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Yongying Jiang

The University of Texas MD Anderson Cancer Center

22H-index
102Paper Count
2.8KCitation Count
Published Papers 40
Publication Date
DCAF11-dependent molecular glue degrader activated by glutathionylation
errNature
IF48.5
err2026-08-05
err0
errOAAI
errHojong Yoon; Franziska Wachter; Katharine A. Barrett; Cyrus Jin; Anna Rodríguez-Pöhnlein; Justine C. Rutter; Ryan J. Lumpkin; Rebecca J. Metivier; Katherine A. Donovan; Kheewoong Baek; Yongying Jiang; Minwoo Lee; Robert W. Kalis; Jianwei Che; Yuan Xiong; Eric S. Fischer; Benjamin L. Ebert
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Structure-Guided Development of NRAS G12D Inhibitors Based on a 5-Azaindole Core
err2026-01-22
err0
PREAI
errJoshua B. Cox; Vinay Nair; Pijus Mandal; Naphtali Reyna; Tuyen Tran; Lisa Maria Mustachio; Jennifer Bardenhagen; Janelle Fawver; Hannah Shepard; Anna M. Hickey; Qi Wu; Christian Rodriguez; Fei Yu; Phuc Phan; Andrea J. Mendiola; Rebecca Johnson; Roopa Thapar; Troy Johnson; Yongying Jiang; Jason B. Cross; Mary K. Geck Do; Philip Jones; Joseph Marsalek; Timothy Heffernan; Michael J. Soth; Edith Nagy
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Nivolumab plus ipilimumab induce hyper-progression in renal medullary carcinoma: results of a phase II trial and preclinical evidence
err2025-11-25
err0
errOAAI
errMelinda Soeung; Xinmiao Yan; Ciro Zanca; Jing Qian; Menuka Karki; Fei Duan; Hania Khan; Li Zhang; David H. Peng; Mariah Williams; Rong He; Ziheng Chen; Luigi Perelli; Jianfeng Chen; Rebecca S. Tidwell; Pankaj K. Chauhan; Courtney N. Le; Truong N. A. Lam; Nirjar Bhattacharya; Rutvi Shah; I-Lin Ho; Jason P. Gay; Caroline C. Carrillo; Ningping Feng; Kang Le; Guang Gao; Teresa L. Perry; Faika Mseeh; Yongying Jiang; Quanyun A. Xu; Niki Marie Zacharias; Rahul A. Sheth; Tharakeswara K. Bathala; Priya Rao; Najat C. Daw; Durga N. Tripathi; Cheryl L. Walker; Mohammad M. Mohammad; Jianhua Zhang; Guangchun Han; Yanshuo Chu; Ruiping Wang; Minghao Dang; Enyu Dai; Fuduan Peng; Yunhe Liu; Akshaya Jadhav; Wenhua Lang; Claudio A. Arrechedera; Leticia Campos Clemente; Edwin R. Parra; Hsinyi Lu; Cara L. Haymaker; Ignacio I. Wistuba; Andrew Futreal; Andrea Viale; Michael J. Soth; Philip Jones; Joseph R. Marszalek; Timothy Heffernan; Giulio F. Draetta; Nizar M. Tannir; Jianjun Gao; Linghua Wang; Giannicola Genovese; Pavlos Msaouel
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Allosteric targeting of RIPK1: discovery of novel inhibitors via parallel virtual screening and structure-guided optimization
err2025-09-27
err0
PREAI
errR. S. K. Vijayan; Matthew M. Hamilton; Dana E. Pfaffinger; Fernando G. Alvarez; Naphtali J. Reyna; Jennifer P. Bardenhagen; Hannah Shepard; Christian Rodriguez; Sunil Goodwani; Yaima Lightfoot; Klaus Maskos; Sven Johannsson; Georg Kempf; Quanyun Alan Xu; Lars Neumann; Yongying Jiang; Mary Geck Do; Philip Jones; Richard T. Lewis; William J. Ray; Jason B. Cross
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Discovery of Novel, Potent, and Orally Bioavailable SMARCA2 Proteolysis-Targeting Chimeras with Synergistic Antitumor Activity in Combination with Kirsten Rat Sarcoma Viral Oncogene Homologue G12C Inhibitors
err2025-04-25
err0
PREAI
errKotagiri, Sasikumar; Wang, Yawen; Han, Yanyan; Liang, Xiaobing; Blazanin, Nicholas; Mazhar, Hira; Sebastian, Manu; Nguyen, Phuong Kieu; Jiang, Yongying; Lissanu, Yonathan
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Discovery of ART0380, a Potent and Selective ATR Kinase Inhibitor Undergoing Phase 2 Clinical Studies for the Treatment of Advanced or Metastatic Solid Cancers
err2024-12-04
err0
PREAI
errCarroll, Christopher L.; Johnson, Michael G.; Ding, Yanbing; Kang, Zhijun; Vijayan, R. S. K.; Bardenhagen, Jennifer P.; Fang, Cheng; Lapointe, David; Li, Meng; Liu, Chiu-Yi; Lv, Xiaobing; Ma, Xiaoyan; Pang, Jihai; Shepard, Hannah E.; Suarez, Catalina; Yau, Anne Ju; Williams, Christopher C.; Wu, Qi; Heald, Robert A.; Robinson, Helen M. R.; Smith, Graeme C. M.; Cross, Jason B.; Do, Mary K. Geck; Jiang, Yongying; Lively, Sarah; Yap, Timothy A.; Giuliani, Virginia; Heffernan, Timothy; Jones, Philip; Di Francesco, M. Emilia
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IACS-16559, a CBP/P300 bromodomain inhibitor for the treatment of specific AML subsets
err2024-03-22
err0
PREAI
errZanca, Ciro; Soth, Michael; Gao, Guang; Gay, Jason; Feng, Ningping; Bristow, Christopher; Le, Kang; Xu, Quanyun; Phuong Nguyen; Jiang, Yongying; Perry, Teresa; Mseeh, Faika; Leonard, Paul; Cross, Jason; Giuliani, Virginia; Marszalek, Joe; Jones, Philip; Heffernan, Tim
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Apolipoprotein A-I Binding Protein Inhibits the Formation of Infantile Hemangioma through Cholesterol-Regulated Hypoxia-Inducible Factor 1a Activation
err2024-03-01
err1
PREAI
errJiang, Yongying; Li, Xingjuan; Liu, Qin; Lei, Gongyun; Wu, Changyue; Chen, Long; Hu, Yinsyae; Xian, Hua; Mao, Renfang
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Discovery of IACS-52825, a Potent and Selective DLK Inhibitor for Treatment of Chemotherapy-Induced Peripheral Neuropathy
err2023-07-12
err9
PREAI
errLe, Kang; Soth, Michael J. J.; Cross, Jason B. B.; Liu, Gang; Ray, William J. J.; Ma, Jiacheng; Goodwani, Sunil G. G.; Acton, Paul J. J.; Buggia-Prevot, Virginie; Akkermans, Onno; Barker, John; Conner, Michael L. L.; Jiang, Yongying; Liu, Zhen; McEwan, Paul; Warner-Schmidt, Jennifer; Xu, Alan; Zebisch, Matthias; Heijnen, Cobi J. J.; Abrahams, Brett; Jones, Philip
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Markov Transition Field Enhanced Deep Domain Adaptation Network for Milling Tool Condition Monitoring
err2022-05-31
err14
errOAAI
errSun, Wei; Zhou, Jie; Sun, Bintao; Zhou, Yuqing; Jiang, Yongying
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The generation of PD-L1 and PD-L2 in cancer cells: From nuclear chromatin reorganization to extracellular presentation
err2022-03-01
err52
errOAAI
errFan, Zhiwei; Wu, Changyue; Chen, Miaomiao; Jiang, Yongying; Wu, Yuanyuan; Mao, Renfang; Fan, Yihui
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Discovery of 6-[(3S,4S)-4-Amino-3-methyl-2-oxa-8-azaspiro[4.5]decan-8-yl]-3-(2,3-dichlorophenyl)-2-methyl-3,4-dihydropyrimidin-4-one (IACS-15414), a Potent and Orally Bioavailable SHP2 Inhibitor
err2021-10-13
err23
PREAI
errCzako, Barbara; Sun, Yuting; McAfoos, Timothy; Cross, Jason B.; Leonard, Paul G.; Burke, Jason P.; Carroll, Christopher L.; Feng, Ningping; Harris, Angela L.; Jiang, Yongying; Kang, Zhijun; Kovacs, Jeffrey J.; Mandal, Pijus; Meyers, Brooke A.; Mseeh, Faika; Parker, Connor A.; Yu, Simon S.; Williams, Christopher C.; Wu, Qi; Di Francesco, Maria Emilia; Draetta, Giulio; Heffernan, Timothy; Marszalek, Joseph R.; Kohl, Nancy E.; Jones, Philip
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Stability of MRI contrast agents in high-energy radiation of a 1.5T MR-Linac
err2021-08-01
err12
errOAAI
errWang, Jihong; Salzillo, Travis; Jiang, Yongying; Mackeyev, Yuri; Fuller, Clifton David; Chung, Caroline; Choi, Seungtaek; Hughes, Neil; Ding, Yao; Yang, Jinzhong; Vedam, Sastry; Krishnan, Sunil
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Discovery of IACS-9779 and IACS-70465 as Potent Inhibitors Targeting Indoleamine 2,3-Dioxygenase 1 (IDO1) Apoenzyme
err2021-07-22
err17
PREAI
errHamilton, Matthew M.; Mseeh, Faika; McAfoos, Timothy J.; Leonard, Paul G.; Reyna, Naphtali J.; Harris, Angela L.; Xu, Alan; Han, Michelle; Soth, Michael J.; Czako, Barbara; Theroff, Jay P.; Mandal, Pijus K.; Burke, Jason P.; Virgin-Downey, Brett; Petrocchi, Alessia; Pfaffinger, Dana; Rogers, Norma E.; Parker, Connor A.; Yu, Simon S.; Jiang, Yongying; Krapp, Stephan; Lammens, Alfred; Trevitt, Graham; Tremblay, Martin R.; Mikule, Keith; Wilcoxen, Keith; Cross, Jason B.; Jones, Philip; Marszalek, Joseph R.; Lewis, Richard T.
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Inhibition of dual leucine zipper kinase prevents chemotherapy-induced peripheral neuropathy and cognitive impairments
errPAIN
IF5.5
err2021-04-15
err16
errOAAI
errMa, Jiacheng; Goodwani, Sunil; Acton, Paul J.; Buggia-Prevot, Virginie; Kesler, Shelli R.; Jamal, Imran; Mahant, Iteeben D.; Liu, Zhen; Mseeh, Faika; Roth, Bruce L.; Chakraborty, Chaitali; Peng, Bo; Wu, Qi; Jiang, Yongying; Le, Kang; Soth, Michael J.; Jones, Philip; Kavelaars, Annemieke; Ray, William J.; Heijnen, Cobi J.
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An enolase inhibitor for the targeted treatment of ENO1-deleted cancers (vol 2, pg 1413, 2020)
err2020-12-18
err0
errOAAI
errLin, Yu-Hsi; Satani, Nikunj; Hammoudi, Naima; Yan, Victoria C.; Barekatain, Yasaman; Khadka, Sunada; Ackroyd, Jeffrey J.; Georgiou, Dimitra K.; Pham, Cong-Dat; Arthur, Kenisha; Maxwell, David; Peng, Zhenghong; Leonard, Paul G.; Czako, Barbara; Pisaneschi, Federica; Mandal, Pijus; Sun, Yuting; Zielinski, Rafal; Pando, Susana Castro; Wang, Xiaobo; Tran, Theresa; Xu, Quanyu; Wu, Qi; Jiang, Yongying; Kang, Zhijun; Asara, John M.; Priebe, Waldemar; Bornmann, William; Marszalek, Joseph R.; DePinho, Ronald A.; Muller, Florian L.
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Allosteric SHP2 Inhibitor, IACS-13909, Overcomes EGFR-Dependent and EGFR-Independent Resistance Mechanisms toward Osimertinib
err2020-11-03
err62
errOAAI
errSun, Yuting; Meyers, Brooke A.; Czako, Barbara; Leonard, Paul; Mseeh, Faika; Harris, Angela L.; Wu, Qi; Johnson, Sarah; Parker, Connor A.; Cross, Jason B.; Di Francesco, Maria Emilia; Bivona, Benjamin J.; Bristow, Christopher A.; Burke, Jason P.; Carrillo, Caroline C.; Carroll, Christopher L.; Chang, Qing; Feng, Ningping; Gao, Guang; Gera, Sonal; Giuliani, Virginia; Huang, Justin K.; Jiang, Yongying; Kang, Zhijun; Kovacs, Jeffrey J.; Liu, Chiu-Yi; Lopez, Anastasia M.; Ma, Xiaoyan; Mandal, Pijus K.; McAfoos, Timothy; Miller, Meredith A.; Mullinax, Robert A.; Peoples, Michael; Ramamoorthy, Vandhana; Seth, Sahil; Spencer, Nakia D.; Suzuki, Erika; Williams, Christopher C.; Yu, Simon S.; Zuniga, Andy M.; Draetta, Giulio F.; Marszalek, Joseph R.; Heffernan, Timothy P.; Kohl, Nancy E.; Jones, Philip
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Discovery of IPN60090, a Clinical Stage Selective Glutaminase-1 (GLS-1) Inhibitor with Excellent Pharmacokinetic and Physicochemical Properties
err2020-10-29
err62
errOAAI
errSoth, Michael J.; Le, Kang; Di Francesco, Maria Emilia; Hamilton, Matthew M.; Liu, Gang; Burke, Jason P.; Carroll, Chris L.; Kovacs, Jeffrey J.; Bardenhagen, Jennifer P.; Bristow, Christopher A.; Cardozo, Mario; Czako, Barbara; de Stanchina, Elisa; Feng, Ningping; Garvey, Jill R.; Gay, Jason P.; Do, Mary K. Geck; Greer, Jennifer; Han, Michelle; Harris, Angela; Herrera, Zachary; Huang, Sha; Giuliani, Virginia; Jiang, Yongying; Johnson, Sarah B.; Johnson, Troy A.; Kang, Zhijun; Leonard, Paul G.; Liu, Zhen; McAfoos, Timothy; Miller, Meredith; Morlacchi, Pietro; Mullinax, Robert A.; Palmer, Wylie S.; Pang, Jihai; Rogers, Norma; Rudin, Charles M.; Shepard, Hannah E.; Spencer, Nakia D.; Theroff, Jay; Wu, Qi; Xu, Alan; Yau, Ju Anne; Draetta, Giulio; Toniatti, Carlo; Heffernan, Timothy P.; Jones, Philip
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Discovery of IACS-9439, a Potent, Exquisitely Selective, and Orally Bioavailable Inhibitor of CSF1R
err2020-07-29
err13
PREAI
errCzako, Barbara; Marszalek, Joseph. R.; Burke, Jason P.; Mandal, Pijus; Leonard, Paul G.; Cross, Jason B.; Mseeh, Faika; Jiang, Yongying; Chang, Edward Q.; Suzuki, Erika; Kovacs, Jeffrey J.; Feng, Ningping; Gera, Sonal; Harris, Angela L.; Liu, Zhen; Mullinax, Robert A.; Pang, Jihai; Parker, Connor A.; Spencer, Nakia D.; Yu, Simon S.; Wu, Qi; Tremblay, Martin R.; Mikule, Keith; Wilcoxen, Keith; Heffernan, Timothy P.; Draetta, Giulio F.; Jones, Philip
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