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Thoughts for the future Alkhalaf, Lona M.; Arrowsmith, Cheryl; Balskus, Emily P.; Bergamini, Giovanna; Bhandari, Rashna; Chang, Christopher J.; Chen, Peng; Chen, Xing; Ciulli, Alessio; Cricco, Julia A.; Davis, Benjamin G.; Delbianco, Martina; Dudareva, Natalia; Dueber, Erin; Ferguson, Fleur; de Giuseppe, Priscila Oliveira; Hamachi, Itaru; Hammond, Ming Chen; Hatzios, Stavroula K.; Do Heo, Won; Janet, Jon Paul; Kamat, Siddhesh S.; Knapp, Stefan; Krishnan, Yamuna; Lang, Kathrin; Laraia, Luca; Leveson-Gower, Reuben B.; Li, Xiang David; Liu, David R.; Liu, Mo-Fang; London, Nir; Mahanta, Nilkamal; Mayor-Ruiz, Cristina; Muir, Tom; Murakami, Mario Tyago; Rhee, Hyun-Woo; Robers, Matt; Satz, Alex; Schulman, Brenda A.; Shen, Ben; Shoichet, Brian; Strauss, Erick; Suzuki, Tsutomu; Tiwary, Pratyush; Waldmann, Herbert; Ward, Thomas R.; Weeks, Amy; Weerapana, Eranthie; Winter, Georg Share Save
Dual targeting of histone deacetylases and MYC as potential treatment strategy for H3-K27M pediatric gliomas Algranati, Danielle; Oren, Roni; Dassa, Bareket; Fellus-Alyagor, Liat; Plotnikov, Alexander; Barr, Haim; Harmelin, Alon; London, Nir; Ron, Guy; Furth, Noa; Shema, Efrat Share Save
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Turning high-throughput structural biology into predictive inhibitor design Saar, Kadi L.; McCorkindale, William; Fearon, Daren; Boby, Melissa; Barr, Haim; Ben-Shmuel, Amir; London, Nir; von Delft, Frank; Chodera, John D.; Lee, Alpha A.; COVID Moonshot, Alpha A. Share Save
Sulfamate Acetamides as Self-Immolative Electrophiles for Covalent Ligand-Directed Release Chemistry Reddi, Rambabu N.; Rogel, Adi; Gabizon, Ronen; Rawale, Dattatraya Gautam; Harish, Battu; Marom, Shir; Tivon, Barr; Arbel, Yamit Shorer; Gurwicz, Neta; Oren, Roni; David, Keren; Liu, Jingjing; Duberstein, Shirly; Itkin, Maxim; Malitsky, Sergey; Barr, Haim; Katz, Ben-Zion; Herishanu, Yair; Shachar, Idit; Shulman, Ziv; London, Nir Share Save
Azapeptide activity-based probes for the SARS-CoV-2 main protease enable visualization of inhibition in infected cells Vanhoutte, Roeland; Barniol-Xicota, Marta; Chiu, Winston; Vangeel, Laura; Jochmans, Dirk; De Jonghe, Steven; Zidane, Hadeer; Barr, Haim M.; London, Nir; Neyts, Johan; Verhelst, Steven H. L. Share Save
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Optimization of Covalent MKK7 Inhibitors via Crude Nanomole- Scale Libraries Gehrtz, Paul; Marom, Shir; Buehrmann, Mike; Hardick, Julia; Kleinboelting, Silke; Shraga, Amit; Dubiella, Christian; Gabizon, Ronen; Wiese, Jan N.; Mueller, Matthias P.; Cohen, Galit; Babaev, Ilana; Shurrush, Khriesto; Avram, Liat; Resnick, Efrat; Barr, Haim; Rauh, Daniel; London, Nir Share Save
Expanding the Repertoire of Low-Molecular-Weight Pentafluorosulfanyl-Substituted Scaffolds Jose, Arathy; Guest, Daniel; LeGay, Remi; Tizzard, Graham J.; Coles, Simon J.; Derveni, Mariliza; Wright, Edward; Marrison, Lester; Lee, Alpha A.; Morris, Aaron; Robinson, Matt; von Delft, Frank; Fearon, Daren; Koekemoer, Lizbe; Matviuk, Tetiana; Aimon, Anthony; Schofield, Christopher J.; Malla, Tika R.; London, Nir; Greenland, Barnaby W.; Bagley, Mark C.; Spencer, John Share Save
Structure-guided design and characterization of a clickable, covalent PARP16 inhibitor Bejan, Daniel S.; Sundalam, Sunil; Jin, Haihong; Morgan, Rory K.; Kirby, Ilsa T.; Siordia, Ivan R.; Tivon, Barr; London, Nir; Cohen, Michael S. Share Save
An automatic pipeline for the design of irreversible derivatives identifies a potent SARS-CoV-2 Mpro inhibitor Zaidman, Daniel; Gehrtz, Paul; Filep, Mihajlo; Fearon, Daren; Gabizon, Ronen; Douangamath, Alice; Prilusky, Jaime; Duberstein, Shirly; Cohen, Galit; Owen, C. David; Resnick, Efrat; Strain-Damerell, Claire; Lukacik, Petra; Barr, Haim; Walsh, Martin A.; von Delft, Frank; London, Nir Share Save
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PDBe-KB: collaboratively defining the biological context of structural data Varadi, Mihaly; Anyango, Stephen; Armstrong, David; Berrisford, John; Choudhary, Preeti; Deshpande, Mandar; Nadzirin, Nurul; Nair, Sreenath S.; Pravda, Lukas; Tanweer, Ahsan; Al-Lazikani, Bissan; Andreini, Claudia; Barton, Geoffrey J.; Bednar, David; Berka, Karel; Blundell, Tom; Brock, Kelly P.; Maria Carazo, Jose; Damborsky, Jiri; David, Alessia; Dey, Sucharita; Dunbrack, Roland; Fernandez Recio, Juan; Fraternali, Franca; Gibson, Toby; Helmer-Citterich, Manuela; Hoksza, David; Hopf, Thomas; Jakubec, David; Kannan, Natarajan; Krivak, Radoslav; Kumar, Manjeet; Levy, Emmanuel D.; London, Nir; Macias, Jose Ramon; Srivatsan, Madhusudhan M.; Marks, Debora S.; Martens, Lennart; McGowan, Stuart A.; McGreig, Jake E.; Modi, Vivek; Gonzalo Parra, R.; Pepe, Gerardo; Piovesan, Damiano; Prilusky, Jaime; Putignano, Valeria; Radusky, Leandro G.; Ramasamy, Pathmanaban; Rausch, Atilio O.; Reuter, Nathalie; Rodriguez, Luis A.; Rollins, Nathan J.; Rosato, Antonio; Serrano, Luis; Singh, Gulzar; Skoda, Petr; Sorzano, Carlos Oscar S.; Stourac, Jan; Sulkowska, Joanna, I; Svobodova, Radka; Tichshenko, Natalia; Tosatto, Silvio C. E.; Vranken, Wim; Wass, Mark N.; Xue, Dandan; Zaidman, Daniel; Thornton, Janet; Sternberg, Michael; Orengo, Christine; Velankar, Sameer Share Save
Cross-reactive antibodies against human coronaviruses and the animal coronavirome suggest diagnostics for future zoonotic spillovers Klompus, Shelley; Leviatan, Sigal; Vogl, Thomas; Mazor, Roei D.; Kalka, Iris N.; Stoler-Barak, Liat; Nathan, Nachum; Peres, Ayelet; Moss, Lihee; Godneva, Anastasia; Ben Tikva, Sharon Kagan; Shinar, Eilat; Cohen-Dvashi, Hadas; Gabizon, Ronen; London, Nir; Diskin, Ron; Yaari, Gur; Weinberger, Adina; Shulman, Ziv; Segal, Eran Share Save