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Photoswitchable COX-2-Selective Inhibitors as Light-Regulated Anti-Inflammatory Agents 光开关COX-2选择性抑制剂作为光调控抗炎剂 Morales, Amanda; Cruz, Alejandro; Perez-Sanchez, Alex; D'Avino, Danilo; Galassi, Gaia; Milano, Erica Ginevra; Bernareggi, Irene; Arenos-Bach, Carla; Grazioso, Giovanni; Alibes, Ramon; Hernando, Jordi; Gorostiza, Pau; Rossi, Antonietta; Pistocchi, Anna; Matera, Carlo; Busque, Felix; Gonzalez-Lafont, Angels; Lluch, Jose M. 分享 收藏
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Design, Synthesis, and Biological Characterization of Macromolecular Ester Prodrugs of a Selective Cyclooxygenase-2 Inhibitor 选择性环氧化酶-2抑制剂的大分子酯前药的设计、合成与生物特性研究 Saletti, Mario; Paolino, Marco; Venditti, Jacopo; Giuliani, Germano; Rossi, Antonietta; D'avino, Danilo; Perna, Sara; Varfaj, Ina; Sardella, Roccaldo; Macchiarulo, Antonio; Maramai, Samuele; Lamponi, Stefania; Cappelli, Andrea; Anzini, Maurizio 分享 收藏
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Sex hormone deprivation abolishes sex-specific differences in murine colon inflammation and related lipid mediator production Pace, Simona; Meyer, Katharina Paula Lydia; Troisi, Fabiana; Bilancia, Rossella; D'Avino, Danilo; Parisi, Olga; Rizza, Roberta; Stiuso, Paola; Gerstmeier, Jana; Schaedel, Patrick; Ialenti, Armando; Sautebin, Lidia; Serhan, Charles N.; Rossi, Antonietta; Borrelli, Francesca; Werz, Oliver 分享 收藏
Cannabidiol acts as molecular switch in innate immune cells to promote the biosynthesis of inflammation-resolving lipid mediators Peltner, Lukas K.; Gluthmann, Lars; Borner, Friedemann; Pace, Simona; Hoffstetter, Robert K.; Kretzer, Christian; Bilancia, Rosella; Pollastro, Federica; Koeberle, Andreas; Appendino, Giovanni; Rossi, Antonietta; Newcomer, Marcia E.; Gilbert, Nathaniel C.; Werz, Oliver; Jordan, Paul M. 分享 收藏
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Design, Synthesis, and Pharmacological Characterization of a Potent Soluble Epoxide Hydrolase Inhibitor for the Treatment of Acute Pancreatitis Musella, Simona; D'Avino, Danilo; Peltner, Lukas Klaus; Di Sarno, Veronica; Cerqua, Ida; Merciai, Fabrizio; Vestuto, Vincenzo; Ciaglia, Tania; Smaldone, Gerardina; Di Matteo, Francesca; Di Micco, Simone; Napolitano, Valeria; Bifulco, Giuseppe; Pepe, Giacomo; Sommella, Eduardo Maria; Basilicata, Manuela Giovanna; Aquino, Giovanna; Gomez-Monterrey, Isabel M. M.; Campiglia, Pietro; Ostacolo, Carmine; Roviezzo, Fiorentina; Werz, Oliver; Rossi, Antonietta; Bertamino, Alessia 分享 收藏
Highly potent and selective 5-lipoxygenase inhibition by new, simple heteroaryl-substituted catechols for treatment of inflammation Krauth, Verena; Bruno, Ferdinando; Pace, Simona; Jordan, Paul M.; Temml, Veronika; Romano, Maria Preziosa; Khan, Haroon; Schuster, Daniela; Rossi, Antonietta; Filosa, Rosanna; Werz, Oliver 分享 收藏
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In Vitro Bioaccessibility and Anti-Inflammatory Activity of a Chemically Characterized Allium cepa L. Extract Rich in Quercetin Derivatives Optimized by the Design of Experiments Ullah, Hammad; Di Minno, Alessandro; Santarcangelo, Cristina; Tantipongpiradet, Ariyawan; Dacrema, Marco; di Matteo, Rita; El-Seedi, Hesham R.; Khalifa, Shaden A. M.; Baldi, Alessandra; Rossi, Antonietta; Daglia, Maria 分享 收藏
Discovery and Optimization of Indoline-Based Compounds as Dual 5-LOX/sEH Inhibitors: In Vitro and In Vivo Anti-Inflammatory Characterization Cerqua, Ida; Musella, Simona; Peltner, Lukas Klaus; D'Avino, Danilo; Di Sarno, Veronica; Granato, Elisabetta; Vestuto, Vincenzo; Di Matteo, Rita; Pace, Simona; Ciaglia, Tania; Bilancia, Rossella; Smaldone, Gerardina; Di Matteo, Francesca; Di Micco, Simone; Bifulco, Giuseppe; Pepe, Giacomo; Basilicata, Manuela Giovanna; Rodriquez, Manuela; Gomez-Monterrey, Isabel M.; Campiglia, Pietro; Ostacolo, Carmine; Roviezzo, Fiorentina; Werz, Oliver; Rossi, Antonietta; Bertamino, Alessia 分享 收藏
Novel analgesic/anti-inflammatory agents: 1,5-Diarylpyrrole nitrooxyethyl sulfides and related compounds as Cyclooxygenase-2 inhibitors containing a nitric oxide donor moiety endowed with vasorelaxant properties 新型镇痛/抗炎剂: 1,5-二芳基吡咯硝基氧乙基硫化物和相关化合物作为Cyclooxygenase-2抑制剂,含有具有血管舒张特性的一氧化氮供体部分 Saletti, Mario; Maramai, Samuele; Reale, Annalisa; Paolino, Marco; Brogi, Simone; Di Capua, Angela; Cappelli, Andrea; Giorgi, Gianluca; D'Avino, Danilo; Rossi, Antonietta; Ghelardini, Carla; Mannelli, Lorenzo Di Cesare; Sardella, Roccaldo; Carotti, Andrea; Woelkart, Gerald; Klosch, Burkhard; Bigogno, Chiara; Dondio, Giulio; Anzini, Maurizio 分享 收藏
A vitamin E long-chain metabolite and the inspired drug candidate a-amplexichromanol relieve asthma features in an experimental model of allergen sensitization Cerqua, Ida; Neukirch, Konstantin; Terlizzi, Michela; Granato, Elisabetta; Caiazzo, Elisabetta; Cicala, Carla; Ialenti, Armando; Capasso, Raffaele; Werz, Oliver; Sorrentino, Rosalinda; Seraphin, Denis; Helesbeux, Jean-Jacques; Cirino, Giuseppe; Koeberle, Andreas; Roviezzo, Fiorentina; Rossi, Antonietta 分享 收藏
Hydroethanolic Extract of Prunus domestica L.: Metabolite Profiling and In Vitro Modulation of Molecular Mechanisms Associated to Cardiometabolic Diseases Ullah, Hammad; Sommella, Eduardo; Santarcangelo, Cristina; D'Avino, Danilo; Rossi, Antonietta; Dacrema, Marco; Di Minno, Alessandro; Di Matteo, Giacomo; Mannina, Luisa; Campiglia, Pietro; Magni, Paolo; Daglia, Maria 分享 收藏
Ethoxy acetalated dextran-based nanocarriers accomplish efficient inhibition of leukotriene formation by a novel FLAP antagonist in human leukocytes and blood 基于乙氧基缩醛化葡聚糖的纳米载体通过新型FLAP拮抗剂在人白细胞和血液中有效抑制白三烯的形成 Kretzer, Christian; Shkodra, Blerina; Klemm, Paul; Jordan, Paul M.; Schroeder, Daniel; Cinar, Gizem; Vollrath, Antje; Schubert, Stephanie; Nischang, Ivo; Hoeppener, Stephanie; Stumpf, Steffi; Banoglu, Erden; Gladigau, Frederike; Bilancia, Rossella; Rossi, Antonietta; Eggeling, Christian; Neugebauer, Ute; Schubert, Ulrich S.; Werz, Oliver 分享 收藏