Offenhaeusser, Andreas; Mueller, Frank; Nikolaev, Viacheslav; Lohse, Martin J.; Baumann, Arnd Share Save