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Karen S. Anderson

Yale University School of Medicine

57H-index
437Paper Count
1.4WCitation Count
Published Papers 116
Publication Date
A virtual screening strategy to repurpose antifolate compounds as W. Bancrofti DHFR inhibitors
err2025-08-12
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PREAI
errSalma Kwarteng; Jacquelyn Wilhelm; Merna Salama; Monika Salama; Klarissa Hollander; Karen S. Anderson; Nina M. Goodey; Kathleen M. Frey
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Design, fabrication, and decontamination of low-cost microfluidics for nucleic acid amplification
err2025-06-19
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errOAAI
errVi T. Nguyen; Clifford Anderson; Karen S. Anderson; Jennifer Blain Christen
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Precision projections of the delay of resistance mutations in non-small cell lung cancer via suppression of APOBEC
err2025-04-01
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errOAAI
errNousias, Orestis; Mandell, Jeffrey D.; Anderson, Karen S.; Townsend, Jeffrey P.
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Exploring Possible Drug-Resistant Variants of SARS-CoV-2 Main Protease (Mpro) with Noncovalent Preclinical Candidate, Mpro61
err2025-01-27
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errOAAI
errKenneson, Jessica R.; Papini, Christina; Tang, Su; Huynh, Kathy; Zhang, Chun-Hui; Jorgensen, William L.; Anderson, Karen S.
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Examination of the correlation between SPT and undrained shear strength: Case study of clay till in Alberta, Canada
err2024-05-01
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PREAI
errKang, Chao; Brotherton, Mark; Anderson, Karen; Semeniuk, Kevin; Mayer, Gavin; Law, Alex; Xia, Zhenyao; Zhang, Lun; Farrag, Ali; You, Jin; Abdallah, Majed
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Proof- of- concept studies with a computationally designed Mpro inhibitor as a synergistic combination regimen alternative to Paxlovid
err2024-04-15
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errOAAI
errPapini, Christina; Ullah, Irfan; Ranjan, Amalendu P.; Zhang, Shuo; Wu, Qihao; Spasov, Krasimir A.; Zhang, Chunhui; Mothes, Walther; Crawford, Jason M.; Lindenbach, Brett D.; Uchil, Pradeep D.; Kumar, Priti; Jorgensen, William L.; Anderson, Karen S.
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Covalent and noncovalent strategies for targeting Lys102 in HIV-1 reverse transcriptase
err2023-12-01
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errOAAI
errPrucha, Giavana R.; Henry, Sean; Hollander, Klarissa; Carter, Zachary J.; Spasov, Krasimir A.; Jorgensen, William L.; Anderson, Karen S.
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A High-Throughput, High-Containment Human Primary Epithelial Airway Organ-on-Chip Platform for SARS-CoV-2 Therapeutic Screening
errCELLS
IF5.2
err2023-11-16
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errOAAI
errFisher, Christine R.; Medie, Felix Mba; Luu, Rebeccah J.; Gaibler, Robert B.; Mulhern, Thomas J.; Miller, Caitlin R.; Zhang, Chelsea J.; Rubio, Logan D.; Marr, Elizabeth E.; Vijayakumar, Vidhya; Gabriel, Elizabeth P.; Quezada, Landys Lopez; Zhang, Chun-Hui; Anderson, Karen S.; Jorgensen, William L.; Alladina, Jehan W.; Medoff, Benjamin D.; Borenstein, Jeffrey T.; Gard, Ashley L.
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Noncanonical HPV carcinogenesis drives radiosensitization of head and neck tumors
err2023-07-31
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errOAAI
errSchrank, Travis P.; Kothari, Aditi; Weir, William H.; Stepp, Wesley H.; Rehmani, Hina; Liu, Xinyi; Wang, Xiaowei; Sewell, Andrew; Li, Xue; Tasoulas, Jason; Kim, Sulgi; Yarbrough, Gray; Xie, Yue; Flamand, Yael; Marur, Shanthi; Hayward, Michele C.; Wu, Di; Burtness, Barbara; Anderson, Karen S.; Baldwin, Albert S.; Yarbrough, Wendell G.; Issaeva, Natalia
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Tackling FGFR3-driven bladder cancer with a promising synergistic FGFR/HDAC targeted therapy
err2023-07-21
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errOAAI
errWang, Zechen; Muthusamy, Viswanathan; Petrylak, Daniel P.; Anderson, Karen S.
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Defining the structure-activity relationship for a novel class of allosteric MKP5 inhibitors
err2022-12-01
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errOAAI
errGannam, Zira T. K.; Jamali, Haya; Kweon, Oh Sang; Herrington, James; Shillingford, Shanelle R.; Papini, Christina; Gentzel, Erik; Lolis, Elias; Bennett, Anton M.; Ellman, Jonathan A.; Anderson, Karen S.
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Leveraging patient derived models of FGFR2 fusion positive intrahepatic cholangiocarcinoma to identify synergistic therapies
err2022-10-23
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errOAAI
errLidsky, Michael E.; Wang, Zechen; Lu, Min; Liu, Annie; Hsu, S. David; McCall, Shannon J.; Sheng, Zhecheng; Granek, Joshua A.; Owzar, Kouros; Anderson, Karen S.; Wood, Kris C.
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Structural Studies and Structure Activity Relationships for Novel Computationally Designed Non-nucleoside Inhibitors and Their Interactions With HIV-1 Reverse Transcriptase
err2022-02-14
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errOAAI
errFrey, Kathleen M.; Bertoletti, Nicole; Chan, Albert H.; Ippolito, Joseph A.; Bollini, Mariela; Spasov, Krasimir A.; Jorgensen, William L.; Anderson, Karen S.
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Optimization of Triarylpyridinone Inhibitors of the Main Protease of SARS-CoV-2 to Low-Nanomolar Antiviral Potency
err2021-07-14
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errOAAI
errZhang, Chun-Hui; Spasov, Krasimir A.; Reilly, Raquel A.; Hollander, Klarissa; Stone, Elizabeth A.; Ippolito, Joseph A.; Liosi, Maria-Elena; Deshmukh, Maya G.; Tirado-Rives, Julian; Zhang, Shuo; Liang, Zhuobin; Miller, Scott J.; Isaacs, Farren; Lindenbach, Brett D.; Anderson, Karen S.; Jorgensen, William L.
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Platelet-derived growth factor receptor beta activates Abl2 via direct binding and phosphorylation
err2021-07-01
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errOAAI
errWu, Kuanlin; Wu, Hanzhi; Lyu, Wanqing; Kim, Youngjoo; Furdui, Cristina M.; Anderson, Karen S.; Koleske, Anthony J.
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Long-acting and extended-release implant and nanoformulations with a synergistic antiretroviral two-drug combination controls HIV-1 infection in a humanized mouse model
err2021-06-26
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errOAAI
errBeloor, Jagadish; Kudalkar, Shalley N.; Buzzelli, Gina; Yang, Fan; Mandl, Hanna K.; Rajashekar, Jyothi K.; Spasov, Krasimir A.; Jorgensen, William L.; Saltzman, W. Mark; Anderson, Karen S.; Kumar, Priti
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Potent Noncovalent Inhibitors of the Main Protease of SARS-CoV-2 from Molecular Sculpting of the Drug Perampanel Guided by Free Energy Perturbation Calculations
err2021-02-22
err186
errOAAI
errZhang, Chun-Hui; Stone, Elizabeth A.; Deshmukh, Maya; Ippolito, Joseph A.; Ghahremanpour, Mohammad M.; Tirado-Rives, Julian; Spasov, Krasimir A.; Zhang, Shuo; Takeo, Yuka; Kudalkar, Shalley N.; Liang, Zhuobin; Isaacs, Farren; Lindenbach, Brett; Miller, Scott J.; Anderson, Karen S.; Jorgensen, William L.
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Covalent Inhibition of Wild-Type HIV-1 Reverse Transcriptase Using a Fluorosulfate Warhead
err2021-01-06
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errOAAI
errIppolito, Joseph A.; Niu, Haichan; Bertoletti, Nicole; Carter, Zachary J.; Jin, Shengyan; Spasov, Krasimir A.; Cisneros, Jose A.; Valhondo, Margarita; Cutrona, Kara J.; Anderson, Karen S.; Jorgensen, William L.
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Identification of 14 Known Drugs as Inhibitors of the Main Protease of SARS-CoV-2
err2020-10-25
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errOAAI
errGhahremanpour, Mohammad M.; Tirado-Rives, Julian; Deshmukh, Maya; Ippolito, Joseph A.; Zhang, Chun-Hui; de Vaca, Israel Cabeza; Liosi, Maria-Elena; Anderson, Karen S.; Jorgensen, William L.
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