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Florence I. Raynaud

The Institute of Cancer Research

75H-index
773Paper Count
1.9WCitation Count
Published Papers 162
Publication Date
Elucidating molecularly stratified single agent, and combination, therapeutic strategies targeting MCL1 for lethal prostate cancer
err2025-10-08
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errJuan M. Jiménez-Vacas; Daniel Westaby; Ines Figueiredo; Alexis De Haven Brandon; Ana Padilha; Wei Yuan; George Seed; Denisa Bogdan; Bora Gurel; Claudia Bertan; Susana Miranda; Maryou Lambros; Antonio J. Montero-Hidalgo; Ilsa Coleman; Ivan Pak Lok Yu; Lorenzo Buroni; Wanting Zeng; Antje J. Neeb; Jon Welti; Jan Rekowski; Roberta Paravati; Florian Gabel; Nicole Pandell; Ana Ferreira; Mateus Crespo; Ruth Riisnaes; Souvik Das; Joe Taylor; Nick Waldron; Emily Hobern; Melanie Valenti; Jian Ning; Ilona Bernett; Kate Liodaki; Thomas Persse; Patricia Galipeau; Scott Wilkinson; Shana Y. Trostel; Fatima Karzai; Cindy H. Chau; Erica L. Beatson; Xiaohu Zhang; Carleen Klumpp-Thomas; Andreas Varkaris; Raul M. Luque; Amanda Swain; Florence Raynaud; Nathan A. Lack; Craig J. Thomas; Gavin Ha; William D. Figg; Marco Bezzi; Adam G. Sowalsky; Peter S. Nelson; Suzanne Carreira; Steven P. Balk; Johann S. de Bono; Adam Sharp
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Exposing 24-hour cycles in bile acids of male humans
err2024-11-19
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errBello, Adesola T.; Sarafian, Magali H.; Wimborne, Elizabeth A.; Middleton, Benita; Revell, Victoria L.; Raynaud, Florence I.; Chowdhury, Namrata R.; van der Veen, Daan R.; Skene, Debra J.
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A NOVEL ROLE FOR ACVR1/ALK2 IN REGULATING CHOLESTEROL BIOSYNTHESIS PROVIDES A NEW COMBINATORIAL THERAPEUTIC APPROACH FOR PATIENTS WITH DMG
err2024-06-18
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errRogers, Rebecca; Grabovaska, Yura; Mackay, Alan; Carvalho, Diana; Dobinson, Claire; Pereira, Rita; Sejdiu, Drenusha; Burford, Anna; Molinari, Valeria; Ruddle, Ruth; Raynaud, Florence; Chew, Nicole; Tsui, Vanessa; Sun, Claire; Firestein, Ron; Jones, Chris
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Discovery of ARID1A loss as a patient biomarker for NXP800-A developmental activator of the integrated stress response (ISR) and inhibitor of the HSF1 pathway in ovarian cancer
err2024-03-22
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PREAI
errte Poele, Robert H.; Powers, Marissa; Sharp, Swee; de Billy, Emmanuel; Taskinen, Maria; Pellegrino, Loredana; Gowan, Sharon; Miah, Asadh; Hayes, Angela; Cheeseman, Matthew; Jones, Keith; Eccles, Suzanne; Raynaud, Florence; Clarke, Paul; Workman, Paul
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Activation of the integrated stress response by NXP800, an orally available, clinical-stage, investigational agent in ARID1A-mutated, platinum resistant ovarian cancer
err2024-03-04
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PREAI
errPowers, Marissa V.; Swap, Swee Y.; te Poele, Robert; Lampraki, Eirini-Maria; Roe, Toby; Pellegrino, Loredana; Taskinen, Maria; Eccles, Suzenne; Raynaud, Florence; Cheeseman, Matthew; Jones, Keith; Clarke, Paul A.; Workman, Paul
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Design, Synthesis, and Evaluation of Inhibitors of Hedgehog Acyltransferase
err2024-01-10
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errRitzefeld, Markus; Zhang, Leran; Xiao, Zhangping; Andrei, Sebastian A.; Boyd, Olivia; Masumoto, Naoko; Rodgers, Ursula R.; Artelsmair, Markus; Sefer, Lea; Hayes, Angela; Gavriil, Efthymios-Spyridon; Raynaud, Florence I.; Burke, Rosemary; Blagg, Julian; Rzepa, Henry S.; Siebold, Christian; Magee, Anthony I.; Lanyon-Hogg, Thomas; Tate, Edward W.
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Results of a phase 1 dose escalation clinical trial of NXP800, a novel GCN2 activator, in patients with advanced or metastatic solid tumors
err2023-12-01
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PREAI
errBanerji, Udai; Pacey, Simon; Finkelstein, Karen; Rodney, Simon; DosReis, Ana Filipa Palma; Codaccipisanelli, Giovanni; Sloan, Mark; Raynaud, Florence I.; Ruddle, Ruth; Swales, Karen; Tall, Matthew; Shemesh, Shay; Marsolini, Diane; Sardone, Megan; Hay, Justin; Bliss, Robin; Poradosu, Enrique; Workman, Paul
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A CONNECT CONSORTIUM PRECLINICAL STUDY IDENTIFIES MEK INHIBITION AND RADIATION AS POTENTIAL COMBINATION PARTNERS FOR THE ALK2 INHIBITOR TP-0184 IN ACVR1-MUTANT DMG
err2023-06-12
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errRogers, Rebecca; Tsoli, Maria; Kumar, Shiva Senthil; Potente, Elisabet Fernandez; Biery, Matt; Grabovska, Yura; Mackay, Alan; Carvalho, Diana; Pereria, Rita; Burford, Anna; Sejdiu, Drenusha; Ruddle, Ruth; Gabel, Florian; Raynaud, Florence; Yadavilli, Sridevi; Mizoguchi, Sean; Subramaniam, Bavani; Kilburn, Lindsey; Hwang, Eugene; Nazarian, Javad; Vitanza, Nicholas; Ziegler, David; Drissi, Rachid; Jones, Chris
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Machine learning estimation of human body time using metabolomic profiling
err2023-04-24
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errWoelders, Tom; Revell, Victoria L.; Middleton, Benita; Ackermann, Katrin; Kayser, Manfred; Raynaud, Florence I.; Skene, Debra J.; Hut, Roelof A.
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Activation of the integrated stress response by the developmental HSF1 pathway inhibitor NXP800
err2023-04-14
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PREAI
errPowers, Marissa V.; Sharp, Swee Y.; Lampraki, Eirini-Maria; Roe, Toby; Pellegrino, Loredana; Taskinen, Maria; Poele, Robert Te; Raynaud, Florence; Eccles, Suzanne; Cheeseman, Matthew; Jones, Keith; Clarke, Paul A.; Workman, Paul
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Discovery of an In Vivo Chemical Probe for BCL6 Inhibition by Optimization of Tricyclic Quinolinones
err2023-04-07
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errHarnden, Alice C.; Davis, Owen A.; Box, Gary M.; Hayes, Angela; Johnson, Louise D.; Henley, Alan T.; Brandon, Alexis K. de Haven; Valenti, Melanie; Cheung, Kwai-Ming J.; Brennan, Alfie; Huckvale, Rosemary; Pierrat, Olivier A.; Talbot, Rachel; Bright, Michael D.; Akpinar, Hafize Aysin; Miller, Daniel S. J.; Tarantino, Dalia; Gowan, Sharon; de Klerk, Selby; McAndrew, Peter Craig; Le Bihan, Yann-Vai; Meniconi, Mirco; Burke, Rosemary; Kirkin, Vladimir; van Montfort, Rob L. M.; Raynaud, Florence I.; Rossanese, Olivia W.; Bellenie, Benjamin R.; Hoelder, Swen
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HSF1 Pathway Inhibitor Clinical Candidate (CCT361814/NXP800) Developed from a Phenotypic Screen as a Potential Treatment for Refractory Ovarian Cancer and Other Malignancies
err2023-04-05
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errPasqua, A. Elisa; Sharp, Swee Y.; Chessum, Nicola E. A.; Hayes, Angela; Pellegrino, Loredana; Tucker, Michael J.; Miah, Asadh; Wilding, Birgit; Evans, Lindsay E.; Rye, Carl S.; Mok, N. Yi; Liu, Manjuan; Henley, Alan T.; Gowan, Sharon; De Billy, Emmanuel; te Poele, Robert; Powers, Marissa; Eccles, Suzanne A.; Clarke, Paul A.; Raynaud, Florence I.; Workman, Paul; Jones, Keith; Cheeseman, Matthew D.
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Discovering cell-active BCL6 inhibitors: effectively combining biochemical HTS with multiple biophysical techniques, X-ray crystallography and cell-based assays
err2022-11-03
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errPierrat, Olivier A.; Liu, Manjuan; Collie, Gavin W.; Shetty, Kartika; Rodrigues, Matthew J.; Le Bihan, Yann-Vai; Gunnell, Emma A.; McAndrew, P. Craig; Stubbs, Mark; Rowlands, Martin G.; Yahya, Norhakim; Shehu, Erald; Talbot, Rachel; Pickard, Lisa; Bellenie, Benjamin R.; Cheung, Kwai-Ming J.; Drouin, Ludovic; Innocenti, Paolo; Woodward, Hannah; Davis, Owen A.; Lloyd, Matthew G.; Varela, Ana; Huckvale, Rosemary; Broccatelli, Fabio; Carter, Michael; Galiwango, David; Hayes, Angela; Raynaud, Florence, I; Bryant, Christopher; Whittaker, Steven; Rossanese, Olivia W.; Hoelder, Swen; Burke, Rosemary; van Montfort, Rob L. M.
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Intracellular Metabolomics Identifies Efflux Transporter Inhibitors in a Routine Caco-2 Cell Permeability Assay-Biological Implications
errCELLS
IF5.2
err2022-10-19
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errNaseem, Afia; Pal, Akos; Gowan, Sharon; Asad, Yasmin; Donovan, Adam; Temesszentandrasi-Ambrus, Csilla; Kis, Emese; Gaborik, Zsuzsanna; Bhalay, Gurdip; Raynaud, Florence
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A phase (Ph) I/II trial of the CXCR2 antagonist AZD5069 in combination with enzalutamide (ENZA) in patients (pts) with metastatic castration resistant prostate cancer (mCRPC)
err2022-09-01
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errGuo, C.; Sharp, A.; Vogl, U.; Colombo, I.; Stathis, A.; Jain, S.; Chandran, K.; Tiu, C.; Paschalis, A.; Matthews, R. E.; Figueiredo, I.; Rekowski, J.; Yap, C.; de la Maza, M. de los Dolores Fenor; Turner, A.; Badham, H. C.; Parmar, M.; Raynaud, F.; Alimonti, A.; de Bono, J. S.
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A Phase I Trial of CT900, a Novel a-Folate Receptor- Mediated Thymidylate Synthase Inhibitor, in Patients with Solid Tumors with Expansion Cohorts in Patients with High-Grade Serous Ovarian Cancer
err2022-08-19
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errBanerjee, Susana; Michalarea, Vasiliki; Ang, Joo Ern; Garces, Alvaro Ingles; Biondo, Andrea; Funingana, Ionut-Gabriel; Little, Martin; Ruddle, Ruth; Raynaud, Florence; Riisnaes, Ruth; Gurel, Bora; Chua, Sue; Tunariu, Nina; Porter, Joanna C.; Prout, Toby; Parmar, Mona; Zachariou, Anna; Turner, Alison; Jenkins, Ben; McIntosh, Stuart; Ainscow, Ed; Minchom, Anna; Lopez, Juanita; de Bono, Johann; Jones, Robert; Hall, Emma; Cook, Natalie; Basu, Bristi; Banerji, Udai
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Optimizing Shape Complementarity Enables the Discovery of Potent Tricyclic BCL6 Inhibitors
err2022-06-03
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errDavis, Owen A.; Cheung, Kwai-Ming J.; Brennan, Alfie; Lloyd, Matthew G.; Rodrigues, Matthew J.; Pierrat, Olivier A.; Collie, Gavin W.; Le Bihan, Yann-Vai; Huckvale, Rosemary; Harnden, Alice C.; Varela, Ana; Bright, Michael D.; Eve, Paul; Hayes, Angela; Henley, Alan T.; Carter, Michael D.; McAndrew, P. Craig; Talbot, Rachel; Burke, Rosemary; van Montfort, Rob L. M.; Raynaud, Florence, I; Rossanese, Olivia W.; Meniconi, Mirco; Bellenie, Benjamin R.; Hoelder, Swen
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Improved Binding Affinity and Pharmacokinetics Enable Sustained Degradation of BCL6 In Vivo
err2022-06-02
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errHuckvale, Rosemary; Harnden, Alice C.; Cheung, Kwai-Ming J.; Pierrat, Olivier A.; Talbot, Rachel; Box, Gary M.; Henley, Alan T.; Brandon, Alexis K. de Haven; Hallsworth, Albert E.; Bright, Michael D.; Akpinar, Hafize Aysin; Miller, Daniel S. J.; Tarantino, Dalia; Gowan, Sharon; Hayes, Angela; Gunnell, Emma A.; Brennan, Alfie; Davis, Owen A.; Johnson, Louise D.; de Klerk, Selby; McAndrew, Craig; Le Bihan, Yann-Vai; Meniconi, Mirco; Burke, Rosemary; Kirkin, Vladimir; van Montfort, Rob L. M.; Raynaud, Florence I.; Rossanese, Olivia W.; Bellenie, Benjamin R.; Hoelder, Swen
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Individualized Prediction of Drug Response and Rational Combination Therapy in NSCLC Using Artificial Intelligence-Enabled Studies of Acute Phosphoproteomic Changes
err2022-04-03
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errCoker, Elizabeth A.; Stewart, Adam; Ozer, Bugra; Minchom, Anna; Pickard, Lisa; Ruddle, Ruth; Carreira, Suzanne; Popat, Sanjay; O'Brien, Mary; Raynaud, Florence; de Bono, Johann; Al-Lazikani, Bissan; Banerji, Udai
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Presence of human breast cancer xenograft changes the diurnal profile of amino acids in mice
err2022-01-19
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errPaula, Rubens, Jr.; Sonehara, Nathalia Martins; Jardim-Perassi, Bruna Victorasso; Pal, Akos; Asad, Yasmin; Almeida Chuffa, Luiz Gustavo; Chammas, Roger; Raynaud, Florence I.; Zuccari, Debora A. P. C.
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