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Nir London

the weizmann institute of science

42H-index
288Paper Count
8.4KCitation Count
Published Papers 66
Publication Date
Targeted Protein Degradation of NUDT5 Dissociates Catalytic Inhibition from Protein Loss in 6-Thioguanine Response
err2026-06-30
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errAnne-Sophie M. C. Marques; Ludwig G. Bauer; Tuan-Anh Nguyen; Alejandro Gonzalez Orta; Jan-Lennart Venne; Carol Cheng; Esra Balıkçı; Yusi Liu; Barr Tivon; Alena Kroupova; Alessio Ciulli; Nir London; Stefan Kubicek; Kilian V. M. Huber
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α-Halothioamide warheads with enhanced cysteine reactivity and specificity for covalent protein labelling
err2026-05-14
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errOAAI
errLászló Petri; Ronen Gabizon; Nikolett Péczka; Péter Ábrányi-Balogh; József Simon; Tímea Imre; György G. Ferenczy; Nir London; György M. Keserű
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Discovery of Covalent Ligands with AlphaFold3
err2026-03-19
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errOAAI
errYoav Shamir; Ronen Gabizon; Adi Rogel; David Yin-wei Lin; Amy H. Andreotti; Nir London
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A pharmacological modality to sequester homomeric proteins
err2026-02-05
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errElla Livnah; Ohad Suss; Adi Rogel; Atar Gilat; Yuval Abdan; José A. Villegas; Ronen Gabizon; Almog Nadir; Yoav Shamir; Noam Y. Steinman; Barr Tivon; Shira Albeck; Tamar Unger; Ofra Golani; Inna Goliand; Nadav Elad; Silvia Carvalho; Khriesto Shurrush; Haim Barr; David Margulies; Emmanuel D. Levy; Nir London
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Thoughts for the future
err2024-12-24
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PREAI
errAlkhalaf, Lona M.; Arrowsmith, Cheryl; Balskus, Emily P.; Bergamini, Giovanna; Bhandari, Rashna; Chang, Christopher J.; Chen, Peng; Chen, Xing; Ciulli, Alessio; Cricco, Julia A.; Davis, Benjamin G.; Delbianco, Martina; Dudareva, Natalia; Dueber, Erin; Ferguson, Fleur; de Giuseppe, Priscila Oliveira; Hamachi, Itaru; Hammond, Ming Chen; Hatzios, Stavroula K.; Do Heo, Won; Janet, Jon Paul; Kamat, Siddhesh S.; Knapp, Stefan; Krishnan, Yamuna; Lang, Kathrin; Laraia, Luca; Leveson-Gower, Reuben B.; Li, Xiang David; Liu, David R.; Liu, Mo-Fang; London, Nir; Mahanta, Nilkamal; Mayor-Ruiz, Cristina; Muir, Tom; Murakami, Mario Tyago; Rhee, Hyun-Woo; Robers, Matt; Satz, Alex; Schulman, Brenda A.; Shen, Ben; Shoichet, Brian; Strauss, Erick; Suzuki, Tsutomu; Tiwary, Pratyush; Waldmann, Herbert; Ward, Thomas R.; Weeks, Amy; Weerapana, Eranthie; Winter, Georg
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Dual targeting of histone deacetylases and MYC as potential treatment strategy for H3-K27M pediatric gliomas
err2024-08-02
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errOAAI
errAlgranati, Danielle; Oren, Roni; Dassa, Bareket; Fellus-Alyagor, Liat; Plotnikov, Alexander; Barr, Haim; Harmelin, Alon; London, Nir; Ron, Guy; Furth, Noa; Shema, Efrat
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Deconvoluting low yield from weak potency in direct-to-biology workflows with machine learning
err2024-01-01
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errOAAI
errMccorkindale, William; Filep, Mihajlo; London, Nir; Lee, Alpha A.; King-Smith, Emma
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A simple method for developing lysine targeted covalent protein reagents
err2023-12-01
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errGabizon, Ronen; Tivon, Barr; Reddi, Rambabu N.; van den Oetelaar, Maxime C. M.; Amartely, Hadar; Cossar, Peter J.; Ottmann, Christian; London, Nir
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Turning high-throughput structural biology into predictive inhibitor design
err2023-03-06
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errSaar, Kadi L.; McCorkindale, William; Fearon, Daren; Boby, Melissa; Barr, Haim; Ben-Shmuel, Amir; London, Nir; von Delft, Frank; Chodera, John D.; Lee, Alpha A.; COVID Moonshot, Alpha A.
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Sulfamate Acetamides as Self-Immolative Electrophiles for Covalent Ligand-Directed Release Chemistry
err2023-02-04
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errReddi, Rambabu N.; Rogel, Adi; Gabizon, Ronen; Rawale, Dattatraya Gautam; Harish, Battu; Marom, Shir; Tivon, Barr; Arbel, Yamit Shorer; Gurwicz, Neta; Oren, Roni; David, Keren; Liu, Jingjing; Duberstein, Shirly; Itkin, Maxim; Malitsky, Sergey; Barr, Haim; Katz, Ben-Zion; Herishanu, Yair; Shachar, Idit; Shulman, Ziv; London, Nir
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Azapeptide activity-based probes for the SARS-CoV-2 main protease enable visualization of inhibition in infected cells
err2023-01-01
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errOAAI
errVanhoutte, Roeland; Barniol-Xicota, Marta; Chiu, Winston; Vangeel, Laura; Jochmans, Dirk; De Jonghe, Steven; Zidane, Hadeer; Barr, Haim M.; London, Nir; Neyts, Johan; Verhelst, Steven H. L.
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Kidney Failure Alters Parathyroid Pin1 Phosphorylation and Parathyroid Hormone mRNA-Binding Proteins Leading to Secondary Hyperparathyroidism
err2022-09-01
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errHassan, Alia; Pollak, Yael E. E.; Kilav-Levin, Rachel; Silver, Justin; London, Nir; Nechama, Morris; Ben-Dov, Iddo Z. Z.; Naveh-Many, Tally
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Optimization of Covalent MKK7 Inhibitors via Crude Nanomole- Scale Libraries
err2022-07-30
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errOAAI
errGehrtz, Paul; Marom, Shir; Buehrmann, Mike; Hardick, Julia; Kleinboelting, Silke; Shraga, Amit; Dubiella, Christian; Gabizon, Ronen; Wiese, Jan N.; Mueller, Matthias P.; Cohen, Galit; Babaev, Ilana; Shurrush, Khriesto; Avram, Liat; Resnick, Efrat; Barr, Haim; Rauh, Daniel; London, Nir
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Expanding the Repertoire of Low-Molecular-Weight Pentafluorosulfanyl-Substituted Scaffolds
err2022-02-22
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errOAAI
errJose, Arathy; Guest, Daniel; LeGay, Remi; Tizzard, Graham J.; Coles, Simon J.; Derveni, Mariliza; Wright, Edward; Marrison, Lester; Lee, Alpha A.; Morris, Aaron; Robinson, Matt; von Delft, Frank; Fearon, Daren; Koekemoer, Lizbe; Matviuk, Tetiana; Aimon, Anthony; Schofield, Christopher J.; Malla, Tika R.; London, Nir; Greenland, Barnaby W.; Bagley, Mark C.; Spencer, John
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Structure-guided design and characterization of a clickable, covalent PARP16 inhibitor
err2022-01-01
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errBejan, Daniel S.; Sundalam, Sunil; Jin, Haihong; Morgan, Rory K.; Kirby, Ilsa T.; Siordia, Ivan R.; Tivon, Barr; London, Nir; Cohen, Michael S.
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An automatic pipeline for the design of irreversible derivatives identifies a potent SARS-CoV-2 Mpro inhibitor
err2021-12-01
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errZaidman, Daniel; Gehrtz, Paul; Filep, Mihajlo; Fearon, Daren; Gabizon, Ronen; Douangamath, Alice; Prilusky, Jaime; Duberstein, Shirly; Cohen, Galit; Owen, C. David; Resnick, Efrat; Strain-Damerell, Claire; Lukacik, Petra; Barr, Haim; Walsh, Martin A.; von Delft, Frank; London, Nir
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Site-Specific Labeling of Endogenous Proteins Using CoLDR Chemistry
err2021-11-24
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errReddi, Rambabu N.; Rogel, Adi; Resnick, Efrat; Gabizon, Ronen; Prasad, Pragati Kishore; Gurwicz, Neta; Barr, Haim; Shulman, Ziv; London, Nir
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PDBe-KB: collaboratively defining the biological context of structural data
err2021-11-10
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errVaradi, Mihaly; Anyango, Stephen; Armstrong, David; Berrisford, John; Choudhary, Preeti; Deshpande, Mandar; Nadzirin, Nurul; Nair, Sreenath S.; Pravda, Lukas; Tanweer, Ahsan; Al-Lazikani, Bissan; Andreini, Claudia; Barton, Geoffrey J.; Bednar, David; Berka, Karel; Blundell, Tom; Brock, Kelly P.; Maria Carazo, Jose; Damborsky, Jiri; David, Alessia; Dey, Sucharita; Dunbrack, Roland; Fernandez Recio, Juan; Fraternali, Franca; Gibson, Toby; Helmer-Citterich, Manuela; Hoksza, David; Hopf, Thomas; Jakubec, David; Kannan, Natarajan; Krivak, Radoslav; Kumar, Manjeet; Levy, Emmanuel D.; London, Nir; Macias, Jose Ramon; Srivatsan, Madhusudhan M.; Marks, Debora S.; Martens, Lennart; McGowan, Stuart A.; McGreig, Jake E.; Modi, Vivek; Gonzalo Parra, R.; Pepe, Gerardo; Piovesan, Damiano; Prilusky, Jaime; Putignano, Valeria; Radusky, Leandro G.; Ramasamy, Pathmanaban; Rausch, Atilio O.; Reuter, Nathalie; Rodriguez, Luis A.; Rollins, Nathan J.; Rosato, Antonio; Serrano, Luis; Singh, Gulzar; Skoda, Petr; Sorzano, Carlos Oscar S.; Stourac, Jan; Sulkowska, Joanna, I; Svobodova, Radka; Tichshenko, Natalia; Tosatto, Silvio C. E.; Vranken, Wim; Wass, Mark N.; Xue, Dandan; Zaidman, Daniel; Thornton, Janet; Sternberg, Michael; Orengo, Christine; Velankar, Sameer
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Cross-reactive antibodies against human coronaviruses and the animal coronavirome suggest diagnostics for future zoonotic spillovers
err2021-07-29
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errKlompus, Shelley; Leviatan, Sigal; Vogl, Thomas; Mazor, Roei D.; Kalka, Iris N.; Stoler-Barak, Liat; Nathan, Nachum; Peres, Ayelet; Moss, Lihee; Godneva, Anastasia; Ben Tikva, Sharon Kagan; Shinar, Eilat; Cohen-Dvashi, Hadas; Gabizon, Ronen; London, Nir; Diskin, Ron; Yaari, Gur; Weinberger, Adina; Shulman, Ziv; Segal, Eran
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